Target Details
| UniProt AC | P07333 |
|---|---|
| Gene Symbol | CSF1R |
| Protein Name | Macrophage colony-stimulating factor 1 receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00047 (ig) PF25305 (Ig_PDGFR_d4) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 896
- Clinical molecules 90
- Avg pChEMBL 7.53
KEGG Pathways (11)
- Acute myeloid leukemia
- Cytokine-cytokine receptor interaction
- Hematopoietic cell lineage
- MAPK signaling pathway
- Osteoclast differentiation
- PI3K-Akt signaling pathway
- Pathways in cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Transcriptional misregulation in cancer
- Viral protein interaction with cytokine and cytokine receptor
Associated Diseases (3)
Active Molecules (896)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VZBIYJBIGRPSOL
|
8.7 | IC50 | 2 | — | |
XEJIAICXFVLKKE
|
8.7 | IC50 | 2 | — | |
XEWYVOAMYRLGMQ
|
8.7 | IC50 | 3 | — | |
YERPHLXVKKTPGK
|
8.7 | IC50 | 2 | — | |
ZCCJKVBTHCOISJ
|
8.7 | Ki | 46 | — | |
HPOCEHFOBYUUJL
|
8.7 | IC50 | 4 | Yes | |
OGRZTQUEBSXDJP
|
8.7 | IC50 | 2 | — | |
QXSDNFDJBVZWQV
|
8.7 | IC50 | 2 | — | |
VXYBEIXZJGRJPA
|
8.7 | IC50 | 2 | — | |
NGKALCMOLVCFHL
|
8.7 | IC50 | 5 | — | |
DZGGGZSDTNTLQN
|
8.7 | IC50 | 5 | Yes | |
QCSPHKYKAODHGS
|
8.7 | IC50 | 3 | — | |
UKGCAEYEQULSSN
|
8.7 | IC50 | 2 | — | |
WDTMMWXYUKMGGU
|
8.6 | Kd | 2 | — | |
GVFQHBBRWBJGNU
|
8.6 | IC50 | 5 | — | |
QPFCHPRFMFYYAG
|
8.6 | IC50 | 2 | — | |
DZSUJUOJJJCWGG
|
8.6 | IC50 | 55 | Yes | |
CJOKUBRCAVWYRX
|
8.6 | IC50 | 4 | Yes | |
FHMFHOQHUFKWBK
|
8.6 | IC50 | 3 | — | |
KLHJDCUHOKZNOP
|
8.6 | IC50 | 5 | Yes | |
KROLCVQARUUHNV
|
8.6 | Ki | 12 | — | |
KTRYEZRTYBBSHL
|
8.6 | IC50 | 3 | — | |
KUNZDWIFPOMUOX
|
8.6 | Ki | 36 | — | |
MHCPAORAYMTGCZ
|
8.6 | Ki | 37 | — | |
PJSBFZAYJQMORO
|
8.6 | Ki | 11 | — | |
RTYJMUXLFRYRBU
|
8.6 | Ki | 35 | — | |
WINHZLLDWRZWRT
|
8.6 | Ki | 66 | — | |
YEQZZLYGLQFEAM
|
8.6 | IC50 | 3 | — | |
YWCKVLPHEKWBJP
|
8.6 | IC50 | 3 | — | |
BDVSEKHVPXXJRI
|
8.6 | IC50 | 3 | — | |
PSWOVPWZYVUKKW
|
8.6 | IC50 | 2 | — | |
ORYMWWSJZRCUSV
|
8.6 | IC50 | 7 | — | |
UGEJLCNSVIVALC
|
8.6 | IC50 | 41 | — | |
BPKVTDLMFZLJIM
|
8.6 | IC50 | 2 | — | |
CIQLUWGXRPQJFF
|
8.6 | IC50 | 2 | — | |
YESKHRZGFKDGEH
|
8.6 | IC50 | 3 | — | |
OMVAYCDDPIHBDR
|
8.5 | IC50 | 5 | — | |
PABZNWOXICIOPN
|
8.5 | IC50 | 2 | — | |
BAEPKCSJXVFDDR
|
8.5 | Kd | 2 | — | |
KFDMABXQUQMQTQ
|
8.5 | IC50 | 3 | — | |
LYHXSDWIWVVZPB
|
8.5 | IC50 | 6 | Yes | |
NDZHXVIMTDMQGZ
|
8.5 | IC50 | 4 | — | |
QHFNVZMOKIFBBE
|
8.5 | IC50 | 3 | — | |
RAVQVOSIVIEHCN
|
8.5 | IC50 | 3 | — | |
RFSFIDGEFVXSQM
|
8.5 | IC50 | 12 | Yes | |
TVGAHWWPABTBCX
|
8.5 | IC50 | 3 | — | |
TVUFMDRGVRGPIS
|
8.5 | IC50 | 3 | — | |
TWRNOCZDGWHEGC
|
8.5 | IC50 | 3 | — | |
UPQKBKLECVIXJR
|
8.5 | IC50 | 12 | — | |
USQDNKJTXHBZRC
|
8.5 | IC50 | 3 | — |