Target Details
| UniProt AC | P07711 |
|---|---|
| Gene Symbol | CTSL |
| Protein Name | Procathepsin L |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF08246 (Inhibitor_I29) PF00112 (Peptidase_C1) |
Summary
- Multi-target molecules 975
- Clinical molecules 8
- Avg pChEMBL 7.35
KEGG Pathways (8)
Active Molecules (975)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LBJZOWAHNPGWGP
|
9.1 | Ki | 3 | — | |
GZBOGFDHJAMENH
|
9.1 | Ki | 4 | — | |
ZZPFZJXGGZUTHR
|
9.1 | IC50 | 4 | — | |
IMOSLUWKGNEVCI
|
9.0 | IC50 | 2 | — | |
JTLMIAYFCQRTPH
|
9.0 | IC50 | 2 | — | |
BHJRNQHHESSIHC
|
9.0 | IC50 | 2 | — | |
NLXIOLKMPAPISS
|
9.0 | Ki | 2 | — | |
PHUPMBKAOHPRFE
|
9.0 | Ki | 3 | — | |
PUNDCXSIFPDSLX
|
9.0 | Ki | 2 | — | |
UWIUSTCLSVVZSO
|
9.0 | IC50 | 3 | — | |
MWBPTVRPPPPZPG
|
9.0 | Ki | 4 | — | |
UEZMKFGTDYYCKL
|
9.0 | IC50 | 3 | — | |
CXLLDJUTVUHIOR
|
8.9 | Ki | 2 | — | |
GJHYTSFTSOMLTG
|
8.9 | IC50 | 2 | — | |
GTBAQTKMASRCMG
|
8.9 | IC50 | 2 | — | |
KZCODYXMOKIMLT
|
8.9 | IC50 | 3 | — | |
YFUZVOLEKQFVCQ
|
8.9 | IC50 | 3 | — | |
YFUZVOLEKQFVCQ
|
8.9 | IC50 | 5 | — | |
JYIZNXQVPSOTAR
|
8.9 | Ki | 2 | — | |
NOMZQLLANMQZNR
|
8.9 | IC50 | 4 | — | |
NOMZQLLANMQZNR
|
8.9 | IC50 | 4 | — | |
BHJRNQHHESSIHC
|
8.9 | IC50 | 2 | — | |
HQHBNXAESHKMIQ
|
8.9 | IC50 | 2 | — | |
AWEFNCACPBKWGG
|
8.8 | Ki | 3 | — | |
LRGPAVMYPWWORG
|
8.8 | Ki | 4 | — | |
GJMFJSMWCBYWQN
|
8.8 | Ki | 2 | — | |
PTKUXWVYYVOZRE
|
8.8 | Ki | 3 | — | |
UTUSRLWZFBUDAM
|
8.8 | Ki | 4 | — | |
WSJWUIDLGZAXID
|
8.8 | IC50 | 4 | — | |
AWOGCPXUTJBQEG
|
8.8 | IC50 | 3 | Yes | |
AKAUMTCIIOMDTI
|
8.8 | IC50 | 3 | — | |
OXOTXDHSGCISLV
|
8.8 | Ki | 3 | — | |
VGIWPEJPLFVKSL
|
8.8 | Ki | 4 | — | |
YRDWNESAGCXMTG
|
8.8 | IC50 | 4 | — | |
YUJAVMJKRUKNMF
|
8.8 | IC50 | 2 | — | |
BFANIUCLYPUKCM
|
8.8 | IC50 | 2 | — | |
GIRULLDKCABKLD
|
8.7 | IC50 | 3 | — | |
ARWSHTCIMVGBCQ
|
8.7 | Ki | 4 | — | |
CXYMWYIUDRQGTR
|
8.7 | Ki | 2 | — | |
IWVHDBTWXSMDEF
|
8.7 | IC50 | 4 | — | |
NVOCHHPUHMFGSJ
|
8.7 | IC50 | 4 | — | |
NVOCHHPUHMFGSJ
|
8.7 | IC50 | 4 | — | |
VIFRNMGMIPTJQJ
|
8.7 | IC50 | 2 | — | |
YYIPDPNKLCJYIH
|
8.7 | IC50 | 2 | — | |
BSPZFJDYQHDZNR
|
8.7 | IC50 | 6 | — | |
XALMMLXCBLXHHZ
|
8.7 | IC50 | 2 | — | |
BJEZNOLUMLFYHR
|
8.7 | Ki | 3 | — | |
FGQCYIJCJZGOCQ
|
8.7 | IC50 | 2 | — | |
GJLXFFKSGIYTBC
|
8.7 | IC50 | 2 | — | |
VBPPNJCVXGAZDD
|
8.7 | Ki | 5 | — |