Target Details
| UniProt AC | P07858 |
|---|---|
| Gene Symbol | CTSB |
| Protein Name | Cathepsin B |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00112 (Peptidase_C1) PF08127 (Propeptide_C1) |
Summary
- Multi-target molecules 494
- Clinical molecules 10
- Avg pChEMBL 7.05
KEGG Pathways (6)
Associated Diseases (2)
Active Molecules (494)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RSEOJELKUSEFQD
|
6.9 | IC50 | 4 | — | |
DAQZLXYFNHPPBP
|
6.8 | Ki | 3 | — | |
JRFCJBAMIBGKTB
|
6.8 | IC50 | 4 | — | |
LMWXYUHYSBCVJI
|
6.8 | Ki | 3 | — | |
OQVJUAAFCYLUII
|
6.8 | IC50 | 4 | — | |
YJYSHOADPNSQGD
|
6.8 | IC50 | 4 | — | |
HEIHTFALJDNKRT
|
6.8 | IC50 | 4 | — | |
POELQXXPKHMGFF
|
6.8 | IC50 | 7 | — | |
BLJKFTVYZPTNBP
|
6.8 | Ki | 3 | — | |
FMYKJLXRRQTBOR
|
6.8 | Ki | 3 | — | |
LNFFLKXYCXMVTE
|
6.8 | IC50 | 4 | — | |
PCJKSKCBOVMYIJ
|
6.8 | Ki | 4 | — | |
QDADLDKSQPFWPK
|
6.8 | IC50 | 2 | — | |
QFRLOVNUDLMMCT
|
6.8 | IC50 | 3 | — | |
WHNDEIMPFCLXJS
|
6.8 | Ki | 4 | — | |
ZIHDCWGBLPZTRG
|
6.8 | IC50 | 2 | — | |
JEBQNHANRCYVLC
|
6.8 | IC50 | 4 | — | |
KGJLXDHUTKATFA
|
6.8 | IC50 | 3 | — | |
LJZGCVPFHDAQAO
|
6.8 | Ki | 4 | — | |
UDWWUBBLCSIJEP
|
6.8 | IC50 | 2 | — | |
WJFVNKKWXMSMCB
|
6.8 | Ki | 3 | — | |
YFHSSOHMKVQRGY
|
6.8 | Ki | 2 | — | |
MCYQKGNJBOSMKC
|
6.8 | IC50 | 4 | — | |
PWINHDRBCUZSHX
|
6.8 | IC50 | 2 | — | |
QQZSKYDYMQGTTF
|
6.8 | IC50 | 3 | — | |
ZBNVNRCRULQVAR
|
6.8 | IC50 | 3 | — | |
JJFSLRIQURRAOH
|
6.8 | IC50 | 4 | — | |
LGACDLUVLNDBOB
|
6.8 | IC50 | 4 | — | |
BHVRFNJEHAGAIV
|
6.8 | IC50 | 4 | — | |
PUMWIMQYYHNBAM
|
6.7 | IC50 | 4 | — | |
AHRNMDRWMJFRTC
|
6.7 | IC50 | 2 | — | |
HDQBKIWKLLGTGO
|
6.7 | IC50 | 4 | — | |
GACCXUQYGGYVOX
|
6.7 | Ki | 2 | — | |
YRDWNESAGCXMTG
|
6.7 | IC50 | 4 | — | |
ZNUMRCPRXWDFHV
|
6.7 | IC50 | 4 | — | |
BBNDBOWNUASXHH
|
6.7 | Ki | 3 | — | |
SSNVUEXJJQDRMC
|
6.7 | IC50 | 2 | — | |
VGIWPEJPLFVKSL
|
6.7 | Ki | 4 | — | |
DVFMRMSQBLLRFB
|
6.7 | IC50 | 3 | — | |
JGMRVBHBMAPFGQ
|
6.7 | Ki | 3 | — | |
MJMYPIVLFFMZAC
|
6.7 | Ki | 3 | — | |
SFXFJMNNVMLAHN
|
6.7 | Ki | 4 | — | |
VMVOHHPQIAPYHG
|
6.7 | IC50 | 4 | — | |
YRVGOKKZUPVDNC
|
6.7 | IC50 | 3 | — | |
HDSWAYTVBYZPAG
|
6.7 | IC50 | 2 | — | |
BBAWEDCPNXPBQM
|
6.7 | IC50 | 9 | — | |
CTYIIVFLDQCJPG
|
6.7 | IC50 | 2 | — | |
CTYIIVFLDQCJPG
|
6.7 | IC50 | 2 | — | |
HCLPDRDQDGUFSD
|
6.7 | IC50 | 4 | — | |
TYDCYAYSUZPKGW
|
6.7 | Ki | 4 | — |