Target Details
| UniProt AC | P07711 |
|---|---|
| Gene Symbol | CTSL |
| Protein Name | Procathepsin L |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF08246 (Inhibitor_I29) PF00112 (Peptidase_C1) |
Summary
- Multi-target molecules 975
- Clinical molecules 8
- Avg pChEMBL 7.35
KEGG Pathways (8)
Active Molecules (975)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZBTGGZNSFPJDHD
|
8.7 | IC50 | 2 | — | |
KEHDYFXOYPSDFQ
|
8.6 | Ki | 3 | — | |
ZLUCDMYLHDPSAI
|
8.6 | Ki | 2 | — | |
MGJMPHPLAZFAST
|
8.6 | Ki | 2 | — | |
NGBKFLTYGSREKK
|
8.6 | IC50 | 6 | Yes | |
RXCRNUBYZRKEGC
|
8.6 | IC50 | 3 | Yes | |
KIDPFKMKRUSRRX
|
8.6 | IC50 | 4 | — | |
KQYFHIPAAHRARB
|
8.6 | Ki | 4 | — | |
NGAUZCRIRRLFOO
|
8.6 | IC50 | 2 | — | |
YBSWDIITMXRJIB
|
8.6 | IC50 | 4 | — | |
NGBKFLTYGSREKK
|
8.6 | IC50 | 4 | — | |
AFTKDSGGPNEFNN
|
8.6 | Ki | 3 | — | |
IMTIJVSUXSYPRE
|
8.5 | Ki | 3 | — | |
ZEFHIBBPLAGQMT
|
8.5 | IC50 | 2 | — | |
OKCRMEZBXWRMEQ
|
8.5 | Ki | 3 | — | |
OLGUEGSEWSHKEY
|
8.5 | IC50 | 2 | — | |
CYEUKAQPQWGZPP
|
8.5 | IC50 | 2 | — | |
YUJAVMJKRUKNMF
|
8.5 | IC50 | 2 | — | |
HSRHZZRELKYVLU
|
8.5 | IC50 | 2 | — | |
BUOGXVARMRYPBH
|
8.5 | IC50 | 2 | — | |
YKYTUXGHFZQFLY
|
8.5 | IC50 | 2 | — | |
FXGIQTGYEVOOOM
|
8.5 | Ki | 3 | — | |
HENHFYXQSRKTQB
|
8.5 | IC50 | 2 | — | |
INGVILAVYNKSSU
|
8.5 | IC50 | 2 | — | |
GLGCLPLEIOLAJV
|
8.4 | IC50 | 2 | — | |
GLGCLPLEIOLAJV
|
8.4 | IC50 | 2 | — | |
SCMSYZJDIQPSDI
|
8.4 | IC50 | 3 | — | |
NJNZLBJSRUADEP
|
8.4 | Ki | 2 | — | |
VJBNYTFCTIYDMG
|
8.4 | IC50 | 3 | — | |
BWYBBMQLUKXECQ
|
8.4 | Ki | 3 | — | |
FQFPEBKHQBECAZ
|
8.4 | IC50 | 2 | — | |
GXDULIFEODNFQZ
|
8.4 | IC50 | 4 | — | |
GXDULIFEODNFQZ
|
8.4 | IC50 | 4 | — | |
NFWSPCREWNOVLH
|
8.4 | Ki | 2 | — | |
NSXOUETVXVPOFT
|
8.4 | IC50 | 4 | — | |
RUJRINHGQAHHCG
|
8.4 | Ki | 2 | — | |
GDBQQVLCIARPGH
|
8.4 | IC50 | 10 | — | |
OLNJKAXRBXUBTB
|
8.4 | IC50 | 10 | Yes | |
RNCDJZGBJBIWFN
|
8.4 | Ki | 2 | — | |
DCWZLGBGEUHXOE
|
8.4 | IC50 | 2 | — | |
LMZYZVWKTJFLSL
|
8.4 | Ki | 2 | — | |
YUMYYTORLYHUFW
|
8.4 | IC50 | 5 | — | |
UZMSYDMWVBDKEM
|
8.4 | IC50 | 4 | — | |
VQKHIDNPFSGTTG
|
8.4 | IC50 | 2 | — | |
KFTMZNIURYIOKI
|
8.4 | Ki | 4 | — | |
BWYBBMQLUKXECQ
|
8.3 | Ki | 3 | — | |
ZDJKOPMEVPPKBM
|
8.3 | IC50 | 2 | — | |
NSNODLMCUTYBRZ
|
8.3 | IC50 | 2 | — | |
SKVFLJGZAOSWLB
|
8.3 | Ki | 2 | — | |
BVJMYPXCAYDMBJ
|
8.3 | Ki | 3 | — |