Target Details
UniProt ACP07384
Gene SymbolCAPN1
Protein NameCalpain-1 catalytic subunit
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF01067 (Calpain_III) PF13833 (EF-hand_8) PF00648 (Peptidase_C2)
Summary
  • Multi-target molecules 168
  • Clinical molecules 5
  • Avg pChEMBL 6.91
Associated Diseases (1)
Top Co-occurrence Targets
Active Molecules (168)
InChIKey pChEMBL Type Targets Clinical
SFZKIYLOJIJGLV 6.7 Ki 2
ODVBWVUZXJFGFP 6.7 IC50 2
BWKQXOPKLULOSF 6.6 Ki 2
GPBVKHGLFLZPRW 6.6 Ki 2
LKVFZCXXFXGYDC 6.6 Ki 3
SFOHMHDPSOPFJL 6.6 Ki 3
PBXPKBVKBJPJNW 6.6 Ki 2
XUFBOUSMDJZDOA 6.6 IC50 2
YIRUASIRQWZPIZ 6.6 IC50 2 Yes
VPUYRFKIVDMDKL 6.5 Ki 2
YLELJBQQWFIURX 6.5 Ki 3
LKJAJQNXOPUHBI 6.5 Ki 2
GDBQQVLCIARPGH 6.5 IC50 10
WNSZSZRXSNLYSL 6.5 Ki 2
XWPMWIRSEUHFET 6.5 Ki 3
GMTPAJDXCPJPRB 6.5 Ki 2
BALDEWOSOSUCAN 6.5 Ki 3
NDHXUSGFCSYNLZ 6.5 Ki 2
XJZJHBWBHUESJD 6.5 Ki 3
CZPUWGZBBOMJKE 6.5 Ki 2
FOBRVMHYTDWMJG 6.5 Ki 2
FUUFQEWEOLXXBO 6.5 Ki 2
MSLYBTUYFAYWQS 6.5 Ki 2
NRYJQWJSMMVVFJ 6.5 Ki 2
QXMOZKBLCRFIAZ 6.5 Ki 2
ZEPJUNYIGZQROD 6.5 IC50 2
YVMYGKAQQWIQNK 6.4 Ki 2
CLBKCGOYQYVDNB 6.4 Ki 2
JJAOOYMOIBDGJA 6.4 Ki 2
LAMTYMVWEHUWRZ 6.4 Ki 2
CAILNONEKASNSH 6.4 IC50 4
CAILNONEKASNSH 6.4 IC50 3
OIKITZBTDSAJQH 6.4 IC50 4
JGMRVBHBMAPFGQ 6.4 Ki 3
RVUJRRBCTAYDMG 6.4 Ki 3
VQYAUQQZKIBVFS 6.3 Ki 2
OCIZFJKKIPDOAQ 6.3 Ki 2
BOLCGBQAKSTBLH 6.3 IC50 2
BXUSCFDRWLTJIE 6.3 Ki 2
OWMWWYSNZALAER 6.3 Ki 3
OWSUSRRECBEBIZ 6.3 Ki 2
PVWAECRYPMJXPR 6.3 Ki 2
VLHHFIURJMMQSU 6.3 Ki 3
XOVPCPRZRHQFBI 6.3 IC50 15
NTZYOTXUVHBKSM 6.3 IC50 2
PCBGEKNWVUOWNB 6.2 Ki 2
ASXVEBPEZMSPHB 6.2 IC50 3
BYDZMKUUIQPQOJ 6.2 Ki 2
CLRFYTGANQZOBS 6.2 IC50 41
YGHHDWRITNGHCH 6.2 IC50 3
2D structure