Target Details
| UniProt AC | P07711 |
|---|---|
| Gene Symbol | CTSL |
| Protein Name | Procathepsin L |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF08246 (Inhibitor_I29) PF00112 (Peptidase_C1) |
Summary
- Multi-target molecules 975
- Clinical molecules 8
- Avg pChEMBL 7.35
KEGG Pathways (8)
Active Molecules (975)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YWXWRCMYHIYBSJ
|
10.6 | Ki | 4 | — | |
VCANIUOBHBAPJH
|
10.4 | Ki | 3 | — | |
LMZYZVWKTJFLSL
|
10.4 | Ki | 3 | — | |
CLOALCKDNZPWBO
|
10.3 | Ki | 4 | — | |
MFWMOUYOCOANSI
|
10.3 | IC50 | 3 | — | |
FMYKJLXRRQTBOR
|
10.2 | Ki | 3 | — | |
QSXBDQVGNKRTPC
|
10.0 | IC50 | 2 | — | |
JICMCJAFBMCIIX
|
10.0 | IC50 | 3 | — | |
LKVLCOTZWXWKQV
|
10.0 | IC50 | 3 | — | |
GWGYOEFAMBIJPC
|
9.9 | Ki | 2 | — | |
TZYWCYJVHRLUCT
|
9.8 | IC50 | 23 | — | |
FTJHEEIVOBBMMC
|
9.8 | Ki | 5 | — | |
VLROHFCAQABUTJ
|
9.8 | IC50 | 3 | — | |
VZSXPUDQSLKVIR
|
9.7 | Ki | 4 | — | |
AUPZRAAKTGPDLC
|
9.7 | Ki | 4 | — | |
ONLDYVSTIWZOLP
|
9.6 | Ki | 4 | — | |
OIKITZBTDSAJQH
|
9.5 | Ki | 4 | — | |
YZBDFADJOLGKFN
|
9.5 | IC50 | 3 | — | |
GASCFELIQZXIAB
|
9.5 | IC50 | 3 | — | |
GUUHOTXBVVLLAX
|
9.5 | IC50 | 2 | — | |
NGBKFLTYGSREKK
|
9.5 | IC50 | 4 | — | |
XWMOCHXKDCBQPV
|
9.4 | Ki | 4 | — | |
BWYBBMQLUKXECQ
|
9.4 | IC50 | 5 | — | |
JESRGSWARNNMLP
|
9.4 | Ki | 4 | — | |
SCCNQBNFEHNRCO
|
9.4 | Ki | 4 | — | |
WFTHOJCUJHBJLJ
|
9.4 | Ki | 2 | — | |
BLJKFTVYZPTNBP
|
9.4 | Ki | 3 | — | |
DVJGXMUWYFGXAS
|
9.4 | IC50 | 4 | Yes | |
KRMYDWCAHQJBOD
|
9.3 | Ki | 4 | — | |
BTSJGBRRCQOXFA
|
9.3 | Ki | 2 | — | |
WJFVNKKWXMSMCB
|
9.3 | Ki | 3 | — | |
HWNYTOPEHDSGOF
|
9.3 | IC50 | 3 | — | |
JOBQWEVUTRQKOK
|
9.3 | IC50 | 3 | — | |
BBECUGKQKLZBOE
|
9.2 | Ki | 4 | — | |
UPWNNHRBMJWIBW
|
9.2 | IC50 | 3 | — | |
VEOFVKMRRKERDB
|
9.2 | Ki | 2 | — | |
ROYCRTHTOWKGBO
|
9.2 | Ki | 3 | — | |
GVIHWZBKUKQYMN
|
9.2 | IC50 | 2 | — | |
MCKCVIDASJTQSU
|
9.2 | Ki | 3 | — | |
QVDJMLQSYRSZKC
|
9.2 | IC50 | 6 | Yes | |
ZGXKAZRUQQNMKC
|
9.2 | Ki | 3 | — | |
PLVWMBFPIAQRHK
|
9.2 | Ki | 5 | — | |
CAQLLDUOKIHSBN
|
9.2 | IC50 | 3 | — | |
BEMWXCUECCHZDO
|
9.2 | IC50 | 4 | — | |
VEZZBPBPTOZPBS
|
9.2 | IC50 | 5 | — | |
OSWTUQCVSFYKDC
|
9.1 | IC50 | 2 | — | |
UGIIPXANIQTIRQ
|
9.1 | IC50 | 2 | — | |
YCYQOGPWUSMXGX
|
9.1 | Ki | 4 | — | |
LCGRTAPRJZMTIT
|
9.1 | IC50 | 3 | — | |
BSPZFJDYQHDZNR
|
9.1 | IC50 | 4 | — |