Target Details
| UniProt AC | P07305 |
|---|---|
| Gene Symbol | H1-0 |
| Protein Name | Histone H1.0 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00538 (Linker_histone) |
Summary
- Multi-target molecules 8
- Clinical molecules 6
- Avg pChEMBL 7.64
Active Molecules (8)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QZUDBNBUXVUHMW
|
9.0 | Ki | 39 | Yes | |
KVWDHTXUZHCGIO
|
8.7 | Ki | 32 | Yes | |
URKOMYMAXPYINW
|
8.0 | Ki | 27 | Yes | |
RAPZEAPATHNIPO
|
7.8 | Ki | 28 | Yes | |
MVWVFYHBGMAFLY
|
7.8 | Ki | 31 | Yes | |
CEUORZQYGODEFX
|
7.5 | Ki | 31 | — | |
ZCCPLJOKGAACRT
|
6.1 | Kd | 599 | — | |
LNEPOXFFQSENCJ
|
6.1 | Ki | 33 | Yes |