Target Details
| UniProt AC | P07333 |
|---|---|
| Gene Symbol | CSF1R |
| Protein Name | Macrophage colony-stimulating factor 1 receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00047 (ig) PF25305 (Ig_PDGFR_d4) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 896
- Clinical molecules 90
- Avg pChEMBL 7.53
KEGG Pathways (11)
- Acute myeloid leukemia
- Cytokine-cytokine receptor interaction
- Hematopoietic cell lineage
- MAPK signaling pathway
- Osteoclast differentiation
- PI3K-Akt signaling pathway
- Pathways in cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Transcriptional misregulation in cancer
- Viral protein interaction with cytokine and cytokine receptor
Associated Diseases (3)
Active Molecules (896)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XLUQUKJVLXWCSN
|
8.0 | IC50 | 2 | — | |
XQGUIRKPWAXDLW
|
8.0 | IC50 | 4 | — | |
YDOPLCNFRXOHCC
|
8.0 | Ki | 28 | — | |
ZELLDMQPTIPJQD
|
8.0 | IC50 | 2 | — | |
AUFWLXVVSPEREI
|
8.0 | IC50 | 3 | — | |
XJXFROJLWMLVQH
|
8.0 | IC50 | 2 | — | |
VKBFHTIUXUCYRQ
|
8.0 | Ki | 66 | — | |
ZJIRIQBCHHNGDO
|
7.9 | IC50 | 2 | — | |
BMEXIUCHJUGPRB
|
7.9 | IC50 | 2 | — | |
JFFNMSINEFWPKX
|
7.9 | IC50 | 2 | — | |
BMBZCEYEGICFNU
|
7.9 | IC50 | 3 | — | |
CVWXJKQAOSCOAB
|
7.9 | Kd | 35 | — | |
GFIAEVSQQPXMCV
|
7.9 | IC50 | 2 | — | |
GTWNQGXKDRADED
|
7.9 | IC50 | 2 | — | |
HKSZLNNOFSGOKW
|
7.9 | Kd | 213 | — | |
HXZURUMJDIMZJI
|
7.9 | IC50 | 3 | — | |
KMYBTZOVMXFXAU
|
7.9 | IC50 | 3 | — | |
XLFNLJYGUOLEJS
|
7.9 | IC50 | 26 | — | |
APUCFXHENVUXCY
|
7.9 | Ki | 15 | — | |
FLEAYYMORDPWAJ
|
7.9 | Ki | 90 | — | |
MFVOIPKDSOFMQO
|
7.9 | IC50 | 3 | — | |
NRGYZNJPCGRCLV
|
7.9 | Ki | 52 | — | |
XOOAAYRIVATZNM
|
7.9 | Ki | 55 | — | |
ADLRDDWBCKMWCY
|
7.9 | IC50 | 3 | — | |
JGWRKYUXBBNENE
|
7.9 | IC50 | 11 | — | |
JVLYHJYNLHAPID
|
7.9 | IC50 | 3 | — | |
MFVOIPKDSOFMQO
|
7.9 | IC50 | 3 | — | |
NFYFLWXBIHYPII
|
7.9 | IC50 | 3 | — | |
XOTYCWCEXOJPBF
|
7.9 | IC50 | 3 | — | |
XXJWYDDUDKYVKI
|
7.9 | Kd | 52 | — | |
DZKMAWNYSJECKX
|
7.8 | IC50 | 12 | — | |
IWPVUHHCWGVPNJ
|
7.8 | IC50 | 5 | Yes | |
LTTJGQBDGMNWHJ
|
7.8 | IC50 | 2 | — | |
NDEXUOWTGYUVGA
|
7.8 | IC50 | 12 | — | |
OLZDZYHEIBZXCI
|
7.8 | IC50 | 2 | — | |
RTWJZWFAMFOLDK
|
7.8 | IC50 | 2 | — | |
RGBMULROFDMOBL
|
7.8 | IC50 | 3 | — | |
AYKPYAOQPANRFS
|
7.8 | IC50 | 3 | — | |
CHZKEAYTNKCUEF
|
7.8 | IC50 | 2 | — | |
FAYAUAZLLLJJGH
|
7.8 | IC50 | 36 | Yes | |
VLHUMLSNFMCPFI
|
7.8 | IC50 | 3 | — | |
YWTXHHRPNVQPIM
|
7.8 | IC50 | 3 | — | |
AYXVSCVVQIADBF
|
7.8 | Ki | 10 | — | |
CQBBMNXXVMOFCA
|
7.8 | Ki | 39 | — | |
FDVSOQRNTAPCHB
|
7.8 | Ki | 40 | — | |
GSRHFOYGPWJXII
|
7.8 | IC50 | 2 | — | |
IIJKGBMUSGQZJO
|
7.8 | IC50 | 3 | — | |
JKZZCHSVFXZBAI
|
7.8 | IC50 | 6 | — | |
KTQYQHLIMZOBSM
|
7.8 | Ki | 12 | — | |
LCGSWTFWYNYUKS
|
7.8 | Ki | 26 | — |