Target Details
| UniProt AC | P07333 |
|---|---|
| Gene Symbol | CSF1R |
| Protein Name | Macrophage colony-stimulating factor 1 receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00047 (ig) PF25305 (Ig_PDGFR_d4) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 896
- Clinical molecules 90
- Avg pChEMBL 7.53
KEGG Pathways (11)
- Acute myeloid leukemia
- Cytokine-cytokine receptor interaction
- Hematopoietic cell lineage
- MAPK signaling pathway
- Osteoclast differentiation
- PI3K-Akt signaling pathway
- Pathways in cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Transcriptional misregulation in cancer
- Viral protein interaction with cytokine and cytokine receptor
Associated Diseases (3)
Active Molecules (896)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BVOWDAQJDDEQSR
|
8.2 | IC50 | 3 | — | |
JUNWLAORTWKJOM
|
8.2 | IC50 | 3 | — | |
PKVRKFYLJXIDJS
|
8.2 | IC50 | 3 | — | |
UFOSAOVNENJKCZ
|
8.2 | IC50 | 3 | — | |
VCLCQJKIOXPDMP
|
8.2 | IC50 | 3 | — | |
WJEOLQLKVOPQFV
|
8.1 | Kd | 24 | — | |
IYPXGGXWYCGJCN
|
8.1 | IC50 | 2 | — | |
ADLPKFFMGIJZIM
|
8.1 | IC50 | 44 | — | |
CUIHSIWYWATEQL
|
8.1 | Kd | 61 | Yes | |
GMUVHXBIPOWLCK
|
8.1 | IC50 | 3 | — | |
GSXRCPJTNIGKSZ
|
8.1 | Ki | 43 | — | |
HKSZLNNOFSGOKW
|
8.1 | Ki | 118 | — | |
HKZKELVPGXJIMW
|
8.1 | Ki | 41 | — | |
JPKSISIJPSXDLA
|
8.1 | IC50 | 10 | Yes | |
TTZAURANQVEMPE
|
8.1 | IC50 | 4 | — | |
VIEKBHGPZROLOI
|
8.1 | IC50 | 3 | — | |
VOJMTTDUYUMNNZ
|
8.1 | IC50 | 3 | — | |
VPDYUDURNXPNMA
|
8.1 | IC50 | 5 | Yes | |
XKZINYYXWJEYEL
|
8.1 | Ki | 37 | — | |
IQKPWLCHWJCSLF
|
8.1 | IC50 | 2 | — | |
JMGCDJNFHYFXDK
|
8.1 | IC50 | 2 | — | |
PUIXMSRTTHLNKI
|
8.1 | IC50 | 12 | — | |
ACFWCPZFEIDRAM
|
8.1 | IC50 | 2 | — | |
BCDAHFZFGKOCPG
|
8.1 | IC50 | 4 | — | |
PHXJVRSECIGDHY
|
8.1 | IC50 | 59 | — | |
YRUDYNCGPZHXRB
|
8.1 | Kd | 6 | — | |
DKNUPRMJNUQNHR
|
8.1 | Kd | 33 | — | |
QAQWRVQXBRITDM
|
8.1 | IC50 | 4 | — | |
UGNXBDMIUNXKPM
|
8.1 | IC50 | 3 | — | |
UVNBMNWTGOQKQF
|
8.1 | IC50 | 8 | Yes | |
VMBRRMNXXVZGCB
|
8.1 | IC50 | 2 | — | |
WPXVVAWAHQHJPF
|
8.1 | IC50 | 41 | — | |
JGHJSVPEMJVPKE
|
8.0 | IC50 | 2 | — | |
HYTINAIANCXBTN
|
8.0 | IC50 | 2 | — | |
BNVPFDRNGHMRJS
|
8.0 | IC50 | 3 | — | |
DZFZXPPHBWCXPQ
|
8.0 | IC50 | 12 | — | |
JBPWJPNLAGHYOY
|
8.0 | IC50 | 2 | — | |
JGFZPZGREYNUPH
|
8.0 | IC50 | 5 | Yes | |
KAPMKULMYGROOA
|
8.0 | IC50 | 2 | — | |
KVCQTKNUUQOELD
|
8.0 | IC50 | 6 | — | |
LGHBDVLAHHANMX
|
8.0 | Ki | 53 | — | |
LKPIGXCNFCFRED
|
8.0 | IC50 | 3 | — | |
LVECPYVAIBNSRV
|
8.0 | Ki | 33 | — | |
MKPUNAONBMYMOE
|
8.0 | IC50 | 2 | — | |
MQRDVGBWWVWMEN
|
8.0 | Ki | 47 | — | |
MUDZWVCKAOGYGL
|
8.0 | IC50 | 2 | — | |
OEUMLQMTMOCCGW
|
8.0 | Kd | 6 | — | |
OZIZBAWFMYRHDD
|
8.0 | IC50 | 3 | — | |
RBXYGQNZRVPDNB
|
8.0 | Ki | 34 | — | |
VCFDMLBPASGZTP
|
8.0 | Ki | 38 | — |