Target Details
UniProt ACP06870
Gene SymbolKLK1
Protein NameKallikrein-1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00089 (Trypsin)
Summary
  • Multi-target molecules 630
  • Clinical molecules 0
  • Avg pChEMBL 7.82
Top Co-occurrence Targets
Active Molecules (630)
InChIKey pChEMBL Type Targets Clinical
XNMJTQFLJFBFHY 6.6 IC50 2
KBNWFXRFMYBDPZ 6.6 IC50 5
CDWKQQJQHYEROC 6.6 IC50 2
CEVDMQKZKKCGLK 6.6 Ki 3
QJVPWUIKUDMGJM 6.6 Ki 6
DKEJQQLJGULWDZ 6.6 Ki 3
YZINAFPRWVMIQH 6.5 IC50 2
XVWWDCXPGPSOQP 6.5 Ki 3
HLWKBMWAJJZWIT 6.5 Ki 5
NKFYMWBVMOGCMS 6.5 IC50 2
MPOZCROQASDFHG 6.5 IC50 2
FRAFAKWXNNKJCF 6.5 IC50 2
HIOJWPJKHKDJAT 6.5 Ki 2
UVCRRKCSIOMXBJ 6.5 IC50 2
VJFYVCLOYQXQNA 6.5 Ki 2
ALVYBVAQSFMTGH 6.5 Ki 3
FCUMAKJXABJJMH 6.5 IC50 2
MRDPVVHRQQSBEC 6.5 IC50 2
MBRTZWCMVQWECS 6.4 IC50 2
XMSAWCPABLSFFM 6.4 Ki 6
FHGOUIMNKLXWAF 6.4 Ki 2
FTZRYRPHXYSWRX 6.4 Ki 2
LECDADCSAFKFQE 6.4 Ki 2
MLQJWDKPHASMIW 6.4 IC50 2
NKPFMFJUENJHQZ 6.4 Ki 2
PDOPCKAPHCDUPT 6.4 Ki 3
YIXUXJDCYJOAHT 6.4 Ki 3
CDJBWPMAVJSWPS 6.4 Ki 6
NWAGTUQRZPXSNY 6.4 IC50 5
UHRIYOJEACOYON 6.4 IC50 3
NRRCXEFBWTVUMX 6.4 IC50 2
OWHBEAUTFNBCPX 6.4 IC50 2
KMJLWAPQPFMUFH 6.4 Ki 2
QEZHMEAWWXNWBV 6.4 IC50 2
RDLNOQFQDDHOTG 6.3 IC50 2
AOPWXUUWEMUVOB 6.3 IC50 2
FAQUHNMIVPDPJH 6.3 IC50 2
CSLOWTUWPRLWOS 6.3 Ki 2
APXAIXPMIFECKD 6.3 Ki 2
UHRIYOJEACOYON 6.3 IC50 3
DIRAHHUANNMTOS 6.3 IC50 2
ASPQAQDFTSKEAM 6.2 IC50 2
FEPIUXBUJVISNN 6.2 Ki 2
LCAJLWIUDOBMSE 6.2 Ki 3
KHVYVAAEFVFJSL 6.2 Ki 3
ZBTNTYAHBLDWER 6.2 IC50 2
QMIPDUHHMKIFHM 6.2 IC50 2
QMRJOIUGPCVZPH 6.2 Ki 6
FKUAJSCZSYQJSF 6.2 IC50 4
LUNUFGFUBAQPEV 6.2 IC50 4
2D structure