Target Details
UniProt ACP06870
Gene SymbolKLK1
Protein NameKallikrein-1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00089 (Trypsin)
Summary
  • Multi-target molecules 630
  • Clinical molecules 0
  • Avg pChEMBL 7.82
Top Co-occurrence Targets
Active Molecules (630)
InChIKey pChEMBL Type Targets Clinical
DKCUPHYMPFYPAB 7.0 Ki 2
ZWIGNYNESQGQBP 7.0 IC50 2
DINGGRQCVMHNRL 7.0 IC50 2
JAXUEOKMIODUOS 7.0 Ki 3
OBBJEUZSEBLKBM 6.9 IC50 2
PKIXUHOSEWIYFD 6.9 Ki 2
JNTUFKHYHGYBBL 6.9 Ki 2
MUPHEXMZSXMJJT 6.9 Ki 6
QGRNPIFRFQQVJW 6.9 Ki 2
VSDPAHALQLIVTA 6.9 IC50 2
YYQCFGQMWCQRTL 6.9 IC50 2
FZNUIBFUDXMFEC 6.9 IC50 2
SVUKIPZHHBQFDL 6.9 Ki 2
BOIJPGRTYUYSOS 6.9 IC50 2
MSRCXFCFCMLGJJ 6.9 IC50 2
NKDPZFVLWOOSBI 6.9 IC50 2
PRAHDYKFUBAHGY 6.9 Ki 2
VAVMIWZZMKRLJD 6.9 IC50 2
DCIOQBFAYLXHBY 6.8 Ki 3
SFGVINOBUNVDBX 6.8 IC50 2
XCYDAVGXMZTCMZ 6.8 IC50 2
MJNFCOZBOUBSHI 6.8 Ki 2
JZXAFDAZYPJHEB 6.8 IC50 2
JZXAFDAZYPJHEB 6.8 IC50 2
FWEWLZSBDNPNAD 6.8 Ki 3
ZCCVEIWTZACMLJ 6.8 IC50 2
CKNDVDLSIUTQOV 6.8 IC50 2
QPBFLOWZPFHTHE 6.8 Ki 6
MRDPVVHRQQSBEC 6.8 IC50 2
UHKUZNDEDMCQLX 6.8 Ki 2
YKHFOMDUJQEALA 6.8 Ki 2
YXHAGUGRTPADHH 6.8 IC50 2
PTCNGRBWQCYOSG 6.7 IC50 2
PRKWITZMBNVLDR 6.7 IC50 2
DAZKRYLEGWSBDU 6.7 Ki 2
RRNRMCAVLZYWDN 6.7 Ki 3
OOFRCFJPOZMMHV 6.7 Ki 3
ZQFKUIZTYMVJHJ 6.7 Ki 2
AJEAFRPCAFBSMW 6.7 IC50 2
WDDXVXICYPNBRY 6.7 IC50 2
SFXBQEQLNCWVDH 6.7 Ki 2
YZINAFPRWVMIQH 6.7 IC50 2
ZASUNCQYGAHWBN 6.6 IC50 3
LGHSOUBTKFLVOU 6.6 IC50 2
MPEZSZKUEPIWCM 6.6 IC50 2
BOVRMDWYQFHWSN 6.6 Ki 2
RMJHMNZGTJDKCS 6.6 IC50 4
ASMYEURNFQLBPE 6.6 IC50 2
DUVLBBOBLCROSD 6.6 IC50 3
NWAGTUQRZPXSNY 6.6 IC50 6
2D structure