Target Details
| UniProt AC | P07333 |
|---|---|
| Gene Symbol | CSF1R |
| Protein Name | Macrophage colony-stimulating factor 1 receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00047 (ig) PF25305 (Ig_PDGFR_d4) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 896
- Clinical molecules 90
- Avg pChEMBL 7.53
KEGG Pathways (11)
- Acute myeloid leukemia
- Cytokine-cytokine receptor interaction
- Hematopoietic cell lineage
- MAPK signaling pathway
- Osteoclast differentiation
- PI3K-Akt signaling pathway
- Pathways in cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Transcriptional misregulation in cancer
- Viral protein interaction with cytokine and cytokine receptor
Associated Diseases (3)
Active Molecules (896)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QJIVDCJIPGAKQZ
|
7.8 | Ki | 25 | — | |
QTQUAHGXBLFSCH
|
7.8 | Ki | 10 | — | |
XJSFDMGICAWQFS
|
7.8 | Ki | 60 | — | |
YACXOXQTGJXYNX
|
7.8 | Ki | 11 | — | |
ZEGUNGLZSRRDSK
|
7.8 | IC50 | 3 | — | |
CQXYAWGSQLDRAK
|
7.8 | IC50 | 3 | — | |
FHEQFUUMLHFZOS
|
7.8 | IC50 | 3 | — | |
HAZVCDSGCISCHC
|
7.8 | IC50 | 3 | — | |
NGYRNPFGDZALOR
|
7.8 | IC50 | 3 | — | |
DRJKEMBRQFSLFC
|
7.8 | IC50 | 3 | — | |
BLBRCCGITKEOBW
|
7.7 | IC50 | 3 | — | |
RHAURHVPLMBUOW
|
7.7 | IC50 | 2 | — | |
SSSQBBWJMZYDLU
|
7.7 | IC50 | 2 | — | |
UHWRZSFKINYFKS
|
7.7 | IC50 | 2 | — | |
YOHLRCOPRAVUCJ
|
7.7 | IC50 | 6 | — | |
GJQVPMWSXKFICV
|
7.7 | IC50 | 3 | — | |
GJQVPMWSXKFICV
|
7.7 | IC50 | 3 | — | |
GVDDEBQJCYQLKV
|
7.7 | IC50 | 3 | — | |
HOFGFUOFMADIHI
|
7.7 | IC50 | 3 | — | |
KTUFNOKKBVMGRW
|
7.7 | Kd | 38 | Yes | |
MMVLETOTGHDVPQ
|
7.7 | IC50 | 7 | — | |
ZWIVMZNSHMYADK
|
7.7 | IC50 | 3 | — | |
NXFPMDWYDKHFMM
|
7.7 | IC50 | 2 | — | |
CLNJNVQBKCEOLA
|
7.7 | IC50 | 3 | — | |
DYSDUQPAIATDAA
|
7.7 | IC50 | 5 | Yes | |
GHPFSYCYZJKVDZ
|
7.7 | Ki | 18 | Yes | |
KBCISYCUHRRWQT
|
7.7 | IC50 | 2 | — | |
KKYPRNBBPBRJQX
|
7.7 | Ki | 40 | — | |
PTVPBWWDGZSEAF
|
7.7 | Ki | 63 | — | |
PYXQMJSGJIJHJT
|
7.7 | Ki | 28 | — | |
QZXMREJVHYOFOD
|
7.7 | IC50 | 2 | — | |
WUBFAXNVDMCVIO
|
7.7 | IC50 | 12 | Yes | |
WUWDLXZGHZSWQZ
|
7.7 | Ki | 41 | — | |
PCXFPRAKEYSDMS
|
7.7 | IC50 | 2 | — | |
RITAVMQDGBJQJZ
|
7.7 | Kd | 43 | — | |
TXAFYFWHBVJGHQ
|
7.7 | IC50 | 2 | — | |
PUHKAOLWMGXVFS
|
7.7 | IC50 | 3 | — | |
YMNHISNDWVXKND
|
7.7 | IC50 | 3 | — | |
BPMAUJVZZZYXDV
|
7.6 | IC50 | 3 | — | |
BQPLWJRDSDNGNE
|
7.6 | Ki | 16 | — | |
DOLVPVSWTLFZMQ
|
7.6 | Ki | 17 | — | |
HIVVRJXSFJMYEH
|
7.6 | IC50 | 3 | — | |
ITDDDMFXMSWPBU
|
7.6 | IC50 | 3 | — | |
JHWZPTAZWZKCEQ
|
7.6 | IC50 | 5 | — | |
KWSZYBNXNYRQCC
|
7.6 | Ki | 21 | — | |
OEQLJMGIZHYYCW
|
7.6 | IC50 | 3 | — | |
OTVCFDOYUHREFJ
|
7.6 | Ki | 26 | — | |
QKBGNVCABCTNCY
|
7.6 | IC50 | 3 | — | |
SEVCBWKJSOLMNQ
|
7.6 | Ki | 38 | — | |
VMOVZKURWYNTLN
|
7.6 | Ki | 7 | — |