Target Details
| UniProt AC | P06870 |
|---|---|
| Gene Symbol | KLK1 |
| Protein Name | Kallikrein-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00089 (Trypsin) |
Summary
- Multi-target molecules 630
- Clinical molecules 0
- Avg pChEMBL 7.82
KEGG Pathways (2)
Active Molecules (630)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LXFPTSIBSQOGTO
|
7.7 | Ki | 3 | — | |
XKFNAKACSRLZKU
|
7.7 | IC50 | 2 | — | |
KECBJDDHVPUGCU
|
7.7 | IC50 | 2 | — | |
LYPVCWJWDVTCFK
|
7.7 | IC50 | 2 | — | |
KFSFQPNJQRTJEH
|
7.7 | IC50 | 2 | — | |
ODPYZUJUVLOFCY
|
7.7 | IC50 | 2 | — | |
VGKVWATXDPBYQQ
|
7.7 | Ki | 5 | — | |
JABFICNTUQQBIE
|
7.7 | IC50 | 2 | — | |
FIMUWRJHRVVZGD
|
7.7 | IC50 | 2 | — | |
MKBQOOYJFKTDGI
|
7.7 | IC50 | 2 | — | |
WDNZCVAWPKFSRF
|
7.7 | IC50 | 2 | — | |
WGWNPJIMCIPPBO
|
7.7 | Ki | 3 | — | |
NTWGGBXXPBSJIC
|
7.7 | IC50 | 2 | — | |
SEGFXDMGZGKYMG
|
7.7 | IC50 | 2 | — | |
BGHGZBOFLCOBHK
|
7.7 | IC50 | 2 | — | |
YEZYETGMGFHWLA
|
7.7 | IC50 | 2 | — | |
ZOWREHOVFWKKPQ
|
7.7 | Ki | 3 | — | |
KHTVBYNJIBMOOX
|
7.7 | Ki | 2 | — | |
ZOWDYXDKZSFHLH
|
7.7 | IC50 | 2 | — | |
JBLNWZHCAUHOQX
|
7.6 | IC50 | 2 | — | |
UWAQLEGUXYPPDC
|
7.6 | Ki | 3 | — | |
LTGICARJTJRTII
|
7.6 | IC50 | 2 | — | |
XRNVFLNSLRLZLB
|
7.6 | IC50 | 2 | — | |
HICIOVQYASGXKO
|
7.6 | IC50 | 2 | — | |
OJZAHFRHHUPVDA
|
7.6 | IC50 | 2 | — | |
BKXPNWHCZUBYGK
|
7.6 | Ki | 3 | — | |
CTKUOVDPJRFGAN
|
7.6 | IC50 | 2 | — | |
GRJIVWODHSGNKI
|
7.6 | IC50 | 2 | — | |
GRWUJZGBOOGLJA
|
7.6 | Ki | 2 | — | |
XQDFKGVDOCCXNS
|
7.6 | Ki | 3 | — | |
NLEPCGDWKIOUSP
|
7.6 | IC50 | 2 | — | |
OVKAPAFXRFWCLH
|
7.6 | IC50 | 2 | — | |
ZTGVBPABLQSRRO
|
7.6 | IC50 | 2 | — | |
CZNQRPCHDCYEPE
|
7.6 | Ki | 2 | — | |
MDHOLYLQXDWVOL
|
7.6 | Ki | 2 | — | |
OBTZRXJTWBMLKC
|
7.6 | Ki | 2 | — | |
VLHZNIDQBGKPGY
|
7.6 | IC50 | 2 | — | |
CFEHXUZXBTXUED
|
7.6 | IC50 | 2 | — | |
FZNUIBFUDXMFEC
|
7.6 | IC50 | 2 | — | |
PNOQSIVRNAIHEJ
|
7.6 | IC50 | 2 | — | |
DOEBANVVBVEAGV
|
7.6 | IC50 | 2 | — | |
NJTXCIYFJHGMJY
|
7.6 | IC50 | 2 | — | |
QZBWFIPTDPIYOH
|
7.6 | IC50 | 2 | — | |
ZNCHPQBFEAYPQI
|
7.6 | IC50 | 2 | — | |
NWFCFQJZLKVYCI
|
7.5 | IC50 | 2 | — | |
AXUFUQJDGXDVQN
|
7.5 | IC50 | 2 | — | |
AZCXDHIGSFNGSP
|
7.5 | IC50 | 2 | — | |
VEMPKZWOJHZWAA
|
7.5 | IC50 | 2 | — | |
ZBFGRVUPGJGBJH
|
7.5 | Ki | 2 | — | |
ZZLLSJIHRSANMJ
|
7.5 | IC50 | 2 | — |