Target Details
UniProt ACP07384
Gene SymbolCAPN1
Protein NameCalpain-1 catalytic subunit
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF01067 (Calpain_III) PF13833 (EF-hand_8) PF00648 (Peptidase_C2)
Summary
  • Multi-target molecules 168
  • Clinical molecules 5
  • Avg pChEMBL 6.91
Associated Diseases (1)
Top Co-occurrence Targets
Active Molecules (168)
InChIKey pChEMBL Type Targets Clinical
GWLZMBFVBYHGBD 7.1 Ki 2
BFOUDLDYLQQVEB 7.1 Ki 2
SEANAGCTCGCPQM 7.1 Ki 3
XJPDKOSJXFJJJW 7.1 IC50 3
OIXYHRZFKWJACP 7.1 IC50 2
NWUVYAAEXDXAHP 7.0 IC50 2
PNRWOFORTRJIMC 7.0 Ki 2
BJVLXPNAIXTDOW 7.0 Ki 3
VMVOHHPQIAPYHG 7.0 IC50 4
BYUMFTKUIXAFNT 7.0 IC50 2
JFFBDCJEPWDUJE 7.0 Ki 2
LTLYEAJONXGNFG 7.0 IC50 9
NGBKFLTYGSREKK 7.0 IC50 4
OFDVDFSINZOAMJ 7.0 IC50 2
OITJHBJCHPRBCI 7.0 IC50 2
ORFNBDAQQVIIPT 7.0 IC50 2
RFLQJGASGWLMCH 7.0 Ki 3
PVEWYPRSIGWUAA 7.0 IC50 2
FYLLWVNXHDSOBP 7.0 IC50 2
ABCDOWZVJWRRMY 7.0 Ki 3
VTIAIZFLWATOKO 7.0 Ki 3
YYVPOIBILWMYMW 7.0 Ki 2
DPHACENAZHGWHS 6.9 IC50 4
FRACLEVIDYQZNB 6.9 Ki 3
IZOVMLGFODKHHH 6.9 Ki 2
ODDXFSGPQQWPEO 6.9 Ki 2
SOPMJELGLOZMNK 6.9 Ki 2
DQCYYWKVEFPNIO 6.9 Ki 3
LWZDBQBMLCPSSM 6.9 Ki 2
OXQKFIHVHFGYRB 6.9 IC50 2
AHEDBTSELMBNTN 6.9 IC50 2
UABYWVBODUFLHL 6.9 IC50 2
BSQXGCSIDWZSHW 6.8 IC50 2
TZVQRMYLYQNBOA 6.8 Ki 2
AYSDUNWXRUGZRO 6.8 IC50 2
ZOBGGAIYJYPPGQ 6.8 IC50 2
PJJKGPCXAZFMMA 6.8 Ki 2
PRVNMMSXHWFZAQ 6.8 Ki 3
MWKSRKSEWLRPBL 6.8 Kd 1075
MDMSJUTXKFAZPC 6.7 Ki 2
BOVPSXHLLSLLHY 6.7 Ki 2
FYNLJGLHDFSIRG 6.7 Ki 2
GOYRCQFAGVGQLH 6.7 Ki 3
QDIFXVWJRNFSAW 6.7 Ki 3
QFMKANIDVYDNPI 6.7 Ki 3
WIWTZPBWDNQRGX 6.7 Ki 2
WJDCRUSBRSNMME 6.7 Ki 3
DJCVSFWGKYHMKH 6.7 Ki 2
VZPAOLJPGFQEEK 6.7 Ki 3
ALWTVFUIPPAQBH 6.7 Ki 2
2D structure