Target Details
| UniProt AC | P06756 |
|---|---|
| Gene Symbol | ITGAV |
| Protein Name | Integrin alpha-V |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01839 (FG-GAP) PF08441 (Integrin_A_Ig_1) PF20805 (Integrin_A_Ig_2) PF20806 (Integrin_A_Ig_3) PF00357 (Integrin_alpha) |
Summary
- Multi-target molecules 1,632
- Clinical molecules 0
- Avg pChEMBL 7.69
KEGG Pathways (20)
- Arrhythmogenic right ventricular cardiomyopathy
- Cell adhesion molecule (CAM) interaction
- Cytoskeleton in muscle cells
- Dilated cardiomyopathy
- ECM-receptor interaction
- Efferocytosis
- Fluid shear stress and atherosclerosis
- Focal adhesion
- Hormone signaling
- Human cytomegalovirus infection
- Human papillomavirus infection
- Hypertrophic cardiomyopathy
- Integrin signaling
- PI3K-Akt signaling pathway
- Pathways in cancer
- Phagosome
- Proteoglycans in cancer
- Regulation of actin cytoskeleton
- Small cell lung cancer
- Thyroid hormone signaling pathway
Associated Diseases (1)
Active Molecules (1,632)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YWGKJZDMSJRNNY
|
9.7 | IC50 | 2 | — | |
GASMFAZDFTXBTB
|
9.6 | IC50 | 4 | — | |
LPDONRQJLDDGHH
|
9.6 | IC50 | 2 | — | |
LPDONRQJLDDGHH
|
9.6 | IC50 | 2 | — | |
BCDVKMOAMMODMM
|
9.6 | IC50 | 4 | — | |
AGSAJJWUDWLFCF
|
9.6 | IC50 | 2 | — | |
ILIAIJBQDWEDLF
|
9.6 | IC50 | 2 | — | |
NNOYJUNBGWLDGM
|
9.6 | IC50 | 3 | — | |
ODFWEQUMDQJBJZ
|
9.6 | IC50 | 2 | — | |
TXDUNPFVQQSUTP
|
9.6 | IC50 | 3 | — | |
SXUVGBBNFRFEFN
|
9.6 | IC50 | 2 | — | |
ZVPFRHUDZYLXOW
|
9.6 | IC50 | 2 | — | |
YTPVKTLAFFSGBR
|
9.6 | IC50 | 3 | — | |
HTULCSBVNFKESE
|
9.5 | IC50 | 2 | — | |
ITHSUPJAQZZIJZ
|
9.5 | IC50 | 2 | — | |
BFQFATKIIYMFLO
|
9.5 | IC50 | 2 | — | |
ITJUXSPTLRWMDJ
|
9.5 | IC50 | 2 | — | |
IZIPDPPLSSBGTL
|
9.5 | IC50 | 2 | — | |
JSXRQHGDURETKY
|
9.5 | IC50 | 2 | — | |
JXVVEFIKDDVLOS
|
9.5 | IC50 | 8 | — | |
KAUTWCRUPICGMP
|
9.5 | IC50 | 2 | — | |
KJTGODHDGKRMDH
|
9.5 | IC50 | 2 | — | |
LTSYOWOYZKAEHL
|
9.5 | IC50 | 2 | — | |
MKIOVSFGHYIVDB
|
9.5 | IC50 | 3 | — | |
MPAIDFBWWZPGEV
|
9.5 | IC50 | 2 | — | |
OTGFOVKWHHNDHF
|
9.5 | IC50 | 3 | — | |
VSAKVGBQGGPIJH
|
9.5 | IC50 | 2 | — | |
VYPOWHUOZSVSQJ
|
9.5 | IC50 | 2 | — | |
XGZVUDGXURHWEC
|
9.5 | IC50 | 3 | — | |
ZFIVYUYYCMBCTR
|
9.5 | IC50 | 2 | — | |
FJUFYEBFJYPEFS
|
9.5 | IC50 | 2 | — | |
JZTSYGNOFKHTHM
|
9.5 | IC50 | 3 | — | |
NBFYQDLZBZGXPB
|
9.5 | IC50 | 4 | — | |
VTJZZOUBHILYBS
|
9.5 | IC50 | 4 | — | |
HLXLTYRHIUOBBV
|
9.5 | IC50 | 2 | — | |
OAUKXLIBIFPGBT
|
9.5 | IC50 | 2 | — | |
PDPLWPUOLLTXCX
|
9.5 | IC50 | 2 | — | |
PTCMVGOQRMWOTP
|
9.5 | IC50 | 4 | — | |
BDFMVIGZRRIXCL
|
9.5 | IC50 | 5 | — | |
LGMXGJOVGIKKKC
|
9.5 | IC50 | 4 | — | |
FDEYYGVHDVBTNW
|
9.5 | IC50 | 4 | — | |
RGDXUISAOHECQH
|
9.5 | IC50 | 2 | — | |
VJTDBRLHPYYFBZ
|
9.5 | IC50 | 2 | — | |
VJTDBRLHPYYFBZ
|
9.5 | IC50 | 2 | — | |
ZBPWDXMZTZUZSY
|
9.5 | IC50 | 2 | — | |
QPZOEIQRDYCGMD
|
9.4 | IC50 | 5 | — | |
FVYSXFUNKAIEAQ
|
9.4 | IC50 | 3 | — | |
ICALNGJCZQBZDD
|
9.4 | IC50 | 2 | — | |
MGVKLGFDHDXKFL
|
9.4 | IC50 | 2 | — | |
YWGKJZDMSJRNNY
|
9.4 | IC50 | 2 | — |