Target Details
| UniProt AC | P07858 |
|---|---|
| Gene Symbol | CTSB |
| Protein Name | Cathepsin B |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00112 (Peptidase_C1) PF08127 (Propeptide_C1) |
Summary
- Multi-target molecules 494
- Clinical molecules 10
- Avg pChEMBL 7.05
KEGG Pathways (6)
Associated Diseases (2)
Active Molecules (494)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZDJKOPMEVPPKBM
|
6.5 | IC50 | 2 | — | |
BTSVYYFWIQTHSO
|
6.5 | IC50 | 2 | — | |
YBJGTORHNOALQH
|
6.5 | IC50 | 2 | — | |
ZKSDUCXACMZPEQ
|
6.5 | IC50 | 2 | — | |
ZZPFZJXGGZUTHR
|
6.5 | IC50 | 4 | — | |
ABCDOWZVJWRRMY
|
6.5 | Ki | 3 | — | |
BXTKCAQATANWLJ
|
6.5 | Ki | 2 | — | |
CJFRYKIQLJALCT
|
6.5 | IC50 | 4 | — | |
HEINWAWHFFDZOZ
|
6.5 | IC50 | 2 | — | |
SLSHNBKPDGBYGO
|
6.5 | IC50 | 3 | — | |
GGWWZSKHPHUDIG
|
6.5 | IC50 | 4 | — | |
OKCRMEZBXWRMEQ
|
6.5 | Ki | 3 | — | |
PACZTXUZEYVPIY
|
6.5 | IC50 | 3 | — | |
XWPMWIRSEUHFET
|
6.5 | Ki | 3 | — | |
WWVOULFEIOXZLF
|
6.5 | IC50 | 4 | — | |
FMQLLJJKTLJHMC
|
6.4 | IC50 | 4 | — | |
YTOZVAMWOLDKNH
|
6.4 | IC50 | 2 | — | |
CZZWUFZBGQIPTE
|
6.4 | Ki | 2 | — | |
LGVMUCFKYMVFOU
|
6.4 | IC50 | 2 | — | |
VIFRNMGMIPTJQJ
|
6.4 | IC50 | 2 | — | |
AZNDDHOZPWLFFK
|
6.4 | Ki | 2 | — | |
OLIMBXKACVCIMM
|
6.4 | IC50 | 3 | — | |
OLIMBXKACVCIMM
|
6.4 | IC50 | 3 | — | |
SACCVMQJINSDGD
|
6.4 | IC50 | 2 | — | |
UULSCOLFHVNVPK
|
6.4 | IC50 | 4 | — | |
VQYXNZIEKJIVRK
|
6.4 | IC50 | 2 | — | |
VQYXNZIEKJIVRK
|
6.4 | IC50 | 2 | — | |
RHJLQMVZXQKJKB
|
6.4 | Ki | 5 | — | |
RHJLQMVZXQKJKB
|
6.4 | Ki | 5 | — | |
XJEBMYGPXQJVFF
|
6.4 | IC50 | 3 | — | |
ZGJILAJMKMDGOC
|
6.4 | IC50 | 4 | — | |
AWOGCPXUTJBQEG
|
6.4 | IC50 | 3 | Yes | |
CABJFQPQQUDNAL
|
6.4 | IC50 | 3 | — | |
KTRQMFTUNYZEES
|
6.4 | IC50 | 2 | — | |
LHEWOPPODOUFHU
|
6.4 | IC50 | 4 | — | |
LLEYFYXOCVQUBI
|
6.4 | IC50 | 6 | — | |
OKEXQFAOCJQYST
|
6.4 | IC50 | 2 | — | |
GJLXFFKSGIYTBC
|
6.4 | IC50 | 2 | — | |
VCZZEMKHLLGOGU
|
6.4 | IC50 | 2 | — | |
MQRWKSMRQVMZEN
|
6.4 | IC50 | 4 | — | |
BIEDNGLUYFVOFK
|
6.4 | Ki | 3 | — | |
GCILXAGICVRZQV
|
6.4 | IC50 | 4 | — | |
TWOOZSOQPIWDLA
|
6.4 | IC50 | 3 | — | |
YAGNDONYTVCOFN
|
6.4 | IC50 | 3 | — | |
FMLMGLVVGNKBJT
|
6.4 | IC50 | 2 | — | |
FRACLEVIDYQZNB
|
6.4 | Ki | 3 | — | |
JPQIXMPQVCDFBY
|
6.4 | Ki | 5 | — | |
MRFFFLZDQYKPHZ
|
6.4 | IC50 | 4 | — | |
UPCGYFVYJJCJTE
|
6.4 | IC50 | 4 | — | |
XGOULJOKRIZKRT
|
6.4 | Ki | 3 | — |