Target Details
| UniProt AC | P06756 |
|---|---|
| Gene Symbol | ITGAV |
| Protein Name | Integrin alpha-V |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01839 (FG-GAP) PF08441 (Integrin_A_Ig_1) PF20805 (Integrin_A_Ig_2) PF20806 (Integrin_A_Ig_3) PF00357 (Integrin_alpha) |
Summary
- Multi-target molecules 1,632
- Clinical molecules 0
- Avg pChEMBL 7.69
KEGG Pathways (20)
- Arrhythmogenic right ventricular cardiomyopathy
- Cell adhesion molecule (CAM) interaction
- Cytoskeleton in muscle cells
- Dilated cardiomyopathy
- ECM-receptor interaction
- Efferocytosis
- Fluid shear stress and atherosclerosis
- Focal adhesion
- Hormone signaling
- Human cytomegalovirus infection
- Human papillomavirus infection
- Hypertrophic cardiomyopathy
- Integrin signaling
- PI3K-Akt signaling pathway
- Pathways in cancer
- Phagosome
- Proteoglycans in cancer
- Regulation of actin cytoskeleton
- Small cell lung cancer
- Thyroid hormone signaling pathway
Associated Diseases (1)
Active Molecules (1,632)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WVOZQEYNBBHACY
|
9.1 | IC50 | 2 | — | |
XCTHUNKHDUMJGV
|
9.1 | IC50 | 2 | — | |
QYKHSZCOMAXNCJ
|
9.0 | IC50 | 5 | — | |
RZYRWEAZPQSSKX
|
9.0 | IC50 | 5 | — | |
YTAHOLPCQRGOAW
|
9.0 | IC50 | 5 | — | |
NRXYMNJDCGQEHP
|
9.0 | IC50 | 2 | — | |
VJTDBRLHPYYFBZ
|
9.0 | IC50 | 2 | — | |
ANCHZQJTSKHDFM
|
9.0 | IC50 | 2 | — | |
BEOOWKDNVJKISL
|
9.0 | IC50 | 3 | — | |
CNNXQMKKHGGQNP
|
9.0 | Ki | 2 | — | |
CYIAZAFUQCTLTE
|
9.0 | IC50 | 2 | — | |
DKSFLHZSAWZIDR
|
9.0 | IC50 | 2 | — | |
FCUCMIIVLCLREX
|
9.0 | IC50 | 3 | — | |
IFDIAYNOLNAOOF
|
9.0 | Ki | 2 | — | |
LXYBJVGMCKOMFL
|
9.0 | IC50 | 2 | — | |
MXVQXMBMRJIIHT
|
9.0 | IC50 | 2 | — | |
PEFBVOAICYLSAF
|
9.0 | IC50 | 8 | — | |
PSWDFAPCKFYFPG
|
9.0 | IC50 | 2 | — | |
QEWKBLVMROGVIO
|
9.0 | IC50 | 6 | — | |
QLBXWVBTUGYSGI
|
9.0 | IC50 | 8 | — | |
UOBZVUNLYKJTSH
|
9.0 | IC50 | 2 | — | |
XJRPJRUXGLBKPY
|
9.0 | IC50 | 2 | — | |
YEEBBNWKQGDACU
|
9.0 | IC50 | 3 | — | |
YTROSQIPEKDADK
|
9.0 | IC50 | 2 | — | |
NIGWPUUZRHIDKJ
|
9.0 | IC50 | 3 | — | |
DHLKXUDAGRMGLV
|
9.0 | IC50 | 2 | — | |
GFGRBKXJVOAPLF
|
9.0 | IC50 | 3 | — | |
KIOVJZCZUNJXQB
|
9.0 | IC50 | 3 | — | |
OUOJYIATFPJDBV
|
9.0 | IC50 | 2 | — | |
PDZBKVNASRLHEK
|
9.0 | IC50 | 2 | — | |
VYVQCVGITLHGKO
|
9.0 | IC50 | 2 | — | |
YGOKSIVHHLSPET
|
9.0 | IC50 | 4 | — | |
YURBLSCQXZUCIK
|
9.0 | IC50 | 2 | — | |
ZAMKDPACDNUZPJ
|
9.0 | IC50 | 8 | — | |
KZYWKHUJTXLNJM
|
8.9 | IC50 | 5 | — | |
SFCYQXKSWPPSIX
|
8.9 | IC50 | 4 | — | |
BCZJAKMDVNIASQ
|
8.9 | IC50 | 3 | — | |
JANXNGXRGZTCLF
|
8.9 | IC50 | 3 | — | |
PZAMXSCMHJPGFV
|
8.9 | IC50 | 3 | — | |
YVGFDNFQFUSINK
|
8.9 | IC50 | 3 | — | |
AZPMNBDRAVVHOL
|
8.9 | IC50 | 3 | — | |
IETWETOHQHTRGK
|
8.9 | IC50 | 2 | — | |
MIFZAPHWMCAHQZ
|
8.9 | IC50 | 5 | — | |
QXAYHAXWXRCLTG
|
8.9 | IC50 | 4 | — | |
RYILTXKXDOUWET
|
8.9 | IC50 | 2 | — | |
UQYFVSMGEHOGBU
|
8.9 | IC50 | 5 | — | |
VOZZIKGZFLWFGA
|
8.9 | IC50 | 3 | — | |
YTKGKCKBCJZBIX
|
8.9 | IC50 | 4 | — | |
ZKGCNKVDPWEGNL
|
8.9 | IC50 | 3 | — | |
HAVKADYFCFXNIM
|
8.9 | IC50 | 4 | — |