Target Details
| UniProt AC | P06756 |
|---|---|
| Gene Symbol | ITGAV |
| Protein Name | Integrin alpha-V |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01839 (FG-GAP) PF08441 (Integrin_A_Ig_1) PF20805 (Integrin_A_Ig_2) PF20806 (Integrin_A_Ig_3) PF00357 (Integrin_alpha) |
Summary
- Multi-target molecules 1,632
- Clinical molecules 0
- Avg pChEMBL 7.69
KEGG Pathways (20)
- Arrhythmogenic right ventricular cardiomyopathy
- Cell adhesion molecule (CAM) interaction
- Cytoskeleton in muscle cells
- Dilated cardiomyopathy
- ECM-receptor interaction
- Efferocytosis
- Fluid shear stress and atherosclerosis
- Focal adhesion
- Hormone signaling
- Human cytomegalovirus infection
- Human papillomavirus infection
- Hypertrophic cardiomyopathy
- Integrin signaling
- PI3K-Akt signaling pathway
- Pathways in cancer
- Phagosome
- Proteoglycans in cancer
- Regulation of actin cytoskeleton
- Small cell lung cancer
- Thyroid hormone signaling pathway
Associated Diseases (1)
Active Molecules (1,632)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MYSBVCKSODARFZ
|
8.7 | IC50 | 3 | — | |
YSHCUQUSNSOANU
|
8.7 | IC50 | 3 | — | |
CICPWOGAFQCAEW
|
8.6 | IC50 | 2 | — | |
DBFQYQDMGSZHES
|
8.6 | IC50 | 2 | — | |
DTCHSFYIOSVBQO
|
8.6 | IC50 | 5 | — | |
UQSXTDKNKMCKEM
|
8.6 | IC50 | 3 | — | |
YUFKABYHWCRYRX
|
8.6 | IC50 | 2 | — | |
HIKCELHIZSKMGI
|
8.6 | IC50 | 5 | — | |
DAFKTUSUEPQPBU
|
8.6 | IC50 | 3 | — | |
JYENEFWTARBUPP
|
8.6 | IC50 | 2 | — | |
RWBOWRDCKZVMOU
|
8.6 | Ki | 2 | — | |
XXBNSEBYSGKBAQ
|
8.6 | IC50 | 4 | — | |
ZNFLNPHHAFFHFM
|
8.6 | IC50 | 2 | — | |
FLTIMXZSLYRKOV
|
8.6 | IC50 | 3 | — | |
BLLLAUHTNAVSQR
|
8.6 | IC50 | 5 | — | |
DTLIDYQJLOBQPK
|
8.6 | Ki | 3 | — | |
JFGWITIVJGEHEK
|
8.6 | Ki | 2 | — | |
JRVUMBDCNCWNEP
|
8.6 | IC50 | 3 | — | |
KUZMKJHBJRIPSL
|
8.6 | Ki | 4 | — | |
STLNBQRXIPETRC
|
8.6 | Ki | 2 | — | |
YYQUWEHEBOMRPH
|
8.6 | IC50 | 2 | — | |
BSTGKAROMCRBDW
|
8.6 | IC50 | 2 | — | |
VUDQMHAFTAQNOM
|
8.6 | IC50 | 4 | — | |
FRCHUTQNZCVLPJ
|
8.6 | IC50 | 2 | — | |
NQIOUHXNYUMMLV
|
8.6 | IC50 | 4 | — | |
NIAUTJLMLQTPHC
|
8.6 | IC50 | 3 | — | |
AQAUYHNXROATLO
|
8.6 | IC50 | 3 | — | |
JYJNRUFKUMSRIN
|
8.6 | IC50 | 6 | — | |
UVNKAYDKTALKMK
|
8.6 | IC50 | 3 | — | |
ZNERAUDQUULBOO
|
8.6 | IC50 | 3 | — | |
ACEBGKIPKRNNIW
|
8.5 | IC50 | 2 | — | |
GPYWNBXZBJVOHR
|
8.5 | Ki | 2 | — | |
IKALVLPAIVXDBO
|
8.5 | IC50 | 3 | — | |
JFZKVQANYRYBMC
|
8.5 | Ki | 2 | — | |
LAROZEWEPNAWMD
|
8.5 | IC50 | 2 | — | |
ZNBWKHIYCLLIHV
|
8.5 | IC50 | 2 | — | |
DMJMBJHEDODVMW
|
8.5 | IC50 | 3 | — | |
FHDYMEIDWKIBAW
|
8.5 | IC50 | 2 | — | |
HGFOOLONGOBCMP
|
8.5 | IC50 | 6 | — | |
KWKNIANILQEFIG
|
8.5 | IC50 | 2 | — | |
RWYVJJKDFYFYFO
|
8.5 | Ki | 2 | — | |
SQQTTWBLXRVPQZ
|
8.5 | IC50 | 2 | — | |
VPPZGLXMAAPXBC
|
8.5 | Ki | 2 | — | |
WNVOEBNTIMVWEQ
|
8.5 | IC50 | 2 | — | |
XMXSNMYAHVBHCD
|
8.5 | IC50 | 2 | — | |
XSXPFCDFDWOKST
|
8.5 | IC50 | 2 | — | |
XUISHROIRBHOIM
|
8.5 | IC50 | 4 | — | |
SGUTWRZFDXCOLS
|
8.5 | IC50 | 2 | — | |
NYIZCWIYRUTEKV
|
8.5 | IC50 | 5 | — | |
ZYPBXFINEXHXPV
|
8.5 | IC50 | 4 | — |