Target Details
| UniProt AC | P07858 |
|---|---|
| Gene Symbol | CTSB |
| Protein Name | Cathepsin B |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00112 (Peptidase_C1) PF08127 (Propeptide_C1) |
Summary
- Multi-target molecules 494
- Clinical molecules 10
- Avg pChEMBL 7.05
KEGG Pathways (6)
Associated Diseases (2)
Active Molecules (494)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KFSSAMTWPDRZDV
|
6.2 | Ki | 3 | — | |
VZRKGDOTBQOIIT
|
6.2 | Ki | 3 | — | |
YGHHDWRITNGHCH
|
6.2 | IC50 | 3 | — | |
YJZKURYVZRISEA
|
6.2 | IC50 | 2 | — | |
QOUJDAITQNPNTN
|
6.2 | IC50 | 3 | — | |
XMBJUJIJDVFEFD
|
6.2 | Ki | 4 | — | |
XRIMMJTYAWYVEL
|
6.1 | Ki | 4 | — | |
LFKWIZQIKIHFJP
|
6.1 | Ki | 4 | — | |
DKJNJGMFODPLQX
|
6.1 | IC50 | 2 | — | |
JZOIPLRHDZPXJN
|
6.1 | Ki | 3 | — | |
PLVWMBFPIAQRHK
|
6.1 | Ki | 5 | — | |
JBUOTMSLPJQXBQ
|
6.1 | IC50 | 2 | — | |
LBLSSIHBMJKAIZ
|
6.1 | Ki | 5 | — | |
UNVBTVJSVLCZTN
|
6.1 | IC50 | 2 | — | |
CQYBUPZZENVLPV
|
6.1 | Ki | 3 | — | |
NEFVERIOUCVCKE
|
6.1 | IC50 | 3 | — | |
WBJZVUPGWANLHC
|
6.1 | IC50 | 3 | — | |
YVQGWXFRALVDJS
|
6.1 | Ki | 3 | — | |
ONABDOMWRCXLPX
|
6.1 | IC50 | 2 | — | |
ARKFDHGHDFNOKH
|
6.1 | Ki | 4 | — | |
FBALKZAVEMIILY
|
6.1 | IC50 | 4 | — | |
YYDQGTWJPADAKS
|
6.1 | IC50 | 3 | Yes | |
HMXHWXUBXOQENS
|
6.1 | IC50 | 2 | — | |
IMTIJVSUXSYPRE
|
6.1 | Ki | 3 | — | |
UIUWSHIRBDIYGM
|
6.1 | IC50 | 3 | — | |
YVXJGGRCDIEJGL
|
6.1 | Ki | 3 | — | |
ZJLUYWUYIFDQKX
|
6.1 | Ki | 3 | — | |
QAVMBNFNRRNITG
|
6.0 | IC50 | 2 | — | |
RDZZBPHZWCRITM
|
6.0 | IC50 | 3 | — | |
RVUJRRBCTAYDMG
|
6.0 | Ki | 3 | — | |
XHBRHGRXSUUCGR
|
6.0 | IC50 | 4 | — | |
SOFNUHHKAHJEAL
|
6.0 | IC50 | 3 | — | |
UHJIJVSKCNIUQD
|
6.0 | Ki | 3 | — | |
VKPLBOPLYIVTRL
|
6.0 | IC50 | 3 | — | |
ZWVSPRDKHNVQBX
|
6.0 | IC50 | 2 | — | |
ZSSCFBDEVDZJNE
|
6.0 | Ki | 3 | — | |
IGWMYMDMZAKLGO
|
6.0 | IC50 | 3 | — | |
KFZXSMATDSSFDD
|
6.0 | IC50 | 2 | — | |
VEZZBPBPTOZPBS
|
6.0 | IC50 | 5 | — | |
FNEUKBQFZSGMQF
|
6.0 | IC50 | 3 | — | |
GHDIYQHGVKVLJX
|
6.0 | IC50 | 2 | — | |
NOTSCKFHTQJLMM
|
6.0 | IC50 | 3 | — | |
NRMMQFXZSPQQES
|
6.0 | Ki | 2 | — | |
VBHYQAVSSHIJNV
|
6.0 | Ki | 3 | — |