Target Details
UniProt ACP06870
Gene SymbolKLK1
Protein NameKallikrein-1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00089 (Trypsin)
Summary
  • Multi-target molecules 630
  • Clinical molecules 0
  • Avg pChEMBL 7.82
Top Co-occurrence Targets
Active Molecules (630)
InChIKey pChEMBL Type Targets Clinical
LVVUHHFTDFPVTP 9.0 IC50 2
MFOPSUXCHYMMON 9.0 IC50 2
MWDLRAJKBFJGKK 9.0 IC50 2
VQSLCEFIEDDAEK 9.0 IC50 2
VQSLCEFIEDDAEK 9.0 IC50 2
ZAAUFWRPGVFJED 9.0 IC50 2
DWKQZTJLIGQXCW 9.0 Ki 2
MWZDBZAKNXWMIQ 9.0 Ki 2
FHSHZYQPCHWIHY 9.0 Ki 2
JECAJHMCUWSKNH 9.0 IC50 2
LPVUJSLNFIOCKO 9.0 Ki 2
MAXMTSOEDMEECX 9.0 IC50 2
NXORRDBNCUDYAK 9.0 IC50 2
PNLUGDPHROPJFD 9.0 IC50 2
ZAAUFWRPGVFJED 9.0 IC50 2
PGSAHHBOACEADY 8.9 Ki 2
GFVCUIPREFSTJU 8.9 Ki 2
NXORRDBNCUDYAK 8.9 IC50 2
WJCLADGMGRNWKM 8.9 IC50 2
XZCGLEWKUHGGKA 8.9 IC50 2
YUWLGIZXLRBQBZ 8.9 IC50 2
CLIRWBHLYSFJBY 8.9 IC50 2
HNUFVWUQCDKPPA 8.9 IC50 2
IBBWHKCZHBYZMD 8.9 Ki 2
LENLDGUBLYMKDL 8.9 IC50 2
VNAXGGMTQORKLC 8.9 IC50 2
IXBCHGOKNQDTMK 8.9 Ki 2
RTTRNHBUOIYTEB 8.9 Ki 2
WYSPEEWZMDMZCQ 8.9 Ki 2
CLIRWBHLYSFJBY 8.8 IC50 2
CZEFUDHQXHHUQU 8.8 Ki 2
KYZQZFBGHSBBOB 8.8 IC50 2
DJNMZGYTLZEVCG 8.8 Ki 2
CCDMNSGZMYDTKI 8.8 IC50 2
GNEYFEXMAZDVQB 8.8 Ki 2
KYXDUSCHLYAUKO 8.8 IC50 2
NPXRJXHXJUAMFX 8.8 Ki 2
OSHSNAXTHDVEBV 8.8 IC50 2
PMILANWLXZUIMA 8.8 Ki 2
WEQQDCQHAUBLNC 8.8 IC50 2
YZYSWFHAZRVXDH 8.8 IC50 2
NONBHNPXISAARR 8.8 Ki 2
IVCKSIWFRVUXGC 8.8 IC50 2
LWSVGTWSIPMVFX 8.8 Ki 2
OFVMNNNCNPSWSV 8.8 Ki 2
VNMIPKFXVDCVBL 8.8 Ki 2
FYGORCLOXSCPCK 8.8 Ki 2
MVWKKAFRZUSZCR 8.8 Ki 2
ROCAVDUDXDRAQM 8.8 IC50 2
VNAXGGMTQORKLC 8.8 IC50 2
2D structure