Target Details
| UniProt AC | P07384 |
|---|---|
| Gene Symbol | CAPN1 |
| Protein Name | Calpain-1 catalytic subunit |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01067 (Calpain_III) PF13833 (EF-hand_8) PF00648 (Peptidase_C2) |
Summary
- Multi-target molecules 168
- Clinical molecules 5
- Avg pChEMBL 6.91
KEGG Pathways (8)
Associated Diseases (1)
Active Molecules (168)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BMJOPMWNNPSOFV
|
6.2 | Ki | 2 | — | |
ITIYFQNKFLZJTC
|
6.2 | Ki | 2 | — | |
XOOLYFKEZMFYKD
|
6.2 | Ki | 2 | — | |
YVQGWXFRALVDJS
|
6.2 | Ki | 3 | — | |
YXADZLOTFPFSML
|
6.2 | Ki | 3 | — | |
IAIIFNKYOCEUDZ
|
6.2 | Ki | 2 | — | |
LKEAIRWHRIHIEF
|
6.1 | Ki | 2 | — | |
MRMDMJWTKTVMPI
|
6.1 | Ki | 2 | — | |
LBWUIVAFNQOLOB
|
6.1 | Ki | 2 | — | |
NLQSCVDOWLITDK
|
6.1 | Ki | 2 | — | |
SFXFJMNNVMLAHN
|
6.1 | Ki | 4 | — | |
YFQOCPUAXDVMOS
|
6.1 | Ki | 2 | — | |
LPIGFPBIPKWMAQ
|
6.1 | Ki | 2 | — | |
WKNXHKNTWIOTFP
|
6.0 | Ki | 2 | — | |
BNGWXRGSXSJXMS
|
6.0 | IC50 | 2 | — | |
JKZCALXNJCQERK
|
6.0 | Ki | 3 | — | |
NQTCNKWSPHAXMS
|
6.0 | Ki | 2 | — | |
ONIATLXCZWBRKB
|
6.0 | Ki | 2 | — |