Target Details
UniProt ACP06870
Gene SymbolKLK1
Protein NameKallikrein-1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00089 (Trypsin)
Summary
  • Multi-target molecules 630
  • Clinical molecules 0
  • Avg pChEMBL 7.82
Top Co-occurrence Targets
Active Molecules (630)
InChIKey pChEMBL Type Targets Clinical
PVQODELEGLZOBK 8.3 IC50 2
RVIWTGJMNJDCRK 8.3 IC50 2
FYWBHLIHHLFVDV 8.3 Ki 2
RLOSSTHVYIUHBJ 8.3 IC50 2
ZCSIVPYQRVGYCW 8.3 Ki 2
IXOVGXQOLPAEOH 8.3 IC50 2
QBCVMKWGKASHGW 8.3 Ki 2
FDFMQACLRPEKIS 8.3 Ki 2
AIMMSBQJPYBMLJ 8.3 IC50 2
IBBWHKCZHBYZMD 8.3 Ki 2
OODWRUWHQPFWHZ 8.3 IC50 2
QVQFBCDNQLDMQV 8.3 Ki 2
MIGLERBRGFKCDU 8.3 IC50 2
QUCMMIZCVDZRRO 8.3 IC50 2
SDXDGYMFFZCAAP 8.3 Ki 2
JBLNWZHCAUHOQX 8.2 IC50 2
ZGFYAJQKHWKTIW 8.2 IC50 2
BKRAEFSPBOVKHB 8.2 IC50 2
GMRLNIZMBUBJGV 8.2 IC50 2
OZMXFCXWDYBGGS 8.2 Ki 2
OFVMNNNCNPSWSV 8.2 Ki 2
VOGLCERUXSVOOF 8.2 IC50 2
WIOMWEFIPXIMKV 8.2 Ki 2
CFBNWNBWGWXWAM 8.2 Ki 2
KWTCVHSGOJYHEM 8.2 IC50 2
PCOLTICMAASINZ 8.2 IC50 2
XQDFKGVDOCCXNS 8.2 Ki 3
DTBBHSYYSBHKBC 8.2 IC50 2
NZOLDAJEMNSVON 8.2 IC50 2
OPOYAWWWOKBVEB 8.2 Ki 6
OPOYAWWWOKBVEB 8.2 Ki 6
RENHVWGXDAZXDL 8.2 IC50 2
YNDNEALMOBHNKA 8.2 IC50 2
AINRYWDEGFLBPI 8.2 Ki 2
PVQISEQZMSDIEY 8.2 IC50 2
CIHHDIMNRRIDCI 8.2 IC50 2
GCFSKVJROIMITC 8.2 IC50 2
VKAPCFRLMHHCNC 8.2 IC50 2
ZOUOCGOVVSXVOD 8.2 IC50 2
KFEHSYNTGJICFQ 8.2 IC50 2
URQDUKICBBZPHW 8.2 IC50 2
KFSFQPNJQRTJEH 8.2 IC50 2
SXZYKWKZBQBQAC 8.2 IC50 2
WTOPQLJCODOPEJ 8.2 Ki 2
WYSDYMNFIVNEBU 8.2 Ki 2
HHBAIMAWMHWCTB 8.2 IC50 2
YUPIEMPZBMGYSW 8.2 IC50 2
GREDTIZAEYKOPI 8.2 Ki 2
KPWQVEJOWBQVGI 8.2 IC50 2
RENHVWGXDAZXDL 8.2 IC50 2
2D structure