Target Details
| UniProt AC | P07333 |
|---|---|
| Gene Symbol | CSF1R |
| Protein Name | Macrophage colony-stimulating factor 1 receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00047 (ig) PF25305 (Ig_PDGFR_d4) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 896
- Clinical molecules 90
- Avg pChEMBL 7.53
KEGG Pathways (11)
- Acute myeloid leukemia
- Cytokine-cytokine receptor interaction
- Hematopoietic cell lineage
- MAPK signaling pathway
- Osteoclast differentiation
- PI3K-Akt signaling pathway
- Pathways in cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Transcriptional misregulation in cancer
- Viral protein interaction with cytokine and cytokine receptor
Associated Diseases (3)
Active Molecules (896)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OIQFBHIJWBNDKU
|
9.5 | IC50 | 2 | — | |
LYHDXABKNJMNEZ
|
9.5 | Ki | 10 | — | |
UUVMNPKFPGJBNX
|
9.5 | Ki | 10 | — | |
FIJWNTPHEHDJQG
|
9.4 | IC50 | 6 | Yes | |
HDUIQNARVJYUGR
|
9.4 | IC50 | 2 | — | |
HNJOCLQAHHIZPS
|
9.4 | IC50 | 2 | — | |
YMMVVFFRNSLEMO
|
9.4 | IC50 | 2 | — | |
LJWVFWLHDDCALO
|
9.4 | IC50 | 3 | — | |
WOHPNZFTBWWWBX
|
9.3 | IC50 | 2 | — | |
XSZHYGYAHGNIKV
|
9.3 | IC50 | 2 | — | |
ZBNZXTGUTAYRHI
|
9.2 | IC50 | 102 | Yes | |
LIFJGDQDPHYFQJ
|
9.2 | Kd | 2 | — | |
DEPRXLRJLFPMSV
|
9.2 | IC50 | 2 | — | |
DMTDZFGYURLLKX
|
9.2 | Ki | 13 | Yes | |
FOONBYIHFUMRSX
|
9.2 | Ki | 12 | — | |
IFPPYSWJNWHOLQ
|
9.2 | Ki | 52 | Yes | |
FOWKLHQOYBAAQY
|
9.2 | IC50 | 2 | — | |
LDFNWQUVEYWFOH
|
9.2 | IC50 | 3 | — | |
VAARYSWULJUGST
|
9.2 | Kd | 119 | Yes | |
GUBJNPWVIUFSTR
|
9.2 | IC50 | 103 | — | |
AWROSJBGNHPYIE
|
9.2 | IC50 | 2 | — | |
IUQURQCHOSRPJM
|
9.2 | IC50 | 4 | Yes | |
YKNNKGNQGPFRTQ
|
9.2 | IC50 | 2 | — | |
UUDPUQDMSHQSKH
|
9.1 | IC50 | 3 | — | |
ZRBHOXZJRFQVDF
|
9.1 | IC50 | 2 | — | |
BDPBZUHWAVABDM
|
9.1 | Ki | 11 | — | |
CNWFAPYYHZIFRD
|
9.1 | IC50 | 2 | — | |
DXPSQKSTVIVZLV
|
9.1 | IC50 | 6 | Yes | |
HAEUZCCQUNTMLI
|
9.1 | IC50 | 2 | — | |
KVTCLWZZBAIUNQ
|
9.1 | IC50 | 2 | — | |
PLVJXCDUGVPNDW
|
9.1 | IC50 | 2 | — | |
FHPTWZJZWOYCKG
|
9.0 | IC50 | 5 | — | |
HQPNLIKXAPLWBQ
|
9.0 | Ki | 12 | Yes | |
KOTRVAMMDDKVHE
|
9.0 | IC50 | 2 | — | |
NCPGPVUTWKUPPM
|
9.0 | Kd | 2 | — | |
YEPNVBNYCRGZRX
|
9.0 | Ki | 26 | — | |
ZQGBDVIGTTVIFV
|
9.0 | IC50 | 3 | — | |
XPCQXAQALLRVJQ
|
9.0 | IC50 | 2 | — | |
ADZBMFGQQWPHMJ
|
9.0 | IC50 | 3 | — | |
MVPRWLBKNHWFPM
|
9.0 | IC50 | 6 | — | |
NLZDIXVVUFRBAV
|
9.0 | IC50 | 2 | — | |
NNMVDGFJIPMXNA
|
9.0 | IC50 | 2 | — | |
QPSVRPUGGFUWCH
|
9.0 | IC50 | 2 | — | |
QSGXWUVUDCSFIZ
|
9.0 | IC50 | 2 | — | |
ZDZWIYNKACEWQC
|
9.0 | IC50 | 3 | — | |
ULCJFJXVIGNWMX
|
8.9 | Kd | 2 | — | |
NGKALCMOLVCFHL
|
8.9 | IC50 | 5 | — | |
FMCLDFJJIAZKCA
|
8.9 | IC50 | 5 | — | |
VQINULODWGEVBB
|
8.9 | IC50 | 4 | — | |
CHLFFSKXUJQLQO
|
8.9 | IC50 | 7 | — |