Target Details
| UniProt AC | P07947 |
|---|---|
| Gene Symbol | YES1 |
| Protein Name | Tyrosine-protein kinase Yes |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 158
- Clinical molecules 54
- Avg pChEMBL 7.39
KEGG Pathways (1)
Active Molecules (158)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JSFCZQSJQXFJDS
|
9.4 | IC50 | 4 | — | |
AQSSMEORRLJZLU
|
9.3 | IC50 | 34 | Yes | |
ZBNZXTGUTAYRHI
|
9.3 | Kd | 102 | Yes | |
SIUNALDMRGZQBR
|
9.2 | IC50 | 3 | — | |
BNRXMSGHPVYSDK
|
9.1 | IC50 | 24 | — | |
SSDFTYWIYVWCIE
|
9.1 | IC50 | 17 | — | |
PHXJVRSECIGDHY
|
9.1 | IC50 | 59 | — | |
SFCBIFOAGRZJNX
|
9.0 | Kd | 22 | — | |
YHVHYWYQEFELOW
|
9.0 | IC50 | 44 | — | |
NCDVMWSJHOBWBM
|
8.9 | IC50 | 3 | — | |
YJSFAHMGDRBZGH
|
8.9 | IC50 | 16 | Yes | |
QOVBTXBRBQUBBP
|
8.9 | IC50 | 3 | — | |
VCIZYTQJDGPPDJ
|
8.9 | IC50 | 6 | — | |
ZBRROTSBDAODQD
|
8.9 | IC50 | 7 | Yes | |
VRCBGBBYFHLJRE
|
8.7 | IC50 | 5 | — | |
WFRLFWGASBLYTC
|
8.7 | IC50 | 15 | Yes | |
ZCWXCBKGPJOAFQ
|
8.7 | IC50 | 13 | — | |
IWODHENDABKBRB
|
8.6 | IC50 | 6 | — | |
VAARYSWULJUGST
|
8.6 | Kd | 119 | Yes | |
WVXNSAVVKYZVOE
|
8.6 | IC50 | 92 | — | |
FIHAXQZQWYILHF
|
8.6 | IC50 | 2 | — | |
HLILQABBLFGERM
|
8.5 | IC50 | 6 | Yes | |
DYHVAHJSHIYCLL
|
8.5 | IC50 | 4 | — | |
DEUUCYCGMWGKGM
|
8.4 | IC50 | 2 | — | |
OUKYUETWWIPKQR
|
8.4 | IC50 | 31 | Yes | |
UBPYILGKFZZVDX
|
8.4 | Kd | 130 | Yes | |
VAWLAPYBUJTXRS
|
8.4 | IC50 | 6 | Yes | |
HKSZLNNOFSGOKW
|
8.4 | IC50 | 408 | — | |
OLGSVSPNJXGSAD
|
8.3 | IC50 | 5 | Yes | |
KSUDUUBCXJUFRL
|
8.3 | Kd | 12 | — | |
DNLQIFRJOZJGCU
|
8.3 | IC50 | 6 | Yes | |
URNMUIDFWOJTPW
|
8.2 | Ki | 7 | Yes | |
LCYSSHSIKSARGO
|
8.2 | IC50 | 19 | — | |
XYFPWWZEPKGCCK
|
8.2 | IC50 | 34 | — | |
BOQLSYBMPFBUNE
|
8.1 | IC50 | 4 | — | |
LRRYSZJODUIJIM
|
8.1 | IC50 | 2 | — | |
BPMIILWVKNVIKR
|
8.0 | IC50 | 6 | Yes | |
DHSWXTYFLRUXKS
|
8.0 | IC50 | 6 | Yes | |
KNRLVDRDQDJIMP
|
8.0 | IC50 | 4 | Yes | |
SKMKVAWCYDFONZ
|
8.0 | IC50 | 5 | Yes | |
USKFMBYPIMKTAD
|
8.0 | IC50 | 6 | Yes | |
VJHWNDGPWFUUKL
|
8.0 | IC50 | 6 | Yes | |
WWSWQMMEPXHAON
|
8.0 | IC50 | 6 | Yes | |
OTTCBLPTHPBEEX
|
8.0 | IC50 | 11 | Yes | |
LBVKEEFIPBQIMD
|
8.0 | IC50 | 4 | — | |
SRSQULBCTWSVKL
|
7.9 | IC50 | 15 | — | |
ZVIWALRWYYSHSU
|
7.9 | IC50 | 3 | — | |
OONFNUWBHFSNBT
|
7.8 | IC50 | 11 | — | |
NDUAHACMVSARNG
|
7.7 | IC50 | 4 | — | |
YYLKKYCXAOBSRM
|
7.7 | Kd | 191 | — |