Target Details
| UniProt AC | P06870 |
|---|---|
| Gene Symbol | KLK1 |
| Protein Name | Kallikrein-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00089 (Trypsin) |
Summary
- Multi-target molecules 630
- Clinical molecules 0
- Avg pChEMBL 7.82
KEGG Pathways (2)
Active Molecules (630)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DUSFQBDHLUPOOL
|
8.1 | IC50 | 2 | — | |
AAECXKAONXCHCZ
|
8.1 | IC50 | 2 | — | |
UXBKOABOOBBNAY
|
8.1 | IC50 | 2 | — | |
UXBKOABOOBBNAY
|
8.1 | IC50 | 2 | — | |
UXBKOABOOBBNAY
|
8.1 | IC50 | 2 | — | |
YTBRECLRKHVGDQ
|
8.1 | IC50 | 2 | — | |
ADOLHLBVAOIJGV
|
8.1 | IC50 | 2 | — | |
BKRAEFSPBOVKHB
|
8.1 | IC50 | 2 | — | |
FCIJZJSYKIPGFH
|
8.1 | IC50 | 2 | — | |
JHGAEZRKRKDCKA
|
8.1 | IC50 | 2 | — | |
QZCMXZHAKDWZOG
|
8.1 | IC50 | 2 | — | |
RPSVGXZDMDZEMA
|
8.1 | IC50 | 2 | — | |
SBELTLOXJSZYPH
|
8.1 | Ki | 2 | — | |
XUWKOBJBCCYWIA
|
8.1 | IC50 | 2 | — | |
ZOWDYXDKZSFHLH
|
8.1 | IC50 | 2 | — | |
ODPYZUJUVLOFCY
|
8.1 | IC50 | 2 | — | |
WBUYZIPRNFWPFT
|
8.1 | IC50 | 2 | — | |
VKAPCFRLMHHCNC
|
8.1 | IC50 | 2 | — | |
JBLNWZHCAUHOQX
|
8.1 | IC50 | 2 | — | |
BRKYUTUGJWHISZ
|
8.1 | IC50 | 2 | — | |
MUESRVUQXGVTLF
|
8.1 | IC50 | 2 | — | |
ZVZPVSAMOLTQDA
|
8.1 | Ki | 2 | — | |
KKGIWARLOKTKIL
|
8.1 | IC50 | 2 | — | |
ONBGAJKCGFMLPR
|
8.1 | IC50 | 2 | — | |
UXBKOABOOBBNAY
|
8.1 | IC50 | 2 | — | |
UZBAMVSBHLGWCL
|
8.1 | IC50 | 2 | — | |
YENCYTMZYKXKQX
|
8.0 | IC50 | 2 | — | |
YENCYTMZYKXKQX
|
8.0 | IC50 | 2 | — | |
BTTXHRACOKUMRC
|
8.0 | IC50 | 2 | — | |
MPOZCROQASDFHG
|
8.0 | IC50 | 2 | — | |
UWAQLEGUXYPPDC
|
8.0 | Ki | 4 | — | |
AJEAFRPCAFBSMW
|
8.0 | IC50 | 2 | — | |
GOBXSXIHPUGHDS
|
8.0 | Ki | 6 | — | |
GZMHLWGWUWMYLQ
|
8.0 | IC50 | 2 | — | |
IXOVGXQOLPAEOH
|
8.0 | IC50 | 2 | — | |
SAHIWIHDGKJMDR
|
8.0 | Ki | 5 | — | |
SRVXDFMBOMTCHO
|
8.0 | IC50 | 2 | — | |
WJNGHXOVBQQPFL
|
8.0 | Ki | 2 | — | |
XFLCKVVRHMCWDE
|
8.0 | IC50 | 2 | — | |
OVKAPAFXRFWCLH
|
8.0 | IC50 | 2 | — | |
QJNZWQVLVDJCSX
|
8.0 | Ki | 2 | — | |
CRDBKDAZZPQFSW
|
8.0 | IC50 | 2 | — | |
MKZAKVVYLTYNQB
|
8.0 | Ki | 2 | — | |
NQGUTBDYFCEIRW
|
8.0 | Ki | 2 | — | |
WOJYOHCXQCTJSI
|
8.0 | Ki | 2 | — | |
ZBFGRVUPGJGBJH
|
8.0 | Ki | 2 | — | |
BKRAEFSPBOVKHB
|
8.0 | IC50 | 2 | — | |
AQJXAFPWULDCCN
|
8.0 | IC50 | 2 | — | |
KAFZMCLLNAVIEP
|
8.0 | IC50 | 2 | — | |
QQQWQABFTREVLI
|
8.0 | Ki | 2 | — |