Target Details
| UniProt AC | P06881 |
|---|---|
| Gene Symbol | CALCA |
| Protein Name | Calcitonin gene-related peptide 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00214 (Calc_CGRP_IAPP) |
Summary
- Multi-target molecules 12
- Clinical molecules 0
- Avg pChEMBL 8.69
Active Molecules (12)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ITIXDWVDFFXNEG
|
10.8 | Ki | 3 | — | |
AZAANWYREOQRFB
|
10.3 | IC50 | 3 | — | |
LVJLXLXVWDOXCC
|
9.7 | IC50 | 4 | — | |
DSMQHSCNENFKPV
|
9.1 | IC50 | 4 | — | |
RLKYTIXOYWIXQK
|
8.9 | IC50 | 4 | — | |
CGDZXLJGHVKVIE
|
8.9 | IC50 | 3 | — | |
VDLYRUOYUCCKKR
|
8.8 | IC50 | 4 | — | |
JNMYUIOIISURGX
|
8.7 | IC50 | 4 | — | |
JXTWPKPSAOKCLS
|
8.7 | IC50 | 4 | — | |
NDACAFBDTQIYCQ
|
8.3 | Ki | 4 | — | |
GUILBDPDYMIGBQ
|
6.1 | IC50 | 3 | — | |
HMXDWDSNPRNUKI
|
6.0 | Ki | 72 | — |