Target Details
| UniProt AC | P06756 |
|---|---|
| Gene Symbol | ITGAV |
| Protein Name | Integrin alpha-V |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01839 (FG-GAP) PF08441 (Integrin_A_Ig_1) PF20805 (Integrin_A_Ig_2) PF20806 (Integrin_A_Ig_3) PF00357 (Integrin_alpha) |
Summary
- Multi-target molecules 1,632
- Clinical molecules 0
- Avg pChEMBL 7.69
KEGG Pathways (20)
- Arrhythmogenic right ventricular cardiomyopathy
- Cell adhesion molecule (CAM) interaction
- Cytoskeleton in muscle cells
- Dilated cardiomyopathy
- ECM-receptor interaction
- Efferocytosis
- Fluid shear stress and atherosclerosis
- Focal adhesion
- Hormone signaling
- Human cytomegalovirus infection
- Human papillomavirus infection
- Hypertrophic cardiomyopathy
- Integrin signaling
- PI3K-Akt signaling pathway
- Pathways in cancer
- Phagosome
- Proteoglycans in cancer
- Regulation of actin cytoskeleton
- Small cell lung cancer
- Thyroid hormone signaling pathway
Associated Diseases (1)
Active Molecules (1,632)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ITGKMDQIQJNXCY
|
8.5 | IC50 | 3 | — | |
PVDGZHKJXXVONO
|
8.5 | IC50 | 2 | — | |
YVWHUWDPZJFVCO
|
8.5 | IC50 | 2 | — | |
YVWHUWDPZJFVCO
|
8.5 | IC50 | 2 | — | |
CUQFEHKORVQEQE
|
8.5 | IC50 | 2 | — | |
DTINBQRHDAOJQT
|
8.5 | Ki | 2 | — | |
HTPRMRASPJUHGG
|
8.5 | IC50 | 3 | — | |
QCZXVUVLNOHNFI
|
8.5 | IC50 | 3 | — | |
WWPKVHRHQNABNG
|
8.5 | IC50 | 3 | — | |
YITSCMGHJOGUNC
|
8.5 | Ki | 3 | — | |
LBBYDFXRXWGQLT
|
8.4 | IC50 | 2 | — | |
DTNKZZXZAPCYPT
|
8.4 | IC50 | 3 | — | |
HHUNTZLKFUBXAE
|
8.4 | IC50 | 3 | — | |
QYRCHDXNDRSUDT
|
8.4 | IC50 | 3 | — | |
SJZFNMIWSQZTHK
|
8.4 | IC50 | 2 | — | |
VJKNTBIICLHWFT
|
8.4 | IC50 | 2 | — | |
VTLYACZOFKLVKB
|
8.4 | IC50 | 2 | — | |
MRXQBHPWVQTUKZ
|
8.4 | IC50 | 3 | — | |
ORWWOJYZCUHJQK
|
8.4 | IC50 | 3 | — | |
TUBIMZBESOVRAC
|
8.4 | IC50 | 2 | — | |
VVILZPGXJJNTRY
|
8.4 | IC50 | 2 | — | |
HVRQQWLXXYKJKU
|
8.4 | IC50 | 3 | — | |
IHJDDZUSFQGHNY
|
8.4 | IC50 | 2 | — | |
ANGDPTFGRFDVLH
|
8.4 | IC50 | 3 | — | |
CJFKBQRLRONQOT
|
8.4 | IC50 | 7 | — | |
FHNGIQUASOHITF
|
8.4 | IC50 | 2 | — | |
WPFBXGBKFBKHDX
|
8.4 | IC50 | 3 | — | |
ZPRQEMGTRXGZPE
|
8.4 | IC50 | 5 | — | |
CNEKZXJTDXCVRA
|
8.4 | Ki | 2 | — | |
DOPHFAZXVAQXOW
|
8.4 | Ki | 2 | — | |
FCTUEQVODTYVHM
|
8.4 | IC50 | 3 | — | |
FSXPSVVMLALNDM
|
8.4 | IC50 | 3 | — | |
HODBWQCCKYDYPY
|
8.4 | IC50 | 3 | — | |
IUFCIFVCEOUHLU
|
8.4 | IC50 | 2 | — | |
JNSBZXVASWNXFL
|
8.4 | Ki | 2 | — | |
KTPKPDHZXPMGRV
|
8.4 | IC50 | 5 | — | |
KUGOKSJJMZIXRT
|
8.4 | IC50 | 2 | — | |
KZYLTZUXEHTOHA
|
8.4 | IC50 | 3 | — | |
LDHLQPMIUKAPSY
|
8.4 | IC50 | 5 | — | |
PQWRZQIWMNBRRU
|
8.4 | IC50 | 3 | — | |
QZTBJCSOVXRYCX
|
8.4 | IC50 | 6 | — | |
RLEVQGAGXMBFLZ
|
8.4 | IC50 | 2 | — | |
SLTMEZLQPRTTBL
|
8.4 | IC50 | 3 | — | |
SXTLBFQXNNGAPB
|
8.4 | Ki | 2 | — | |
XNPQTWYQUUYENN
|
8.4 | Ki | 2 | — | |
AVVMNAYVLDAZHD
|
8.4 | IC50 | 2 | — | |
BGLLQJHWAUGNSA
|
8.4 | IC50 | 3 | — | |
QPBKEMRNMDTBPC
|
8.4 | IC50 | 2 | — | |
HVDDJMWVUNHMDN
|
8.4 | IC50 | 2 | — | |
RBSUHEPCSZKVSP
|
8.4 | IC50 | 4 | — |