Target Details
| UniProt AC | P07858 |
|---|---|
| Gene Symbol | CTSB |
| Protein Name | Cathepsin B |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00112 (Peptidase_C1) PF08127 (Propeptide_C1) |
Summary
- Multi-target molecules 494
- Clinical molecules 10
- Avg pChEMBL 7.05
KEGG Pathways (6)
Associated Diseases (2)
Active Molecules (494)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NJKWZQGOBIFPBG
|
7.2 | IC50 | 3 | — | |
SFHXUNXRQNJLAE
|
7.2 | IC50 | 3 | — | |
AJAZMOFONMJGNP
|
7.2 | IC50 | 3 | — | |
CGAOFGCVDRGRSC
|
7.2 | IC50 | 4 | — | |
HBIOASKCQSACJZ
|
7.2 | IC50 | 2 | — | |
WISLRZADXFYSET
|
7.2 | IC50 | 4 | — | |
WUCMINQNTKBQNK
|
7.2 | IC50 | 2 | — | |
LLCRBOWRJOUJAE
|
7.2 | IC50 | 4 | — | |
PJOCENBBWQXQGY
|
7.2 | Ki | 3 | — | |
UABYWVBODUFLHL
|
7.2 | Ki | 2 | — | |
YBSWDIITMXRJIB
|
7.2 | IC50 | 4 | — | |
HRJIPNPMMDEUDH
|
7.2 | Ki | 3 | — | |
UZMSYDMWVBDKEM
|
7.2 | IC50 | 4 | — | |
ZGXKAZRUQQNMKC
|
7.2 | Ki | 3 | — | |
VHNVOAVIDBRLFO
|
7.2 | IC50 | 4 | — | |
VQKHIDNPFSGTTG
|
7.2 | IC50 | 2 | — | |
XXCXONRLKKHITM
|
7.2 | Ki | 3 | — | |
YUMYYTORLYHUFW
|
7.2 | Ki | 3 | — | |
YUMYYTORLYHUFW
|
7.2 | Ki | 3 | — | |
ZPVHBQIGHVBBKF
|
7.2 | IC50 | 3 | — | |
CAILNONEKASNSH
|
7.2 | IC50 | 4 | — | |
CAILNONEKASNSH
|
7.2 | IC50 | 3 | — | |
AIBOMLIMFLTQOS
|
7.2 | IC50 | 3 | — | |
JLZPHDGPTVJCOI
|
7.2 | IC50 | 4 | — | |
KRBOYQNUSRICHT
|
7.2 | Ki | 4 | — | |
DSMGEPBRPIEQKD
|
7.2 | IC50 | 4 | — | |
FYNZPHYKPPZBFB
|
7.2 | IC50 | 4 | — | |
JNRHNGGTJOBXHL
|
7.2 | IC50 | 3 | Yes | |
UUBYFYHAUYKPFR
|
7.2 | IC50 | 4 | — | |
YCPWFRMYSJKIIG
|
7.2 | IC50 | 4 | — | |
HJXOIRIPJDWFBS
|
7.2 | IC50 | 8 | — | |
KTAAIKREGSDHNS
|
7.2 | Ki | 4 | — | |
SYBYCMXFKUMMNW
|
7.2 | IC50 | 4 | — | |
YYVYNDITYXLIBI
|
7.2 | IC50 | 4 | — | |
DMDNERFCUCYCGM
|
7.1 | IC50 | 9 | — | |
GMHBWGMFTPGDOI
|
7.1 | IC50 | 3 | — | |
KVMJONNVSMEASA
|
7.1 | Ki | 4 | — | |
QFFDVXSXLOXTPD
|
7.1 | Ki | 4 | — | |
QQPGHYGBHVMSNJ
|
7.1 | IC50 | 3 | — | |
XQNARHBXPKVMJL
|
7.1 | Ki | 2 | — | |
BQWWAZOZDJROFE
|
7.1 | IC50 | 4 | — | |
WSJWUIDLGZAXID
|
7.1 | IC50 | 2 | — | |
BPWNJPXVAFVVPP
|
7.1 | IC50 | 4 | — | |
DSMGEPBRPIEQKD
|
7.1 | IC50 | 3 | — | |
JBXZNIFMTVSEQN
|
7.1 | IC50 | 4 | — | |
PXAFUBGFZCXLCE
|
7.1 | IC50 | 4 | — | |
DWZIHGHEWITDKK
|
7.1 | Ki | 2 | — | |
RSIVRPBUNKODPD
|
7.1 | IC50 | 4 | — | |
OXQKFIHVHFGYRB
|
7.1 | Ki | 2 | — | |
RHHVUDLUXPBHLT
|
7.1 | Ki | 3 | — |