Target Details
| UniProt AC | P06870 |
|---|---|
| Gene Symbol | KLK1 |
| Protein Name | Kallikrein-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00089 (Trypsin) |
Summary
- Multi-target molecules 630
- Clinical molecules 0
- Avg pChEMBL 7.82
KEGG Pathways (2)
Active Molecules (630)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
APXAIXPMIFECKD
|
6.2 | Ki | 2 | — | |
DLIVTYIYTMUJNA
|
6.2 | IC50 | 4 | — | |
HQFKZMCNWILBNJ
|
6.2 | IC50 | 3 | — | |
HSNORKMSWCSMOD
|
6.2 | IC50 | 2 | — | |
IOLSRAXZCKDSPO
|
6.2 | Ki | 6 | — | |
MQQNFDZXWVTQEH
|
6.2 | IC50 | 11 | — | |
QEKIKQCZDOHATQ
|
6.2 | IC50 | 2 | — | |
QQRQFIXRVWJLNT
|
6.2 | IC50 | 10 | — | |
RAHPBFRSLVDBER
|
6.2 | Ki | 3 | — | |
RETOSFBTHJWCPW
|
6.2 | IC50 | 3 | — | |
RNYFAJPMYTZRIV
|
6.2 | IC50 | 4 | — | |
VZCLQKXKPFPMJM
|
6.2 | IC50 | 3 | — | |
ZVYUEFHDJYEETD
|
6.2 | Ki | 5 | — | |
HTYIYAXOMLBJLR
|
6.2 | Ki | 2 | — | |
SVWVNWWLYZGNGT
|
6.2 | IC50 | 2 | — | |
WOJYOHCXQCTJSI
|
6.2 | Ki | 2 | — | |
LRUDFXHPVCNXTP
|
6.2 | IC50 | 2 | — | |
LRUDFXHPVCNXTP
|
6.2 | IC50 | 2 | — | |
UKCYVIAOXIAUDI
|
6.2 | IC50 | 2 | — | |
QHYGSRQJBXWIGI
|
6.1 | Ki | 2 | — | |
RYNFLMWBCAHKMX
|
6.1 | Ki | 3 | — | |
IVGMDANEFALECQ
|
6.1 | IC50 | 5 | — | |
OHKHDWZCCRSLRV
|
6.1 | Ki | 2 | — | |
UAZKGEHRMPZZHB
|
6.1 | IC50 | 2 | — | |
UTFYJKDMFNGYLM
|
6.1 | IC50 | 2 | — | |
FHJDRBBZAGYRKH
|
6.0 | Ki | 4 | — | |
GTQYYNKRYLNCBH
|
6.0 | IC50 | 2 | — | |
SBMNLZABUQEIIC
|
6.0 | IC50 | 2 | — | |
CVKDCLNWMMYRKW
|
6.0 | Ki | 2 | — | |
GRQLDCHTDNYVQI
|
6.0 | Ki | 2 | — |