Target Details
| UniProt AC | P06756 |
|---|---|
| Gene Symbol | ITGAV |
| Protein Name | Integrin alpha-V |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01839 (FG-GAP) PF08441 (Integrin_A_Ig_1) PF20805 (Integrin_A_Ig_2) PF20806 (Integrin_A_Ig_3) PF00357 (Integrin_alpha) |
Summary
- Multi-target molecules 1,632
- Clinical molecules 0
- Avg pChEMBL 7.69
KEGG Pathways (20)
- Arrhythmogenic right ventricular cardiomyopathy
- Cell adhesion molecule (CAM) interaction
- Cytoskeleton in muscle cells
- Dilated cardiomyopathy
- ECM-receptor interaction
- Efferocytosis
- Fluid shear stress and atherosclerosis
- Focal adhesion
- Hormone signaling
- Human cytomegalovirus infection
- Human papillomavirus infection
- Hypertrophic cardiomyopathy
- Integrin signaling
- PI3K-Akt signaling pathway
- Pathways in cancer
- Phagosome
- Proteoglycans in cancer
- Regulation of actin cytoskeleton
- Small cell lung cancer
- Thyroid hormone signaling pathway
Associated Diseases (1)
Active Molecules (1,632)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YJVQTPGCEVENKR
|
8.8 | IC50 | 4 | — | |
IALCADUNFMACEG
|
8.8 | IC50 | 3 | — | |
LPWSHOGTPIIOBC
|
8.8 | IC50 | 5 | — | |
NENWIXCUUFUHIH
|
8.8 | IC50 | 3 | — | |
OCFMIMLTAYUZOV
|
8.8 | IC50 | 2 | — | |
RRYMQSFBOJUJEI
|
8.8 | IC50 | 2 | — | |
YRIJMZJTWNXHBY
|
8.8 | IC50 | 2 | — | |
IFUROQAKNZUNFY
|
8.8 | IC50 | 5 | — | |
MXSJSHDIEDILST
|
8.8 | IC50 | 4 | — | |
OLQOZUUGUUUOMF
|
8.8 | IC50 | 3 | — | |
LAKQAEHCCWPUIS
|
8.7 | IC50 | 3 | — | |
LMFGOELGOHYQNF
|
8.7 | IC50 | 2 | — | |
ZMVBGJMBSDZOLI
|
8.7 | IC50 | 2 | — | |
CTOPQASYIWIPDN
|
8.7 | IC50 | 3 | — | |
KRAZOLZZRSRPAE
|
8.7 | IC50 | 4 | — | |
BDICDHJCLYIIQR
|
8.7 | IC50 | 2 | — | |
HOXCYDQJLHZQJW
|
8.7 | IC50 | 2 | — | |
MDGSJXNNVZDXCV
|
8.7 | IC50 | 2 | — | |
NGWFKQKKCNUAJQ
|
8.7 | IC50 | 3 | — | |
UQEWVVUNGPKKKR
|
8.7 | IC50 | 6 | — | |
XGBKKOOTEJXBQX
|
8.7 | IC50 | 2 | — | |
AMBKCWJWRSLIIL
|
8.7 | IC50 | 3 | — | |
BNTMUQHWJSORQO
|
8.7 | IC50 | 3 | — | |
BZRUQNTYVLMGAR
|
8.7 | IC50 | 3 | — | |
CKPFLCVDCRYWAY
|
8.7 | IC50 | 3 | — | |
DTLIDYQJLOBQPK
|
8.7 | IC50 | 2 | — | |
GITHMVUAHBUYNI
|
8.7 | IC50 | 2 | — | |
JCZHWFZLHYLGEG
|
8.7 | Ki | 2 | — | |
MHOGEKRNTRTBND
|
8.7 | IC50 | 3 | — | |
NUQYRSCTGCUBSM
|
8.7 | IC50 | 2 | — | |
PVNQAXDNDZYXIW
|
8.7 | Ki | 2 | — | |
UAYIUFJSMAVZPH
|
8.7 | Ki | 2 | — | |
UHXBOYLWYUPYDA
|
8.7 | IC50 | 3 | — | |
VKOQXUDGMWQFAJ
|
8.7 | IC50 | 2 | — | |
XFHCUQCLLGVBIK
|
8.7 | IC50 | 3 | — | |
XSDMZRDIJUIWTH
|
8.7 | Ki | 2 | — | |
YLEXAKYOIPPMHL
|
8.7 | IC50 | 3 | — | |
ASSOJPJBNSNTEH
|
8.7 | IC50 | 2 | — | |
JMPYJQPICLIXCK
|
8.7 | IC50 | 3 | — | |
LCNAIFMSOWTUTF
|
8.7 | IC50 | 2 | — | |
UEIWSFUOMHYAMK
|
8.7 | IC50 | 4 | — | |
GJZSXEXGYRGEQC
|
8.7 | IC50 | 3 | — | |
HOXLTGNIFJUOIA
|
8.7 | IC50 | 6 | — | |
KAVRMLREXXGTPY
|
8.7 | IC50 | 3 | — | |
UVRKETLYFWGQPV
|
8.7 | IC50 | 2 | — | |
VRLVARCYYMQMEO
|
8.7 | IC50 | 3 | — | |
WEXQBLSMARBRMG
|
8.7 | IC50 | 6 | — | |
XHPZRPHYLGZLTO
|
8.7 | IC50 | 5 | — | |
IYUQNBTYGGJEAT
|
8.7 | IC50 | 3 | — | |
IZJKOCVIGXNCTL
|
8.7 | IC50 | 3 | — |