Target Details
| UniProt AC | P06870 |
|---|---|
| Gene Symbol | KLK1 |
| Protein Name | Kallikrein-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00089 (Trypsin) |
Summary
- Multi-target molecules 630
- Clinical molecules 0
- Avg pChEMBL 7.82
KEGG Pathways (2)
Active Molecules (630)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PVQODELEGLZOBK
|
8.3 | IC50 | 2 | — | |
RVIWTGJMNJDCRK
|
8.3 | IC50 | 2 | — | |
FYWBHLIHHLFVDV
|
8.3 | Ki | 2 | — | |
RLOSSTHVYIUHBJ
|
8.3 | IC50 | 2 | — | |
ZCSIVPYQRVGYCW
|
8.3 | Ki | 2 | — | |
IXOVGXQOLPAEOH
|
8.3 | IC50 | 2 | — | |
QBCVMKWGKASHGW
|
8.3 | Ki | 2 | — | |
FDFMQACLRPEKIS
|
8.3 | Ki | 2 | — | |
AIMMSBQJPYBMLJ
|
8.3 | IC50 | 2 | — | |
IBBWHKCZHBYZMD
|
8.3 | Ki | 2 | — | |
OODWRUWHQPFWHZ
|
8.3 | IC50 | 2 | — | |
QVQFBCDNQLDMQV
|
8.3 | Ki | 2 | — | |
MIGLERBRGFKCDU
|
8.3 | IC50 | 2 | — | |
QUCMMIZCVDZRRO
|
8.3 | IC50 | 2 | — | |
SDXDGYMFFZCAAP
|
8.3 | Ki | 2 | — | |
JBLNWZHCAUHOQX
|
8.2 | IC50 | 2 | — | |
ZGFYAJQKHWKTIW
|
8.2 | IC50 | 2 | — | |
BKRAEFSPBOVKHB
|
8.2 | IC50 | 2 | — | |
GMRLNIZMBUBJGV
|
8.2 | IC50 | 2 | — | |
OZMXFCXWDYBGGS
|
8.2 | Ki | 2 | — | |
OFVMNNNCNPSWSV
|
8.2 | Ki | 2 | — | |
VOGLCERUXSVOOF
|
8.2 | IC50 | 2 | — | |
WIOMWEFIPXIMKV
|
8.2 | Ki | 2 | — | |
CFBNWNBWGWXWAM
|
8.2 | Ki | 2 | — | |
KWTCVHSGOJYHEM
|
8.2 | IC50 | 2 | — | |
PCOLTICMAASINZ
|
8.2 | IC50 | 2 | — | |
XQDFKGVDOCCXNS
|
8.2 | Ki | 3 | — | |
DTBBHSYYSBHKBC
|
8.2 | IC50 | 2 | — | |
NZOLDAJEMNSVON
|
8.2 | IC50 | 2 | — | |
OPOYAWWWOKBVEB
|
8.2 | Ki | 6 | — | |
OPOYAWWWOKBVEB
|
8.2 | Ki | 6 | — | |
RENHVWGXDAZXDL
|
8.2 | IC50 | 2 | — | |
YNDNEALMOBHNKA
|
8.2 | IC50 | 2 | — | |
AINRYWDEGFLBPI
|
8.2 | Ki | 2 | — | |
PVQISEQZMSDIEY
|
8.2 | IC50 | 2 | — | |
CIHHDIMNRRIDCI
|
8.2 | IC50 | 2 | — | |
GCFSKVJROIMITC
|
8.2 | IC50 | 2 | — | |
VKAPCFRLMHHCNC
|
8.2 | IC50 | 2 | — | |
ZOUOCGOVVSXVOD
|
8.2 | IC50 | 2 | — | |
KFEHSYNTGJICFQ
|
8.2 | IC50 | 2 | — | |
URQDUKICBBZPHW
|
8.2 | IC50 | 2 | — | |
KFSFQPNJQRTJEH
|
8.2 | IC50 | 2 | — | |
SXZYKWKZBQBQAC
|
8.2 | IC50 | 2 | — | |
WTOPQLJCODOPEJ
|
8.2 | Ki | 2 | — | |
WYSDYMNFIVNEBU
|
8.2 | Ki | 2 | — | |
HHBAIMAWMHWCTB
|
8.2 | IC50 | 2 | — | |
YUPIEMPZBMGYSW
|
8.2 | IC50 | 2 | — | |
GREDTIZAEYKOPI
|
8.2 | Ki | 2 | — | |
KPWQVEJOWBQVGI
|
8.2 | IC50 | 2 | — | |
RENHVWGXDAZXDL
|
8.2 | IC50 | 2 | — |