Target Details
UniProt ACP06870
Gene SymbolKLK1
Protein NameKallikrein-1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00089 (Trypsin)
Summary
  • Multi-target molecules 630
  • Clinical molecules 0
  • Avg pChEMBL 7.82
Top Co-occurrence Targets
Active Molecules (630)
InChIKey pChEMBL Type Targets Clinical
HTHLQXUFXYHTMY 7.9 IC50 2
NQZSLHCRCYIUAY 7.9 IC50 2
SMWQOSDRYHJPPA 7.9 IC50 2
ASCMCEWVQORYKW 7.9 IC50 2
BKRAEFSPBOVKHB 7.9 IC50 2
NQGUTBDYFCEIRW 7.9 Ki 2
HGFLURZFAQWPLR 7.9 IC50 2
ZKLCJRLCFGBSGA 7.9 Ki 2
DSGJGCWDAAFVCG 7.9 IC50 2
IDENTQOMZWXYGU 7.9 IC50 2
OVKAPAFXRFWCLH 7.9 IC50 2
HWFLDTXCWCFGER 7.9 Ki 2
IKEJGJUOBZGDOD 7.9 IC50 2
JQVLREYTTRETFW 7.9 IC50 2
KECBJDDHVPUGCU 7.9 IC50 2
ZYDTWGUZIQERDW 7.9 IC50 2
CRDBKDAZZPQFSW 7.9 IC50 2
IXZXPNBZRHAYNV 7.9 IC50 2
IXZXPNBZRHAYNV 7.9 IC50 2
KQWKVRKABGLNPZ 7.9 IC50 2
OMENXXVSZPDLLB 7.9 IC50 2
STZWKGJXXKBGFV 7.9 Ki 2
IBSZKJJMBBAAER 7.9 Ki 2
JWAYMQSLLVTGIU 7.9 Ki 2
SDDKIJBIOWRQRZ 7.9 IC50 2
RRMAWHFUAWZMMH 7.9 Ki 2
FSOFQVIEIFGWHM 7.8 IC50 2
GRJIVWODHSGNKI 7.8 IC50 2
ANHGWVXCHSOCLJ 7.8 IC50 2
RGSCMJYPKPAYNA 7.8 IC50 2
RUGSQKFFXUUTRG 7.8 Ki 2
VKAPCFRLMHHCNC 7.8 IC50 2
LYPVCWJWDVTCFK 7.8 IC50 2
HJEHSGSNZZLJBX 7.8 Ki 2
YBLXUAHRYXEFCL 7.8 Ki 4
KFWCOVCZDQWIMX 7.8 IC50 2
PVQISEQZMSDIEY 7.8 IC50 2
SJLAOHNQZJMTMQ 7.8 IC50 2
ZQMGGZLOEIDXMK 7.8 IC50 2
OMENXXVSZPDLLB 7.8 IC50 2
AZCXDHIGSFNGSP 7.8 IC50 2
HPVUNVAPBUWLHX 7.8 IC50 2
JZJCSOJLMQSMFE 7.8 IC50 2
FYGORCLOXSCPCK 7.8 Ki 2
JHGAEZRKRKDCKA 7.8 IC50 2
MIFOAUXADAKDBK 7.8 Ki 2
SGOMEIXLTHTTFC 7.8 IC50 2
VEMPKZWOJHZWAA 7.8 IC50 2
YEKRGICETZKVET 7.8 IC50 2
YMSXZQBIKNRDIU 7.8 IC50 2
2D structure