Target Details
| UniProt AC | P07858 |
|---|---|
| Gene Symbol | CTSB |
| Protein Name | Cathepsin B |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00112 (Peptidase_C1) PF08127 (Propeptide_C1) |
Summary
- Multi-target molecules 494
- Clinical molecules 10
- Avg pChEMBL 7.05
KEGG Pathways (6)
Associated Diseases (2)
Active Molecules (494)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VZJRPBWJESTYLV
|
7.1 | IC50 | 4 | — | |
KIDPFKMKRUSRRX
|
7.1 | IC50 | 4 | — | |
PGOQBJBMASKTEL
|
7.1 | IC50 | 3 | Yes | |
QVDJMLQSYRSZKC
|
7.1 | IC50 | 6 | Yes | |
DFQDPBLCCLZOCK
|
7.1 | IC50 | 6 | — | |
SWPXTIFAGIZWNX
|
7.1 | IC50 | 3 | — | |
DXLLSNZJTDGBRA
|
7.0 | IC50 | 4 | — | |
WYMQUJDMERVVKY
|
7.0 | Ki | 4 | — | |
GZGBHAIADJLADQ
|
7.0 | IC50 | 4 | — | |
MIKDFLKJUSAVHP
|
7.0 | IC50 | 3 | — | |
YODJPZCMOLJXNN
|
7.0 | Ki | 4 | — | |
NGBKFLTYGSREKK
|
7.0 | IC50 | 4 | — | |
APTHLSASJXHTAY
|
7.0 | Ki | 4 | — | |
PYZOXRXOZRPQAH
|
7.0 | IC50 | 4 | — | |
QFXNURNWJUSIOB
|
7.0 | Ki | 4 | — | |
UHNROXZSASTRFP
|
7.0 | IC50 | 4 | — | |
WJFAAUIYJQVQJJ
|
7.0 | IC50 | 3 | Yes | |
AODZHARIGFCGAC
|
7.0 | Ki | 2 | — | |
BNXDYZBRHZMVRA
|
7.0 | IC50 | 4 | — | |
IMOSLUWKGNEVCI
|
7.0 | IC50 | 2 | — | |
KRMYDWCAHQJBOD
|
7.0 | Ki | 4 | — | |
LWTHIEWNFZTHDQ
|
7.0 | IC50 | 4 | — | |
PMFBLJXNSAHZSG
|
7.0 | Ki | 3 | Yes | |
PMFBLJXNSAHZSG
|
7.0 | Ki | 2 | — | |
QLCDJMHVAVRDAU
|
7.0 | Ki | 3 | — | |
XERMNVUWYPYRPN
|
7.0 | Ki | 3 | — | |
FHIFVYKWPHPFEV
|
7.0 | Ki | 4 | — | |
NILSEPPHIUAUFQ
|
7.0 | IC50 | 4 | — | |
WAWCVPQCGNEDNX
|
7.0 | IC50 | 4 | — | |
ASDYDEDXCKSKAM
|
7.0 | Ki | 3 | — | |
AXVMAPSVAWPASZ
|
7.0 | Ki | 3 | — | |
BKMARWROUWRNAF
|
7.0 | IC50 | 3 | — | |
FGQCYIJCJZGOCQ
|
7.0 | IC50 | 2 | — | |
NAYHGPCOIURHDG
|
7.0 | Ki | 3 | — | |
YGOOSESWCCPOHN
|
7.0 | IC50 | 4 | — | |
HBSWEZXYFZOCOH
|
6.9 | IC50 | 4 | — | |
OSWTUQCVSFYKDC
|
6.9 | IC50 | 2 | — | |
XJKKWXRUCDAJHK
|
6.9 | IC50 | 4 | — | |
XJPDKOSJXFJJJW
|
6.9 | Ki | 3 | — | |
IYGWXNGZSDQPFR
|
6.9 | IC50 | 4 | — | |
VMUVUIMPWWGDDN
|
6.9 | IC50 | 4 | — | |
HMRWYWBGKLAOAI
|
6.9 | Ki | 3 | — | |
HQSRTSNGRWFCQM
|
6.9 | Ki | 2 | — | |
RYQRKWPMUFTILJ
|
6.9 | IC50 | 2 | — | |
XHGOLGYGBDIOFD
|
6.9 | IC50 | 3 | — | |
ANZFZARZEQENJQ
|
6.9 | Ki | 4 | — | |
FIVYCSWOCXEWSE
|
6.9 | IC50 | 4 | — | |
GTUQEIQBOYMZGW
|
6.9 | IC50 | 2 | — | |
BVJMYPXCAYDMBJ
|
6.9 | Ki | 3 | — | |
TYRKGQFUSLPRSY
|
6.9 | IC50 | 4 | — |