Target Details
| UniProt AC | P07858 |
|---|---|
| Gene Symbol | CTSB |
| Protein Name | Cathepsin B |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00112 (Peptidase_C1) PF08127 (Propeptide_C1) |
Summary
- Multi-target molecules 494
- Clinical molecules 10
- Avg pChEMBL 7.05
KEGG Pathways (6)
Associated Diseases (2)
Active Molecules (494)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MWKOOGAFELWOCD
|
8.2 | Ki | 2 | — | |
LNRUTWQSWUTEMQ
|
8.2 | IC50 | 3 | — | |
QPGAIIGEIAEEEV
|
8.1 | Ki | 2 | — | |
HNMPKMOYOSYDNW
|
8.1 | Ki | 4 | — | |
LXQHAGZZTQHHEO
|
8.1 | Ki | 3 | — | |
YOGVFFRGTMXMRZ
|
8.1 | IC50 | 5 | — | |
OLNJKAXRBXUBTB
|
8.1 | IC50 | 10 | Yes | |
YKGCZJXHFVVNSC
|
8.1 | IC50 | 3 | — | |
RGJONKKMBWPLQS
|
8.1 | IC50 | 4 | — | |
PHUPMBKAOHPRFE
|
8.0 | IC50 | 3 | — | |
GDBQQVLCIARPGH
|
8.0 | IC50 | 10 | — | |
KEMMYXYZFDGSMT
|
8.0 | Ki | 2 | — | |
LTLYEAJONXGNFG
|
8.0 | IC50 | 9 | — | |
OCAFABUKPVDIBK
|
8.0 | IC50 | 3 | — | |
LTLYEAJONXGNFG
|
7.9 | IC50 | 5 | — | |
FSMMLXYBGWEIQQ
|
7.9 | Ki | 3 | — | |
KNHLEJQNWOTWPT
|
7.9 | Ki | 3 | — | |
NVLVLDJDOAWDLZ
|
7.9 | Ki | 3 | — | |
VUELCPPLRJAJCW
|
7.9 | Ki | 3 | — | |
LIQDTPYQUQZTGR
|
7.9 | Ki | 2 | — | |
NHFKTEZZOWFJBK
|
7.9 | IC50 | 4 | — | |
BWYBBMQLUKXECQ
|
7.9 | IC50 | 5 | — | |
VHDAHAMWVNXMSP
|
7.9 | IC50 | 7 | — | |
DVJGXMUWYFGXAS
|
7.8 | IC50 | 4 | Yes | |
WSJWUIDLGZAXID
|
7.8 | IC50 | 4 | — | |
ZQXYZTRTLGOBEJ
|
7.8 | IC50 | 4 | — | |
ZQXYZTRTLGOBEJ
|
7.7 | IC50 | 4 | — | |
SFIPFERDZPGSNY
|
7.7 | IC50 | 2 | — | |
NFPHFQIUODNJRD
|
7.7 | IC50 | 5 | — | |
UVZYTLSBNQCQLB
|
7.7 | IC50 | 2 | — | |
FQFPEBKHQBECAZ
|
7.6 | IC50 | 2 | — | |
MANOSMRLHJERON
|
7.6 | IC50 | 3 | — | |
MRAGOGINUXYQRY
|
7.6 | Ki | 3 | — | |
BBECUGKQKLZBOE
|
7.6 | Ki | 4 | — | |
GIRULLDKCABKLD
|
7.6 | IC50 | 3 | — | |
NGBKFLTYGSREKK
|
7.6 | Ki | 4 | — | |
JCUWWLFQYPMDMI
|
7.6 | Ki | 4 | — | |
PWVVGLGMUWKXFN
|
7.6 | Ki | 3 | — | |
DNRVBUZMGUEKCJ
|
7.6 | IC50 | 3 | — | |
PVEWYPRSIGWUAA
|
7.6 | Ki | 2 | — | |
ZLZXUNHJWVLGTE
|
7.6 | IC50 | 4 | — | |
ZUKNWGIRWRHHPH
|
7.6 | IC50 | 4 | — | |
XIICSQSWOYKKRN
|
7.6 | Ki | 3 | — | |
KFJNQHUVTVCSPY
|
7.5 | Ki | 3 | — | |
ASRBKZHDORPEHO
|
7.5 | IC50 | 5 | — | |
ZBRHHBWBGUXOAL
|
7.5 | IC50 | 4 | — | |
IWVHDBTWXSMDEF
|
7.5 | IC50 | 4 | — | |
JTLMIAYFCQRTPH
|
7.5 | IC50 | 2 | — | |
QCEJIUAKOBMHJA
|
7.5 | IC50 | 2 | — | |
OFNOZMJQFVWTHP
|
7.5 | IC50 | 4 | — |