Target Details
UniProt ACP06870
Gene SymbolKLK1
Protein NameKallikrein-1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00089 (Trypsin)
Summary
  • Multi-target molecules 630
  • Clinical molecules 0
  • Avg pChEMBL 7.82
Top Co-occurrence Targets
Active Molecules (630)
InChIKey pChEMBL Type Targets Clinical
YNZSWQWEUNSYNO 8.8 IC50 2
XNUZGMGGZBYRHC 8.8 Ki 2
YEGKPXHVNZMVTA 8.8 Ki 2
JVYVKXHJCKLQLH 8.7 IC50 2
POTJJQWDESCPNE 8.7 IC50 2
JSRVCERHRMKWGS 8.7 Ki 2
MJYJOBMDCRLLNJ 8.7 Ki 2
CLIRWBHLYSFJBY 8.7 IC50 2
DDRDPYRGFWAZJN 8.7 Ki 2
DEPURXGJRSOKEM 8.7 IC50 2
MKZAKVVYLTYNQB 8.7 Ki 2
NMXNAXRKFMOCLE 8.7 IC50 2
OPFZSEXPDYGLSZ 8.7 IC50 2
RHYWTBCOSUQEKX 8.7 IC50 2
RLOSSTHVYIUHBJ 8.7 IC50 2
RNXAGUZREAEFHM 8.7 IC50 2
RNXAGUZREAEFHM 8.7 IC50 2
XIDZSQJVHBAEMA 8.7 IC50 2
XXEQNMKFGPOSIN 8.7 IC50 2
ZAAUFWRPGVFJED 8.7 IC50 2
YFXJVNCSNTUTEC 8.7 Ki 2
MYGBAZYZNBWDOA 8.7 IC50 2
SBELTLOXJSZYPH 8.7 Ki 2
ZGFYAJQKHWKTIW 8.7 IC50 2
BOQMRDJDSKQVRQ 8.7 Ki 2
MOXAUHOCUONRLG 8.7 Ki 2
AIJFMBGQAXLEDD 8.7 Ki 2
NXORRDBNCUDYAK 8.7 IC50 2
UJQNOBUUTOYXDR 8.7 Ki 2
MKAAOSLIXYNBND 8.7 Ki 2
JSNGKNZIRNUXEB 8.7 IC50 2
CGGGFYPPUKBYJI 8.6 IC50 2
AEXWSPSOCUVQFS 8.6 IC50 2
CUPBSGSACINCEQ 8.6 Ki 2
KYXDUSCHLYAUKO 8.6 IC50 2
CQCYRPKTICMEFH 8.6 IC50 2
HJEHSGSNZZLJBX 8.6 Ki 2
JDNWFFYXCJRGCY 8.6 IC50 2
OODWRUWHQPFWHZ 8.6 IC50 2
XINDYJQYDORVJG 8.6 IC50 2
YCWWFFYCUWADJG 8.6 IC50 2
DDALAILZEUWVJE 8.6 IC50 2
FDFMQACLRPEKIS 8.6 Ki 2
QYPVPNVUKSFMPZ 8.6 Ki 2
RILHSNVVDGUBBS 8.6 Ki 2
RVIWTGJMNJDCRK 8.6 IC50 2
WRKWQDBVPUMDIA 8.6 Ki 2
PKIXUHOSEWIYFD 8.6 Ki 2
YXRZWOCALHAMDN 8.6 IC50 2
BKOMRHGWSXFZSH 8.5 IC50 3
2D structure