Target Details
| UniProt AC | P07384 |
|---|---|
| Gene Symbol | CAPN1 |
| Protein Name | Calpain-1 catalytic subunit |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01067 (Calpain_III) PF13833 (EF-hand_8) PF00648 (Peptidase_C2) |
Summary
- Multi-target molecules 168
- Clinical molecules 5
- Avg pChEMBL 6.91
KEGG Pathways (8)
Associated Diseases (1)
Active Molecules (168)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XVYMHUPUYXWRAO
|
9.7 | Ki | 3 | — | |
LXQHAGZZTQHHEO
|
9.5 | Ki | 3 | — | |
BPXIXWUDIQQWFO
|
9.4 | Ki | 2 | — | |
UEGOQZVAGRIZMF
|
9.4 | Ki | 2 | — | |
ALMQDMPRSWZSDO
|
8.5 | Ki | 2 | — | |
XGJGWYRHLPSMLW
|
8.3 | IC50 | 2 | — | |
PMFBLJXNSAHZSG
|
8.2 | Ki | 3 | Yes | |
PMFBLJXNSAHZSG
|
8.2 | Ki | 2 | — | |
WSJWUIDLGZAXID
|
8.1 | IC50 | 2 | — | |
YTSRZPGVQKOFFF
|
8.1 | IC50 | 2 | — | |
AODZHARIGFCGAC
|
8.1 | Ki | 2 | — | |
UNCOFUQMWOIDMS
|
8.1 | Ki | 3 | — | |
LFXDKGYPGBYESW
|
8.0 | IC50 | 3 | — | |
UZISLNFABGKCDY
|
7.9 | IC50 | 2 | — | |
BSPZFJDYQHDZNR
|
7.8 | IC50 | 4 | — | |
CSKGFHNQMOIAFM
|
7.7 | IC50 | 4 | Yes | |
PLVWMBFPIAQRHK
|
7.7 | Ki | 5 | — | |
WQBLPTWYDVNJDE
|
7.7 | IC50 | 2 | — | |
WSJWUIDLGZAXID
|
7.7 | IC50 | 4 | — | |
RJWLAIMXRBDUMH
|
7.6 | IC50 | 2 | — | |
DSYDMMPAZVEHMK
|
7.6 | IC50 | 2 | — | |
SMHWTXZVZOFOFA
|
7.6 | IC50 | 2 | — | |
PAURRTCLMITPQE
|
7.5 | IC50 | 3 | — | |
HBIOASKCQSACJZ
|
7.5 | IC50 | 2 | — | |
VXFRMVRMWOZAFZ
|
7.5 | IC50 | 2 | — | |
RXCRNUBYZRKEGC
|
7.5 | IC50 | 3 | Yes | |
WNILNJHVHCOVFU
|
7.4 | IC50 | 2 | — | |
NGBKFLTYGSREKK
|
7.4 | IC50 | 4 | — | |
SCMSYZJDIQPSDI
|
7.4 | IC50 | 3 | — | |
QAVMBNFNRRNITG
|
7.3 | IC50 | 2 | — | |
PGGUOGKHUUUWAF
|
7.3 | IC50 | 3 | — | |
BPDWJQKYAHEPMF
|
7.3 | IC50 | 2 | — | |
WYYJIPJWAOEKRW
|
7.3 | Ki | 2 | — | |
ZIHDCWGBLPZTRG
|
7.3 | IC50 | 2 | — | |
BQWHGKILBWBBEZ
|
7.3 | Ki | 3 | — | |
RLWHWANZNLEGCV
|
7.3 | IC50 | 3 | — | |
HHNHYEDODWWQEY
|
7.3 | IC50 | 2 | — | |
XUZYDWHWSIJZRS
|
7.3 | IC50 | 2 | — | |
KFJNQHUVTVCSPY
|
7.2 | Ki | 3 | — | |
MRAGOGINUXYQRY
|
7.2 | IC50 | 3 | — | |
YQBJQKXVOBLSJT
|
7.2 | IC50 | 3 | — | |
FBLCORIGBOTKPH
|
7.2 | IC50 | 3 | — | |
DSEJDNPJKDDYTK
|
7.2 | Ki | 2 | — | |
GLNKVXFQBYGNDP
|
7.2 | Ki | 3 | — | |
NGBKFLTYGSREKK
|
7.2 | IC50 | 6 | Yes | |
ZWWFTIUCCNWEGY
|
7.2 | IC50 | 3 | — | |
BSPZFJDYQHDZNR
|
7.1 | IC50 | 6 | — | |
GLEMPIVMKMAASA
|
7.1 | Ki | 3 | — | |
NTZYOTXUVHBKSM
|
7.1 | IC50 | 2 | — | |
WUCMINQNTKBQNK
|
7.1 | IC50 | 2 | — |