Target Details
UniProt ACP06870
Gene SymbolKLK1
Protein NameKallikrein-1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00089 (Trypsin)
Summary
  • Multi-target molecules 630
  • Clinical molecules 0
  • Avg pChEMBL 7.82
Top Co-occurrence Targets
Active Molecules (630)
InChIKey pChEMBL Type Targets Clinical
KAUYBZJFBAONCO 11.3 Ki 6
ZBFGRVUPGJGBJH 9.8 Ki 2
OZHSSBBIGXHETL 9.7 Ki 2
RYSVSPUJOFJUCF 9.6 Ki 2
YWANJCPORQUSJY 9.6 Ki 2
QPOLNDRLBGEWMU 9.5 Ki 2
LPVUJSLNFIOCKO 9.5 Ki 2
NQHRMYDBUNKTFA 9.5 Ki 2
SBVGFLWILRJNQM 9.5 Ki 2
FZFPYNKLVBCZMF 9.4 Ki 2
GABXXTIRMXPUTH 9.4 IC50 2
OFVMNNNCNPSWSV 9.4 Ki 2
OIZRTRZVPKYRKU 9.4 IC50 2
DABQZHUZIQWQLQ 9.4 Ki 2
TUSKELNUILZYRS 9.4 Ki 2
OMMREAWBRLWOAO 9.3 Ki 2
KWJCEENMJCVGKA 9.3 Ki 2
PMILANWLXZUIMA 9.3 Ki 2
GNEYFEXMAZDVQB 9.3 Ki 2
HKBZVXMQYIGMEV 9.2 IC50 2
WOJYOHCXQCTJSI 9.2 Ki 2
GBNNJVPDIBQYPY 9.2 IC50 2
JECAJHMCUWSKNH 9.2 IC50 2
QAMDYRLZBXKYIV 9.2 Ki 2
XXEQNMKFGPOSIN 9.2 IC50 2
FLUCBLLJFWRIKM 9.2 Ki 2
XHKKWYQSDAQWHO 9.2 Ki 2
GABXXTIRMXPUTH 9.2 IC50 2
JECAJHMCUWSKNH 9.2 IC50 2
OIZRTRZVPKYRKU 9.2 IC50 2
OSHSNAXTHDVEBV 9.2 IC50 2
SJSZCUOGQWOGFI 9.2 Ki 2
VCQTWIVEFHEKDZ 9.2 IC50 2
XZCGLEWKUHGGKA 9.2 IC50 2
YBGKJMRVRJKZGR 9.2 Ki 2
WWWJBEWOQREFGE 9.1 Ki 2
OLHHQMRNSGUPLQ 9.1 Ki 2
CFAFTAKKKKAEGI 9.1 IC50 2
NXDBZRSRGJYZAK 9.1 Ki 2
RYSVSPUJOFJUCF 9.1 Ki 2
TUZQUJRYIVEFEH 9.1 Ki 2
LVVUHHFTDFPVTP 9.1 IC50 2
XZCGLEWKUHGGKA 9.1 IC50 2
KAKBBSOLSJWTRB 9.1 Ki 2
PYAIUIRWRUKFGI 9.1 Ki 2
OIZRTRZVPKYRKU 9.1 IC50 2
OSHSNAXTHDVEBV 9.1 IC50 2
DYLHBKKFYOXVTC 9.0 Ki 2
IPMBKJBCZMJJID 9.0 IC50 2
KHKMNGWOVOQDJO 9.0 IC50 2
2D structure