Target Details
UniProt ACP07477
Gene SymbolPRSS1
Protein NameSerine protease 1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00089 (Trypsin)
Summary
  • Multi-target molecules 1,293
  • Clinical molecules 1
  • Avg pChEMBL 7.57
Associated Diseases (1)
Top Co-occurrence Targets
Active Molecules (1,293)
InChIKey pChEMBL Type Targets Clinical
OCGKHKOQHRZKIM 8.3 Ki 2
YNGAKUMMINESNS 8.3 Ki 2
YYWBBLNCZBADRS 8.3 Ki 2
JPZAPLAFJYUWQP 8.3 Ki 2
LNNRGSRYUTXGEX 8.3 Ki 2
RDISPMRBPXPXDR 8.3 Ki 2
JBHHRVQRHSBNTN 8.3 Ki 2
QCKHQIYRKNPRBR 8.3 Ki 2
BLCYCYHFLMGVPO 8.3 Ki 3
GEGPKJUQKQSQAE 8.3 Ki 2
VTJKUQVDQBWOCA 8.3 Ki 2
FCUZICMQZZVVKV 8.2 Ki 2
ISYNRVLFJWYDPA 8.2 Ki 2
MZDLVWCRTMDQMT 8.2 Ki 2
ZCJLCJMVJJVEQE 8.2 Ki 5
ORIXUOJACQINEN 8.2 Ki 2
PJQIIQDUTSQWIS 8.2 Ki 2
ZXIZUNRFGBZCHV 8.2 Ki 4
RDSVRCGNSLPORJ 8.2 Ki 5
MWJAQZALXIOOQS 8.2 Ki 2
RNXYWZSBKYGCIA 8.2 Ki 2
GFXFOCFFDUYUAQ 8.2 Ki 5
KHTRPJFHQNRISN 8.2 Ki 5
LGUMIBZFRCAMKL 8.2 Ki 2
LGUMIBZFRCAMKL 8.2 Ki 2
OOSAWCAECZEMCW 8.2 Ki 6
VAHZBDOLKHNQEE 8.2 Ki 4
DKWNMCUOEDMMIN 8.1 IC50 6
OSXWFMAUTQKVIB 8.1 Ki 2
UWJTXKREKAAFAE 8.1 Ki 2
ARUHNEJEVKQAPD 8.1 Ki 2
HESPFXXTEAPSNR 8.1 Ki 2
OBRCAKGVHQFHGX 8.1 Ki 4
VPRDEDQBTIFZDM 8.1 Ki 6
VXDAVYUFYPFGDX 8.1 IC50 3
ACEUOZVTHUQNKZ 8.1 Ki 2
KAGLWQUWUNBAOO 8.1 IC50 5
MHWPNEADOGSOHV 8.1 Ki 4
NZEAENHOWXTKPM 8.1 IC50 5
OLNJKAXRBXUBTB 8.1 Ki 10 Yes
QRSQMHVQHCFHOA 8.1 Ki 2
TYNHUYPNNVQELL 8.1 IC50 2
VXDAVYUFYPFGDX 8.1 Ki 5
ANSWPKCJQAZJTJ 8.1 Ki 3
PGPODLSJZFFJCS 8.1 Ki 2
PLAZRHIWSZYQOZ 8.1 IC50 2
VGPDGESAAIVXNO 8.1 Ki 3
XJDVJJDJQXRAOB 8.1 Ki 4
YELLYQPFWRBWSX 8.1 Ki 2
KZTWLZSQCPXGLA 8.1 Ki 2
2D structure