Target Details
| UniProt AC | P06756 |
|---|---|
| Gene Symbol | ITGAV |
| Protein Name | Integrin alpha-V |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01839 (FG-GAP) PF08441 (Integrin_A_Ig_1) PF20805 (Integrin_A_Ig_2) PF20806 (Integrin_A_Ig_3) PF00357 (Integrin_alpha) |
Summary
- Multi-target molecules 1,632
- Clinical molecules 0
- Avg pChEMBL 7.69
KEGG Pathways (20)
- Arrhythmogenic right ventricular cardiomyopathy
- Cell adhesion molecule (CAM) interaction
- Cytoskeleton in muscle cells
- Dilated cardiomyopathy
- ECM-receptor interaction
- Efferocytosis
- Fluid shear stress and atherosclerosis
- Focal adhesion
- Hormone signaling
- Human cytomegalovirus infection
- Human papillomavirus infection
- Hypertrophic cardiomyopathy
- Integrin signaling
- PI3K-Akt signaling pathway
- Pathways in cancer
- Phagosome
- Proteoglycans in cancer
- Regulation of actin cytoskeleton
- Small cell lung cancer
- Thyroid hormone signaling pathway
Associated Diseases (1)
Active Molecules (1,632)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GTSHXMCHGDUGRQ
|
9.2 | IC50 | 4 | — | |
SXIKNOJEFQXCPA
|
9.2 | IC50 | 4 | — | |
XIHAPPZUKXNKFE
|
9.2 | IC50 | 2 | — | |
DLJDTWYGOQOTKA
|
9.2 | IC50 | 3 | — | |
FMXCDFVBSWABHQ
|
9.2 | IC50 | 3 | — | |
FSJCFVNPVGEGOY
|
9.2 | IC50 | 2 | — | |
NOWFLJYSWCXTKI
|
9.2 | IC50 | 2 | — | |
NEEFZJDFXACOOY
|
9.2 | IC50 | 4 | — | |
OKEKRFLAQTYOCR
|
9.2 | IC50 | 3 | — | |
PRTDUHZCDXSBIZ
|
9.2 | IC50 | 5 | — | |
SMMNOJYHMMCWQP
|
9.2 | IC50 | 5 | — | |
SQIDFFKYMURYAR
|
9.2 | IC50 | 2 | — | |
YYMWWKGGQOZSCP
|
9.2 | IC50 | 2 | — | |
BBIYGWDMRXFPEQ
|
9.2 | IC50 | 3 | — | |
DKCBOEVMYBPSHB
|
9.2 | Ki | 2 | — | |
DRZSFOQHHTVBQV
|
9.2 | Ki | 2 | — | |
HUIVUZCGJQLTSS
|
9.2 | IC50 | 3 | — | |
HWQHXIKXIJDPTP
|
9.2 | IC50 | 2 | — | |
KZUKILQARHOBHB
|
9.2 | IC50 | 2 | — | |
LIFIBSDQAZPDID
|
9.2 | IC50 | 4 | — | |
NXFFLBNDPLJURV
|
9.2 | IC50 | 2 | — | |
OHKIVHLQMSGSHE
|
9.2 | IC50 | 2 | — | |
OSNKDBJRGIQKQV
|
9.2 | IC50 | 3 | — | |
PUNZTUWXCLUSNO
|
9.2 | IC50 | 2 | — | |
UCBYYQWMMNUSGH
|
9.2 | IC50 | 8 | — | |
XRXSSPOFDFFALK
|
9.2 | IC50 | 8 | — | |
ZIYZOTDZIZBOGY
|
9.1 | IC50 | 2 | — | |
CKABJNNBXOFZHJ
|
9.1 | IC50 | 2 | — | |
LWHWQLNSWIQIMG
|
9.1 | IC50 | 4 | — | |
XOCAITJQZBYGFQ
|
9.1 | IC50 | 5 | — | |
CKSXICJFAQGSNU
|
9.1 | IC50 | 2 | — | |
GSUDEEPNSDSFMO
|
9.1 | IC50 | 2 | — | |
HVLKUEZLWREEFF
|
9.1 | IC50 | 2 | — | |
ISFSENBRVGRPMH
|
9.1 | IC50 | 2 | — | |
NXLUFIUFDMMQQF
|
9.1 | IC50 | 3 | — | |
PTLBVOXYOSUBEO
|
9.1 | IC50 | 2 | — | |
SDUQEHZORCVRMT
|
9.1 | IC50 | 2 | — | |
VSGFRHHVICROBS
|
9.1 | IC50 | 2 | — | |
WVVNTARUPZRDCO
|
9.1 | IC50 | 3 | — | |
ZEDVVTNZWFMRKR
|
9.1 | IC50 | 3 | — | |
ZMKLPAJURKFWIQ
|
9.1 | IC50 | 5 | — | |
FIEWTBHPTPMJPY
|
9.1 | IC50 | 2 | — | |
SLTMEZLQPRTTBL
|
9.1 | IC50 | 3 | — | |
XAHWDFRDQNVXQX
|
9.1 | IC50 | 2 | — | |
AIBKMZWFGWJRQW
|
9.1 | IC50 | 3 | — | |
BOPPVVPCLIACBR
|
9.1 | IC50 | 2 | — | |
BPFSDEAWEWNYMO
|
9.1 | IC50 | 2 | — | |
HSACVEKFGJAKFH
|
9.1 | IC50 | 3 | — | |
VTZMVMKHYIBVPC
|
9.1 | IC50 | 3 | — | |
VWXQFGQQZYTQPI
|
9.1 | IC50 | 2 | — |