Target Details
| UniProt AC | P06870 |
|---|---|
| Gene Symbol | KLK1 |
| Protein Name | Kallikrein-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00089 (Trypsin) |
Summary
- Multi-target molecules 630
- Clinical molecules 0
- Avg pChEMBL 7.82
KEGG Pathways (2)
Active Molecules (630)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
AKZYZEZPKMKMSU
|
8.5 | Ki | 2 | — | |
REGGTQZTMSDNRQ
|
8.5 | Ki | 2 | — | |
DVMDKOVGIYJULU
|
8.5 | IC50 | 4 | — | |
DXCOONBXASCQJO
|
8.5 | IC50 | 4 | — | |
FAHGWDZMXOZASA
|
8.5 | IC50 | 2 | — | |
FYZGILZDVGOGLF
|
8.5 | IC50 | 2 | — | |
KKTSRKPADJIMFN
|
8.5 | IC50 | 2 | — | |
KPLOPAOSJILVIG
|
8.5 | IC50 | 4 | — | |
LFUVXXPUSUZVRA
|
8.5 | IC50 | 2 | — | |
OGEBHANRXXUPQA
|
8.5 | IC50 | 3 | — | |
OQHYZXMZPSUAEY
|
8.5 | IC50 | 7 | — | |
RVIHDYFOYNJDSF
|
8.5 | IC50 | 2 | — | |
SBFVHGJSVOMQJH
|
8.5 | IC50 | 4 | — | |
UIDZBPBORJEKHP
|
8.5 | IC50 | 2 | — | |
NLYDCXAJZVAQQJ
|
8.5 | Ki | 2 | — | |
OVGDEZZDMAHZLS
|
8.5 | Ki | 2 | — | |
VOYZISZEQQAVDQ
|
8.5 | IC50 | 2 | — | |
XWUNHSSUNZGXRP
|
8.5 | Ki | 2 | — | |
FBTXUKOVWOKZRA
|
8.5 | IC50 | 2 | — | |
PYZHBRHUQRIFKO
|
8.5 | IC50 | 2 | — | |
VOGLCERUXSVOOF
|
8.5 | IC50 | 2 | — | |
FVBDKHAIINLDPZ
|
8.5 | IC50 | 2 | — | |
VJFYVCLOYQXQNA
|
8.5 | Ki | 2 | — | |
WNLGVIFWASWXSX
|
8.5 | IC50 | 2 | — | |
VOGLCERUXSVOOF
|
8.5 | IC50 | 2 | — | |
WAIWQRFSSSDGJI
|
8.5 | Ki | 2 | — | |
YBGKJMRVRJKZGR
|
8.5 | Ki | 2 | — | |
BAQNISDOFDTQKU
|
8.4 | IC50 | 2 | — | |
FYMRCWCAZGYPBP
|
8.4 | IC50 | 2 | — | |
OQEGTLNZIDZKAC
|
8.4 | IC50 | 2 | — | |
VUEARWXFJLMQGY
|
8.4 | IC50 | 2 | — | |
YUPIEMPZBMGYSW
|
8.4 | IC50 | 2 | — | |
CHGFKSDZFXYHGV
|
8.4 | Ki | 2 | — | |
IFUCPBUUGKRAME
|
8.4 | Ki | 2 | — | |
FPDFFZRWYNWVAS
|
8.4 | IC50 | 2 | — | |
ICXJDHNNRWEYID
|
8.4 | IC50 | 2 | — | |
LQNRYTIVDBYPKV
|
8.4 | Ki | 2 | — | |
YMOZEYBQSOZSPV
|
8.4 | IC50 | 2 | — | |
RPSVGXZDMDZEMA
|
8.4 | IC50 | 2 | — | |
CZUOCGQPWJDNLG
|
8.4 | IC50 | 2 | — | |
PMJWRMCIFYNHJS
|
8.4 | IC50 | 2 | — | |
OQRJAZUZBGOFMJ
|
8.4 | IC50 | 2 | — | |
VFZKDTFVYOOMHI
|
8.4 | IC50 | 2 | — | |
XSGPDUZKFYZVSS
|
8.4 | IC50 | 2 | — | |
KKGIWARLOKTKIL
|
8.3 | IC50 | 2 | — | |
KAMFPVZVPCQXKG
|
8.3 | IC50 | 2 | — | |
NOXFGPUWXKVJBR
|
8.3 | IC50 | 2 | — | |
NUXZVLIUOXHZOK
|
8.3 | IC50 | 2 | — | |
CQCYRPKTICMEFH
|
8.3 | IC50 | 2 | — | |
DJVQAYJQHVWWID
|
8.3 | Ki | 2 | — |