Target Details
| UniProt AC | P06756 |
|---|---|
| Gene Symbol | ITGAV |
| Protein Name | Integrin alpha-V |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01839 (FG-GAP) PF08441 (Integrin_A_Ig_1) PF20805 (Integrin_A_Ig_2) PF20806 (Integrin_A_Ig_3) PF00357 (Integrin_alpha) |
Summary
- Multi-target molecules 1,632
- Clinical molecules 0
- Avg pChEMBL 7.69
KEGG Pathways (20)
- Arrhythmogenic right ventricular cardiomyopathy
- Cell adhesion molecule (CAM) interaction
- Cytoskeleton in muscle cells
- Dilated cardiomyopathy
- ECM-receptor interaction
- Efferocytosis
- Fluid shear stress and atherosclerosis
- Focal adhesion
- Hormone signaling
- Human cytomegalovirus infection
- Human papillomavirus infection
- Hypertrophic cardiomyopathy
- Integrin signaling
- PI3K-Akt signaling pathway
- Pathways in cancer
- Phagosome
- Proteoglycans in cancer
- Regulation of actin cytoskeleton
- Small cell lung cancer
- Thyroid hormone signaling pathway
Associated Diseases (1)
Active Molecules (1,632)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MSGZVCWOFQOMDA
|
8.9 | IC50 | 2 | — | |
ZSYFEFOBOJYQCG
|
8.9 | IC50 | 2 | — | |
LWCKRBHIZLBAFM
|
8.9 | IC50 | 2 | — | |
MYSBVCKSODARFZ
|
8.9 | IC50 | 3 | — | |
OQDKBZBKHWYBSI
|
8.9 | IC50 | 3 | — | |
BHDLQEOXHBGVFT
|
8.9 | IC50 | 2 | — | |
FQTMTTZENZSMQU
|
8.9 | IC50 | 2 | — | |
JTQSBYUBJLIDAK
|
8.9 | IC50 | 5 | — | |
MHGHYXQIIPLSCN
|
8.9 | Ki | 2 | — | |
XFNZYXKVDFJAFI
|
8.9 | IC50 | 6 | — | |
ZEEBGVAVQWCFLT
|
8.9 | IC50 | 3 | — | |
BZPNVJGCQPADST
|
8.9 | IC50 | 3 | — | |
ZQAQMOMRTYIDJU
|
8.9 | IC50 | 4 | — | |
FPSTULSQRYACMJ
|
8.9 | IC50 | 3 | — | |
LTTIHWWYCLBIKC
|
8.9 | IC50 | 3 | — | |
RTHTZKFWJRGDKZ
|
8.9 | IC50 | 4 | — | |
AEFPUSNNPXBSKD
|
8.8 | IC50 | 3 | — | |
CDIQJJMJTFHODD
|
8.8 | IC50 | 2 | — | |
CXHCNOMGODVIKB
|
8.8 | IC50 | 7 | — | |
DKCBOEVMYBPSHB
|
8.8 | Ki | 2 | — | |
IJIQSYZFWKZVHL
|
8.8 | Ki | 2 | — | |
PLPDPJUYPOKPOK
|
8.8 | IC50 | 2 | — | |
QKCFDPUKGKJIML
|
8.8 | IC50 | 7 | — | |
RGPCXWUHNLAAMX
|
8.8 | IC50 | 2 | — | |
SBROZGGPOIEKJM
|
8.8 | IC50 | 2 | — | |
YWCFKVFIEXQDJL
|
8.8 | IC50 | 3 | — | |
DRAZWXSJTKLZTP
|
8.8 | IC50 | 2 | — | |
WOXAQXBQXVXPHE
|
8.8 | IC50 | 2 | — | |
CJDLVBMPCKYVJE
|
8.8 | IC50 | 2 | — | |
FZBGGWKHCWPGOF
|
8.8 | IC50 | 2 | — | |
GARROJJZLJSGSW
|
8.8 | IC50 | 4 | — | |
HRJYJLGVTFNBBO
|
8.8 | IC50 | 2 | — | |
IXYJRFZTWSBREE
|
8.8 | IC50 | 2 | — | |
JARATYKMRJHXBN
|
8.8 | IC50 | 2 | — | |
UJAJKKVATBUTAU
|
8.8 | IC50 | 2 | — | |
VMCREQBBFYDYNW
|
8.8 | Ki | 2 | — | |
YDHAGPCZRFQPOI
|
8.8 | IC50 | 6 | — | |
DGHLGBHZIKLZQQ
|
8.8 | IC50 | 2 | — | |
FNKFUBZIIVXPMV
|
8.8 | IC50 | 2 | — | |
HXARURWAKJJNNF
|
8.8 | IC50 | 3 | — | |
UBSZHEXPLSECRR
|
8.8 | IC50 | 3 | — | |
CTHYLBXDQVAGEJ
|
8.8 | IC50 | 5 | — | |
DIMDWQUSJSWNOO
|
8.8 | IC50 | 5 | — | |
DSVRSYVZAMHQET
|
8.8 | IC50 | 2 | — | |
GNIPEZAXNSJOFR
|
8.8 | IC50 | 3 | — | |
JTUKSGXZGMYCDU
|
8.8 | IC50 | 2 | — | |
KXYAXQVLPNBUFO
|
8.8 | IC50 | 5 | — | |
LJKWPNDKPDWWIA
|
8.8 | IC50 | 4 | — | |
QYKHSZCOMAXNCJ
|
8.8 | IC50 | 6 | — | |
UMSKKXXFLOGWFX
|
8.8 | IC50 | 4 | — |