Target Details
| UniProt AC | P06870 |
|---|---|
| Gene Symbol | KLK1 |
| Protein Name | Kallikrein-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00089 (Trypsin) |
Summary
- Multi-target molecules 630
- Clinical molecules 0
- Avg pChEMBL 7.82
KEGG Pathways (2)
Active Molecules (630)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZGPLTWLOJCQFNY
|
7.5 | IC50 | 2 | — | |
PMILANWLXZUIMA
|
7.5 | Ki | 2 | — | |
YGBZFHXWPPQSHR
|
7.5 | Ki | 2 | — | |
BTDAJYRWGQUKHR
|
7.5 | IC50 | 2 | — | |
HKBSTFULNGWVHG
|
7.5 | IC50 | 2 | — | |
HKBSTFULNGWVHG
|
7.5 | IC50 | 2 | — | |
QDYFKRMDVOVQRF
|
7.5 | IC50 | 2 | — | |
GCYYRDQPBANMMK
|
7.5 | IC50 | 2 | — | |
MTGQBIHLRYXSAD
|
7.5 | IC50 | 3 | — | |
VCXPFNIRYFIASG
|
7.5 | IC50 | 2 | — | |
VLHZNIDQBGKPGY
|
7.5 | IC50 | 2 | — | |
WGCQTEXRPFWXEH
|
7.5 | IC50 | 2 | — | |
FDCBFBSFHLWFFU
|
7.5 | Ki | 6 | — | |
HWGUJACAWRDFKM
|
7.5 | IC50 | 2 | — | |
MCLDCXMFXNEDHA
|
7.5 | IC50 | 2 | — | |
YLICDVIPJRKVDF
|
7.5 | Ki | 4 | — | |
AHEIEXXGHCSZMY
|
7.5 | Ki | 4 | — | |
DEAVIHBHHLTWOF
|
7.5 | IC50 | 2 | — | |
HFNLRBFNQNHHQU
|
7.5 | Ki | 2 | — | |
JXQBMULDVDVTCD
|
7.5 | IC50 | 2 | — | |
DLQLOXULDLQSRU
|
7.5 | IC50 | 2 | — | |
MCLDCXMFXNEDHA
|
7.5 | IC50 | 2 | — | |
NQLCHVHYURZDNS
|
7.5 | IC50 | 2 | — | |
QHRMBTFZPZOACO
|
7.5 | IC50 | 2 | — | |
UBIGFKPKPJHBQK
|
7.5 | IC50 | 2 | — | |
UWSQVXSKTNKQNK
|
7.5 | IC50 | 2 | — | |
BAQNISDOFDTQKU
|
7.4 | IC50 | 2 | — | |
OYBWJNOXCFNTBV
|
7.4 | Ki | 3 | — | |
XSNJFJLMDHYDKD
|
7.4 | Ki | 2 | — | |
LTJPWZKTFQLBBF
|
7.4 | Ki | 2 | — | |
WGCNTVPWRMGTQZ
|
7.4 | Ki | 2 | — | |
ANHGWVXCHSOCLJ
|
7.4 | IC50 | 2 | — | |
JZJCSOJLMQSMFE
|
7.4 | IC50 | 2 | — | |
MUIZDSQZEXIWJW
|
7.4 | IC50 | 2 | — | |
CSWQJKHBMACTGB
|
7.4 | Ki | 6 | — | |
PVQODELEGLZOBK
|
7.4 | IC50 | 2 | — | |
YHFXCZDCIALUJO
|
7.4 | IC50 | 2 | — | |
DLQLOXULDLQSRU
|
7.4 | IC50 | 2 | — | |
RTPDDFLFZXREMW
|
7.4 | Ki | 3 | — | |
YWOOOSNQCNIOEJ
|
7.4 | IC50 | 2 | — | |
GCYYRDQPBANMMK
|
7.4 | IC50 | 2 | — | |
DEZHVNNZGNUIKF
|
7.3 | IC50 | 2 | — | |
DEZHVNNZGNUIKF
|
7.3 | IC50 | 2 | — | |
DJLOUHUQRVRYAZ
|
7.3 | IC50 | 2 | — | |
ZVQVAMLHDBSHQK
|
7.3 | IC50 | 2 | — | |
KPAYQIUVHCSBRE
|
7.3 | IC50 | 2 | — | |
VUNBMDNJNGUDCP
|
7.3 | IC50 | 2 | — | |
JFVFFRJAEQBBMJ
|
7.3 | Ki | 2 | — | |
KECBJDDHVPUGCU
|
7.3 | IC50 | 2 | — | |
HZIABZGYWLDYBC
|
7.3 | IC50 | 2 | — |