Target Details
| UniProt AC | P07333 |
|---|---|
| Gene Symbol | CSF1R |
| Protein Name | Macrophage colony-stimulating factor 1 receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00047 (ig) PF25305 (Ig_PDGFR_d4) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 896
- Clinical molecules 90
- Avg pChEMBL 7.53
KEGG Pathways (11)
- Acute myeloid leukemia
- Cytokine-cytokine receptor interaction
- Hematopoietic cell lineage
- MAPK signaling pathway
- Osteoclast differentiation
- PI3K-Akt signaling pathway
- Pathways in cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Transcriptional misregulation in cancer
- Viral protein interaction with cytokine and cytokine receptor
Associated Diseases (3)
Active Molecules (896)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DKIXPZZJZUEUGI
|
8.9 | IC50 | 3 | — | |
FGOGRVVUAJAJDC
|
8.9 | Kd | 2 | — | |
LPSHFMAZVFWNPX
|
8.9 | IC50 | 2 | — | |
SXHIZYRFWJFSEN
|
8.9 | IC50 | 2 | — | |
AZTMYWWWILJAKW
|
8.9 | Ki | 16 | Yes | |
QAKMQVCMEPKBHL
|
8.9 | Ki | 11 | — | |
ZQQVWTACALNOAJ
|
8.9 | Ki | 11 | — | |
BHXZFEQWQQPISU
|
8.9 | Kd | 2 | — | |
MWSYDGNFQSXUAU
|
8.9 | IC50 | 2 | — | |
RPSRSUPHEANJKD
|
8.9 | IC50 | 2 | — | |
ZSVFWIDDNJEWEB
|
8.9 | IC50 | 2 | — | |
KVBFMJDTLAIVSN
|
8.9 | IC50 | 2 | — | |
BRTHUECZMVKNMQ
|
8.9 | IC50 | 7 | — | |
KRCPKGPVOUOHOW
|
8.8 | IC50 | 3 | — | |
NGKALCMOLVCFHL
|
8.8 | IC50 | 5 | — | |
UURBEBBVEFUFRK
|
8.8 | IC50 | 2 | — | |
NGKALCMOLVCFHL
|
8.8 | IC50 | 5 | — | |
AYTDCXHHGYDWLU
|
8.8 | IC50 | 3 | — | |
SPZDCHRXPBSIHM
|
8.8 | IC50 | 6 | — | |
ZNXXPZKXDKVVIC
|
8.8 | IC50 | 2 | — | |
DBXOMQJZSQLQED
|
8.8 | Ki | 12 | — | |
KNARVZUUCLIBGV
|
8.8 | Ki | 33 | — | |
MCCCQFAOMZMZKE
|
8.8 | Ki | 52 | — | |
QDOBTYVGPGFRCM
|
8.8 | Ki | 11 | — | |
QKFZNOQWHCBRSM
|
8.8 | Kd | 2 | — | |
SJMFZIGFOIPNPE
|
8.8 | Ki | 10 | — | |
YHNSOVKRVXWDLY
|
8.8 | IC50 | 2 | — | |
LCNJPGQTVUJHBZ
|
8.8 | IC50 | 2 | — | |
MUHWRSWKWURVPP
|
8.8 | IC50 | 2 | — | |
CXQHYVUVSFXTMY
|
8.7 | Kd | 154 | — | |
PBNPHBXRMOAALS
|
8.7 | Kd | 2 | — | |
PSABAQPTDYJLPZ
|
8.7 | Kd | 2 | — | |
SEJGTFPOEJWEGG
|
8.7 | Kd | 149 | — | |
NIPQEVVSMAZUMD
|
8.7 | IC50 | 2 | — | |
CXVBPWYIUWZVJO
|
8.7 | IC50 | 4 | — | |
FTWLELHFVFNVSG
|
8.7 | IC50 | 3 | — | |
GDEJPGKNPRJNGE
|
8.7 | Ki | 6 | — | |
GEGCXGMFUYJULA
|
8.7 | IC50 | 30 | Yes | |
GWMATETWMAQOFL
|
8.7 | Ki | 36 | — | |
HBHOKIDZSIYNGE
|
8.7 | Ki | 3 | — | |
HVRWZFQFSQUILC
|
8.7 | IC50 | 4 | — | |
KZVIZFHCMVWFNT
|
8.7 | IC50 | 7 | — | |
MTCHBJMHQSHCIK
|
8.7 | IC50 | 3 | — | |
MZPQDMUNWXBKLC
|
8.7 | IC50 | 3 | — | |
NSKFXNDKPCVDIN
|
8.7 | Ki | 12 | — | |
NXRSAGDKLSDJBW
|
8.7 | IC50 | 3 | — | |
OIANGKGOYKDGQV
|
8.7 | IC50 | 10 | — | |
OZFHIGAKHHLPEF
|
8.7 | IC50 | 3 | — | |
PEJCGJUJBCLDFV
|
8.7 | Kd | 2 | — | |
PMTYXROLPZFSKY
|
8.7 | IC50 | 3 | — |