Target Details
| UniProt AC | P06756 |
|---|---|
| Gene Symbol | ITGAV |
| Protein Name | Integrin alpha-V |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01839 (FG-GAP) PF08441 (Integrin_A_Ig_1) PF20805 (Integrin_A_Ig_2) PF20806 (Integrin_A_Ig_3) PF00357 (Integrin_alpha) |
Summary
- Multi-target molecules 1,632
- Clinical molecules 0
- Avg pChEMBL 7.69
KEGG Pathways (20)
- Arrhythmogenic right ventricular cardiomyopathy
- Cell adhesion molecule (CAM) interaction
- Cytoskeleton in muscle cells
- Dilated cardiomyopathy
- ECM-receptor interaction
- Efferocytosis
- Fluid shear stress and atherosclerosis
- Focal adhesion
- Hormone signaling
- Human cytomegalovirus infection
- Human papillomavirus infection
- Hypertrophic cardiomyopathy
- Integrin signaling
- PI3K-Akt signaling pathway
- Pathways in cancer
- Phagosome
- Proteoglycans in cancer
- Regulation of actin cytoskeleton
- Small cell lung cancer
- Thyroid hormone signaling pathway
Associated Diseases (1)
Active Molecules (1,632)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BWAUVRFZNDRMLY
|
9.4 | IC50 | 8 | — | |
GDEQKRGKHZOXGD
|
9.4 | IC50 | 8 | — | |
MFCABRSSOZYCRL
|
9.4 | IC50 | 8 | — | |
RIXFBZVXQWVSQN
|
9.4 | IC50 | 2 | — | |
RTYLRDWEJUNBLU
|
9.4 | IC50 | 8 | — | |
USYHJFFPGOCQTN
|
9.4 | IC50 | 2 | — | |
VQFZVRMJIHFIPZ
|
9.4 | IC50 | 2 | — | |
WBIUNXVKIMTWNG
|
9.4 | IC50 | 2 | — | |
WRJHOBGONWLLMD
|
9.4 | IC50 | 2 | — | |
YPAMHQMVIMQKOR
|
9.4 | IC50 | 8 | — | |
YSUOCWJZGZEUQT
|
9.4 | IC50 | 2 | — | |
KSSPHFGIOASRDE
|
9.4 | IC50 | 2 | — | |
RIRSYRXZEYNCLO
|
9.4 | IC50 | 4 | — | |
FSKOAKSLUAJDDL
|
9.4 | IC50 | 3 | — | |
MSJFRVFQMDZEFH
|
9.3 | IC50 | 3 | — | |
QGOXLUXYLLZODC
|
9.3 | IC50 | 3 | — | |
XRFHJLOFJUFLJB
|
9.3 | IC50 | 2 | — | |
WUEFOEAIDROUBP
|
9.3 | IC50 | 3 | — | |
KBRCQTXEFPMTDE
|
9.3 | IC50 | 2 | — | |
RXTBIRIYBNVLMP
|
9.3 | IC50 | 2 | — | |
YUYFHARZOUACDE
|
9.3 | IC50 | 3 | — | |
CJRDXSVCUSRJDR
|
9.3 | IC50 | 8 | — | |
CNSDHPHNXQALLW
|
9.3 | IC50 | 2 | — | |
CPOXHOJHCZSECN
|
9.3 | Ki | 2 | — | |
JZHPHPOLAVKTRC
|
9.3 | IC50 | 2 | — | |
JZHPHPOLAVKTRC
|
9.3 | IC50 | 2 | — | |
MLRJOXSFEYKLLF
|
9.3 | Ki | 4 | — | |
OBOJFQICXTYCRY
|
9.3 | IC50 | 8 | — | |
OLCXJKREUBWULJ
|
9.3 | IC50 | 2 | — | |
OMISPTOHCAHRQR
|
9.3 | IC50 | 3 | — | |
PRILHZGEUSLPLF
|
9.3 | IC50 | 2 | — | |
QTBFGJFGHGTDRF
|
9.3 | IC50 | 8 | — | |
WWUJBWRZVJNABY
|
9.3 | IC50 | 3 | — | |
YRCDKPLXZYFHKS
|
9.3 | IC50 | 2 | — | |
PWDSDBVBKCIRHN
|
9.3 | IC50 | 4 | — | |
SWSSTJOKJXGDQH
|
9.3 | IC50 | 3 | — | |
SXIKNOJEFQXCPA
|
9.3 | IC50 | 4 | — | |
TZEHAFMMPSPZTD
|
9.3 | IC50 | 2 | — | |
RQMPMSIEFFKLGD
|
9.3 | IC50 | 3 | — | |
AMLYAMJWYAIXIA
|
9.2 | IC50 | 3 | — | |
LHGHYRBRMNOGPF
|
9.2 | IC50 | 2 | — | |
INPJXWNSGITHFI
|
9.2 | IC50 | 2 | — | |
ABVOSXLHVDENOA
|
9.2 | IC50 | 2 | — | |
BQYBIJDRTDZCAJ
|
9.2 | IC50 | 8 | — | |
HIKDGFUZLZJZCB
|
9.2 | IC50 | 8 | — | |
MMTMLJZCVSAZFC
|
9.2 | IC50 | 3 | — | |
OJTBKASAMAYZRX
|
9.2 | IC50 | 2 | — | |
OTRLSMNUUKTGCC
|
9.2 | IC50 | 3 | — | |
WGHOQSIOKMBZIJ
|
9.2 | IC50 | 3 | — | |
WROMAHOUFMMNHT
|
9.2 | IC50 | 2 | — |