Target Details
UniProt ACP07478
Gene SymbolPRSS2
Protein NameTrypsin-2
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00089 (Trypsin)
Summary
  • Multi-target molecules 391
  • Clinical molecules 0
  • Avg pChEMBL 7.38
Associated Diseases (1)
Top Co-occurrence Targets
Active Molecules (391)
InChIKey pChEMBL Type Targets Clinical
NUHGXVSVNKUAAI 9.3 IC50 3
BTSOZAZYTDQHPD 9.3 IC50 3
JFRJDMYJBSGXDU 9.2 IC50 3
CIRQDIOMPWNRRE 9.2 IC50 3
QTHYYFNVNGQYDW 9.2 IC50 3
TYHYKNFAOZOJQV 9.2 IC50 3
CFUSBNZMUXPGOM 9.2 IC50 3
FSIZAFKKEFITQY 9.2 IC50 3
PFCOFKBCTGBATD 9.2 Ki 6
PJWRVDWTVAOOQV 9.2 Ki 7
ZQKIULTYLSTXBM 9.2 IC50 3
WSQXGFKMOUOXGW 9.1 IC50 3
JRNGHBUUFQDBPT 9.0 Ki 8
UNIOGIZCWAGOKV 8.9 Ki 6
JXJBQAMLLCEHTI 8.9 IC50 3
ANKIJLVYTUKGJM 8.8 Ki 6
KEWCBOBJEQHYIV 8.8 Ki 6
HUQGFODZSCBSLP 8.8 IC50 4
BUGKCANFLDYYKD 8.8 IC50 6
CDJAIRYCIJZATA 8.8 Ki 6
ZKPKJBOKOMILAA 8.8 Ki 6
CROZVKXDALXCPS 8.7 IC50 6
ZAXKLHPTMZESOW 8.6 IC50 5
XASIMHXSUQUHLV 8.6 IC50 7
XJJMRYCODRNFRY 8.6 Ki 5
FXYCTDRIKLDZRI 8.6 IC50 3
RSJYFASOCLFHRR 8.5 Ki 6
HAQNCPOGRFKYNP 8.5 Ki 4
BWSHEIOUBFDLNO 8.5 Ki 5
ZLJCFXPKCSWCGG 8.5 Ki 4
BHQDUYVBGREBCB 8.4 Ki 8
XQGVJTLGUGOPAJ 8.4 Ki 5
LAOYKAPCPZXMLS 8.4 Ki 5
PGUPEOWWTCYVPK 8.4 Ki 4
HTIXLULNBZFLJX 8.4 Ki 5
PRAPXLGHGHDFCO 8.3 Ki 5
DSEQCUGXKCOSSU 8.3 IC50 5
ZCJLCJMVJJVEQE 8.2 Ki 5
ZXIZUNRFGBZCHV 8.2 Ki 4
RDSVRCGNSLPORJ 8.2 Ki 5
GFXFOCFFDUYUAQ 8.2 Ki 5
KHTRPJFHQNRISN 8.2 Ki 5
OOSAWCAECZEMCW 8.2 Ki 6
DKWNMCUOEDMMIN 8.1 IC50 6
LFWUMCWXZZLCOX 8.1 IC50 3
OBRCAKGVHQFHGX 8.1 Ki 4
VPRDEDQBTIFZDM 8.1 Ki 6
VXDAVYUFYPFGDX 8.1 IC50 3
MHWPNEADOGSOHV 8.1 Ki 4
XJDVJJDJQXRAOB 8.1 Ki 4
2D structure