Target Details
| UniProt AC | P06870 |
|---|---|
| Gene Symbol | KLK1 |
| Protein Name | Kallikrein-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00089 (Trypsin) |
Summary
- Multi-target molecules 630
- Clinical molecules 0
- Avg pChEMBL 7.82
KEGG Pathways (2)
Active Molecules (630)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HTHLQXUFXYHTMY
|
7.9 | IC50 | 2 | — | |
NQZSLHCRCYIUAY
|
7.9 | IC50 | 2 | — | |
SMWQOSDRYHJPPA
|
7.9 | IC50 | 2 | — | |
ASCMCEWVQORYKW
|
7.9 | IC50 | 2 | — | |
BKRAEFSPBOVKHB
|
7.9 | IC50 | 2 | — | |
NQGUTBDYFCEIRW
|
7.9 | Ki | 2 | — | |
HGFLURZFAQWPLR
|
7.9 | IC50 | 2 | — | |
ZKLCJRLCFGBSGA
|
7.9 | Ki | 2 | — | |
DSGJGCWDAAFVCG
|
7.9 | IC50 | 2 | — | |
IDENTQOMZWXYGU
|
7.9 | IC50 | 2 | — | |
OVKAPAFXRFWCLH
|
7.9 | IC50 | 2 | — | |
HWFLDTXCWCFGER
|
7.9 | Ki | 2 | — | |
IKEJGJUOBZGDOD
|
7.9 | IC50 | 2 | — | |
JQVLREYTTRETFW
|
7.9 | IC50 | 2 | — | |
KECBJDDHVPUGCU
|
7.9 | IC50 | 2 | — | |
ZYDTWGUZIQERDW
|
7.9 | IC50 | 2 | — | |
CRDBKDAZZPQFSW
|
7.9 | IC50 | 2 | — | |
IXZXPNBZRHAYNV
|
7.9 | IC50 | 2 | — | |
IXZXPNBZRHAYNV
|
7.9 | IC50 | 2 | — | |
KQWKVRKABGLNPZ
|
7.9 | IC50 | 2 | — | |
OMENXXVSZPDLLB
|
7.9 | IC50 | 2 | — | |
STZWKGJXXKBGFV
|
7.9 | Ki | 2 | — | |
IBSZKJJMBBAAER
|
7.9 | Ki | 2 | — | |
JWAYMQSLLVTGIU
|
7.9 | Ki | 2 | — | |
SDDKIJBIOWRQRZ
|
7.9 | IC50 | 2 | — | |
RRMAWHFUAWZMMH
|
7.9 | Ki | 2 | — | |
FSOFQVIEIFGWHM
|
7.8 | IC50 | 2 | — | |
GRJIVWODHSGNKI
|
7.8 | IC50 | 2 | — | |
ANHGWVXCHSOCLJ
|
7.8 | IC50 | 2 | — | |
RGSCMJYPKPAYNA
|
7.8 | IC50 | 2 | — | |
RUGSQKFFXUUTRG
|
7.8 | Ki | 2 | — | |
VKAPCFRLMHHCNC
|
7.8 | IC50 | 2 | — | |
LYPVCWJWDVTCFK
|
7.8 | IC50 | 2 | — | |
HJEHSGSNZZLJBX
|
7.8 | Ki | 2 | — | |
YBLXUAHRYXEFCL
|
7.8 | Ki | 4 | — | |
KFWCOVCZDQWIMX
|
7.8 | IC50 | 2 | — | |
PVQISEQZMSDIEY
|
7.8 | IC50 | 2 | — | |
SJLAOHNQZJMTMQ
|
7.8 | IC50 | 2 | — | |
ZQMGGZLOEIDXMK
|
7.8 | IC50 | 2 | — | |
OMENXXVSZPDLLB
|
7.8 | IC50 | 2 | — | |
AZCXDHIGSFNGSP
|
7.8 | IC50 | 2 | — | |
HPVUNVAPBUWLHX
|
7.8 | IC50 | 2 | — | |
JZJCSOJLMQSMFE
|
7.8 | IC50 | 2 | — | |
FYGORCLOXSCPCK
|
7.8 | Ki | 2 | — | |
JHGAEZRKRKDCKA
|
7.8 | IC50 | 2 | — | |
MIFOAUXADAKDBK
|
7.8 | Ki | 2 | — | |
SGOMEIXLTHTTFC
|
7.8 | IC50 | 2 | — | |
VEMPKZWOJHZWAA
|
7.8 | IC50 | 2 | — | |
YEKRGICETZKVET
|
7.8 | IC50 | 2 | — | |
YMSXZQBIKNRDIU
|
7.8 | IC50 | 2 | — |