Target Details
| UniProt AC | P07333 |
|---|---|
| Gene Symbol | CSF1R |
| Protein Name | Macrophage colony-stimulating factor 1 receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00047 (ig) PF25305 (Ig_PDGFR_d4) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 896
- Clinical molecules 90
- Avg pChEMBL 7.53
KEGG Pathways (11)
- Acute myeloid leukemia
- Cytokine-cytokine receptor interaction
- Hematopoietic cell lineage
- MAPK signaling pathway
- Osteoclast differentiation
- PI3K-Akt signaling pathway
- Pathways in cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Transcriptional misregulation in cancer
- Viral protein interaction with cytokine and cytokine receptor
Associated Diseases (3)
Active Molecules (896)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HGOSXKUMUKYUKG
|
8.3 | IC50 | 3 | — | |
KSSUPGRPFLARDM
|
8.3 | IC50 | 2 | — | |
HKIJOVMUJUDWGI
|
8.3 | IC50 | 4 | — | |
XUJIISUKTLKCLK
|
8.3 | IC50 | 3 | — | |
QJJXDLUIDBRYRG
|
8.3 | IC50 | 3 | — | |
UXXQOJXBIDBUAC
|
8.3 | Kd | 21 | Yes | |
YBJQFWOWWBZCJS
|
8.3 | Kd | 2 | — | |
AMHUBFWCCMLLCJ
|
8.3 | IC50 | 15 | — | |
AYJBHLUSGLQYDG
|
8.3 | Ki | 16 | — | |
BIKYDWLMTPRSQL
|
8.3 | Ki | 50 | — | |
BYKOKZMCLVWDCZ
|
8.3 | IC50 | 3 | — | |
CJXUHPRULWSPBE
|
8.3 | IC50 | 7 | — | |
FHMPZYDTSRUDTD
|
8.3 | IC50 | 3 | — | |
GJKVMXDBPDDFHI
|
8.3 | Ki | 27 | — | |
GUYRCSVNTIHWAI
|
8.3 | IC50 | 3 | — | |
INFXGMKRYCEOFJ
|
8.3 | IC50 | 4 | — | |
JNXJKTXDSPWNRP
|
8.3 | Ki | 30 | — | |
KDCGROMZSUCCMF
|
8.3 | IC50 | 3 | — | |
NKEUPUJTVALZIK
|
8.3 | Ki | 28 | — | |
OFGUFFNSCXNTNV
|
8.3 | IC50 | 4 | — | |
OIZJENLXXROKNH
|
8.3 | IC50 | 3 | — | |
PMAXBYMGMQSUFK
|
8.3 | IC50 | 3 | — | |
POVOYMIAJXXYSA
|
8.3 | IC50 | 3 | — | |
QGYZTXJGBDCZHX
|
8.3 | IC50 | 3 | — | |
SFPWNTQWFFNJIH
|
8.3 | Ki | 48 | — | |
SHPFDGWALWEPGS
|
8.3 | IC50 | 35 | — | |
UXQLMVSZSYZFID
|
8.3 | Ki | 12 | — | |
XIXBPLMTEROWPD
|
8.3 | IC50 | 3 | — | |
WIAYJYJAAXMOLH
|
8.3 | IC50 | 3 | — | |
MPDAYIPCEWJKOY
|
8.3 | IC50 | 4 | — | |
LVMAULGVWBINFP
|
8.3 | IC50 | 6 | — | |
RAHBGWKEPAQNFF
|
8.2 | Kd | 26 | — | |
VKBFHTIUXUCYRQ
|
8.2 | IC50 | 8 | — | |
ODPGGGTTYSGTGO
|
8.2 | Kd | 153 | — | |
FQXQXOYNTXHBKK
|
8.2 | IC50 | 7 | — | |
MLFZJIDNGFABRH
|
8.2 | IC50 | 3 | — | |
BTSSYEBPODNPPC
|
8.2 | IC50 | 3 | — | |
GTADZVOESZXMOQ
|
8.2 | IC50 | 3 | — | |
RNSPJNIKRAJKOU
|
8.2 | IC50 | 2 | — | |
DTKVEGSQVRWLEQ
|
8.2 | Kd | 2 | — | |
HBWUNGZZOZIRLQ
|
8.2 | IC50 | 2 | — | |
INURPMRKCUUSHP
|
8.2 | IC50 | 2 | — | |
QGLUQQCIZIEJHF
|
8.2 | IC50 | 2 | — | |
XOSIKVLXVWWHON
|
8.2 | IC50 | 3 | — | |
FJZXDUKUMALHNP
|
8.2 | Ki | 10 | — | |
GMYYMEOGFRKSFS
|
8.2 | Ki | 29 | — | |
UOOZSMNSBYVUGZ
|
8.2 | Ki | 32 | — | |
UXMNYFJHEBEDJS
|
8.2 | Ki | 19 | Yes | |
CANPTKDXQQAVKO
|
8.2 | IC50 | 2 | — | |
GMHSCMWFLYBPIU
|
8.2 | IC50 | 3 | — |