Target Details
UniProt ACP07477
Gene SymbolPRSS1
Protein NameSerine protease 1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00089 (Trypsin)
Summary
  • Multi-target molecules 1,293
  • Clinical molecules 1
  • Avg pChEMBL 7.57
Associated Diseases (1)
Top Co-occurrence Targets
Active Molecules (1,293)
InChIKey pChEMBL Type Targets Clinical
WBFBQDAAAKLBHB 11.6 Ki 2
LHVRINJTNXVOIY 10.7 IC50 2
KWSMBEJYQLCPRA 10.5 Ki 6
FXFYPTZERULUBS 10.3 Ki 3
FXFYPTZERULUBS 10.3 Ki 5
AHMVMZSRXLKIHQ 10.3 Ki 2
QQBRBPSSMDPLLA 10.3 Ki 5
NUFFEXHLLOWDJE 10.1 Ki 2
QQBRBPSSMDPLLA 10.0 Ki 4
VEZVTGKCTALENO 10.0 Ki 3
WRDBDBHZQFTGKU 10.0 Ki 2
DNTBEYIBOAUAAQ 9.9 Ki 2
LHVRINJTNXVOIY 9.9 IC50 2
AOURNCMLYSCKQM 9.8 Ki 2
IWNWXPRWSFWNMU 9.8 Ki 5
WLLYNBSNNIWCMO 9.8 Ki 5
MMGDDXDPHXOWCE 9.8 IC50 3
CAZDAAGVXGRUJG 9.7 Ki 2
JBNVPTQXOVALOW 9.7 IC50 3
VUEKGNQWFYIQDE 9.7 Ki 2
YSOABFZKTWHRBK 9.7 Ki 2
CAZDAAGVXGRUJG 9.7 Ki 2
UTVUAMNDZNEKQJ 9.7 Ki 2
DBKBHOJMFKSRDI 9.7 Ki 2
GLUNNQRGCXKATF 9.7 Ki 2
IZIUQJQPQGQZKY 9.7 IC50 3
UCLUAJGIZROTHN 9.7 IC50 3
DAIBADVQGWIEFB 9.7 IC50 3
PPLWQAMMKNZODE 9.7 Ki 2
RFEWBKIWAZDYIJ 9.7 Ki 2
UIEZZGBGVSZNGO 9.7 IC50 3
ZDHSABZRIYUHBN 9.7 Ki 2
PJXAFQKIXSYHNC 9.7 Ki 2
TYCYCBSPZNGACF 9.7 IC50 3
YIGYWYRLQOYYSK 9.7 Ki 2
BLKGMXVBRRZSBK 9.6 Ki 2
OBIKLPPECWOYDP 9.6 IC50 3
OZWQWPUGYJDKEB 9.6 IC50 3
XSCPZORUJWDPBT 9.6 IC50 3
BTUCLQIWMTZBRU 9.6 IC50 3
CWRWISLBWBEDFR 9.6 IC50 3
KSTWXAMIEVDBQH 9.6 Ki 2
UMHVCSSJGIEZFT 9.6 Ki 2
UTVUAMNDZNEKQJ 9.6 Ki 2
DYLRVSKCRNOULJ 9.6 IC50 3
IMPSSSBKEBYTAU 9.6 IC50 3
URBHOBROHUTPDR 9.6 IC50 3
ALVURNATRNYWEF 9.6 Ki 2
BWLGESZOIWZYBW 9.6 IC50 3
CEBSLTBKCPYKRD 9.5 Ki 2
2D structure