Target Details
| UniProt AC | P07333 |
|---|---|
| Gene Symbol | CSF1R |
| Protein Name | Macrophage colony-stimulating factor 1 receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00047 (ig) PF25305 (Ig_PDGFR_d4) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 896
- Clinical molecules 90
- Avg pChEMBL 7.53
KEGG Pathways (11)
- Acute myeloid leukemia
- Cytokine-cytokine receptor interaction
- Hematopoietic cell lineage
- MAPK signaling pathway
- Osteoclast differentiation
- PI3K-Akt signaling pathway
- Pathways in cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Transcriptional misregulation in cancer
- Viral protein interaction with cytokine and cytokine receptor
Associated Diseases (3)
Active Molecules (896)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VRIWWBXFSKWVDK
|
8.5 | IC50 | 3 | — | |
FVXFEJBGHYVGML
|
8.5 | Kd | 2 | — | |
HKSZLNNOFSGOKW
|
8.5 | IC50 | 408 | — | |
FGSVLADZCDNNOC
|
8.5 | Ki | 11 | — | |
RAPYFGJGASETOS
|
8.5 | Ki | 11 | — | |
RKLGMDOZEOTQEM
|
8.5 | Ki | 12 | — | |
ULHGAQSVFPOUDY
|
8.5 | Ki | 43 | — | |
UTQPKPHUIMHAAN
|
8.5 | Ki | 22 | — | |
XBYVOPRDASFDMY
|
8.5 | Ki | 42 | — | |
XHORJSJFHVABEA
|
8.5 | Ki | 5 | — | |
XHORJSJFHVABEA
|
8.5 | Ki | 49 | — | |
ZXYVWKYLUPYZGL
|
8.5 | IC50 | 5 | — | |
WPHKIQPVPYJNAX
|
8.5 | IC50 | 81 | — | |
XPBJIFLFRWUBPO
|
8.5 | IC50 | 3 | — | |
HKYNFPUDKGPKDB
|
8.5 | IC50 | 2 | — | |
LYADGAGFYYXXIO
|
8.5 | IC50 | 82 | — | |
DVPCNIKFABUUTG
|
8.5 | Kd | 2 | — | |
MPVGZUGXCQEXTM
|
8.5 | IC50 | 61 | Yes | |
QYCFHBDOJSLVRL
|
8.5 | IC50 | 5 | — | |
PPOKAKSETFBBEQ
|
8.5 | IC50 | 2 | — | |
SREKLVZBGOOWFZ
|
8.5 | IC50 | 2 | — | |
CTNPALGJUAXMMC
|
8.4 | Kd | 151 | — | |
KXUSCHVJJBSONI
|
8.4 | IC50 | 2 | — | |
OKHZIVXQKINVAO
|
8.4 | IC50 | 4 | — | |
ZHOQUFGTKOHQBB
|
8.4 | IC50 | 2 | — | |
ZXAMVJNNDJRGFG
|
8.4 | IC50 | 4 | — | |
AMZWYWQCAVGQIH
|
8.4 | IC50 | 3 | — | |
QNXOYMFBIACDSL
|
8.4 | IC50 | 5 | — | |
INOASWZOZPQAQM
|
8.4 | IC50 | 5 | — | |
NCPIMEOPSFOWKB
|
8.4 | IC50 | 4 | — | |
YXARVHZXTQVAOP
|
8.4 | IC50 | 11 | — | |
BRTHUECZMVKNMQ
|
8.4 | Ki | 31 | — | |
DIGOSQFGMNNGOP
|
8.4 | IC50 | 3 | — | |
DLPARMNJOHFOLU
|
8.4 | Ki | 14 | Yes | |
HZIZEKOMOILAJT
|
8.4 | IC50 | 6 | Yes | |
IYCITBYBDPSBBJ
|
8.4 | IC50 | 6 | — | |
JAMUFNNBMXMUIC
|
8.4 | IC50 | 3 | — | |
KHYVUPSEVVSFJS
|
8.4 | IC50 | 2 | — | |
KNACLJBHKVSTDL
|
8.4 | Ki | 40 | — | |
RPDVCUCXMGWTFA
|
8.4 | Ki | 10 | — | |
SGBCJLVNLGNYBT
|
8.4 | IC50 | 3 | — | |
SPMHGQZFMNZCBV
|
8.4 | Ki | 30 | Yes | |
SXAVOOSGLYHVJW
|
8.4 | IC50 | 4 | — | |
VDPIYNSZQSYYGQ
|
8.4 | IC50 | 5 | — | |
XNEPVLVYFUGJLF
|
8.4 | Ki | 27 | — | |
JVCWPUFNLFSKFS
|
8.4 | IC50 | 5 | — | |
WYLCQKJYTVNVCY
|
8.4 | IC50 | 2 | — | |
WMWHVTDZNIVNIE
|
8.4 | IC50 | 9 | — | |
WMWHVTDZNIVNIE
|
8.4 | IC50 | 9 | — | |
BGVQPQHIUOTLBT
|
8.4 | Kd | 6 | — |