Target Details
| UniProt AC | P06756 |
|---|---|
| Gene Symbol | ITGAV |
| Protein Name | Integrin alpha-V |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01839 (FG-GAP) PF08441 (Integrin_A_Ig_1) PF20805 (Integrin_A_Ig_2) PF20806 (Integrin_A_Ig_3) PF00357 (Integrin_alpha) |
Summary
- Multi-target molecules 1,632
- Clinical molecules 0
- Avg pChEMBL 7.69
KEGG Pathways (20)
- Arrhythmogenic right ventricular cardiomyopathy
- Cell adhesion molecule (CAM) interaction
- Cytoskeleton in muscle cells
- Dilated cardiomyopathy
- ECM-receptor interaction
- Efferocytosis
- Fluid shear stress and atherosclerosis
- Focal adhesion
- Hormone signaling
- Human cytomegalovirus infection
- Human papillomavirus infection
- Hypertrophic cardiomyopathy
- Integrin signaling
- PI3K-Akt signaling pathway
- Pathways in cancer
- Phagosome
- Proteoglycans in cancer
- Regulation of actin cytoskeleton
- Small cell lung cancer
- Thyroid hormone signaling pathway
Associated Diseases (1)
Active Molecules (1,632)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BCRUFWDIRARGLM
|
8.4 | IC50 | 2 | — | |
HOJQNBKLKYCOIL
|
8.3 | IC50 | 6 | — | |
LNCJYAZJFUDHSC
|
8.3 | IC50 | 2 | — | |
RBJQMIIPTLTYFP
|
8.3 | IC50 | 8 | — | |
VCYXSHVQNGNXQO
|
8.3 | IC50 | 3 | — | |
FHIDQJNETPMUKT
|
8.3 | IC50 | 2 | — | |
FPHTZWODHSAREX
|
8.3 | IC50 | 3 | — | |
KNVMGBKMZYKHLR
|
8.3 | IC50 | 5 | — | |
YKFFKLLBAOJGON
|
8.3 | IC50 | 2 | — | |
FQMVMULCHDNQMG
|
8.3 | IC50 | 3 | — | |
ILKRHUYCJMCBRQ
|
8.3 | IC50 | 8 | — | |
MLEGBHJXMACOKD
|
8.3 | IC50 | 2 | — | |
POHCCPZJODTAKF
|
8.3 | IC50 | 3 | — | |
UICIXEUWXCRGCE
|
8.3 | IC50 | 3 | — | |
BOGKCCITBZWXSX
|
8.3 | Ki | 2 | — | |
BWOKYFQNZCEABS
|
8.3 | IC50 | 3 | — | |
CFCPTSHVAOVLJR
|
8.3 | IC50 | 3 | — | |
CYKGGZKCPJYWKZ
|
8.3 | IC50 | 3 | — | |
NSLLXYFCBUUZFG
|
8.3 | IC50 | 2 | — | |
QFEXPKRHMFCDGL
|
8.3 | IC50 | 2 | — | |
QFUAOXPDMSSGEO
|
8.3 | IC50 | 3 | — | |
WSAQSLNUSGZKRH
|
8.3 | IC50 | 3 | — | |
XKXMEMPIHRKAQX
|
8.3 | IC50 | 5 | — | |
ZDUUJAZQZQAJEO
|
8.3 | IC50 | 6 | — | |
OSFFDUZCJDKYFG
|
8.3 | Ki | 2 | — | |
VDXWNRXEYNGPST
|
8.3 | IC50 | 4 | — | |
IGRZOKIVRZOBLQ
|
8.3 | IC50 | 4 | — | |
MLCFOKYQRPBDTP
|
8.3 | IC50 | 3 | — | |
DPFLAGDMGNKRSD
|
8.3 | IC50 | 4 | — | |
HHDFZZZPZFQCII
|
8.3 | IC50 | 2 | — | |
KLOOZQSECCCWDS
|
8.3 | IC50 | 3 | — | |
LZXHGKPQGMADDV
|
8.2 | IC50 | 3 | — | |
WMAYUSHYHMSHFY
|
8.2 | IC50 | 6 | — | |
HARYXLBGCPNWSN
|
8.2 | IC50 | 3 | — | |
SGWKNXDQAJXYHU
|
8.2 | IC50 | 3 | — | |
UBCYLCJDLQOXGZ
|
8.2 | IC50 | 2 | — | |
VJGKWMZBCANVTK
|
8.2 | IC50 | 2 | — | |
ZWPCJINLOLYZBQ
|
8.2 | IC50 | 4 | — | |
YBFKWPJDYFKQMV
|
8.2 | IC50 | 2 | — | |
CBZJLJSPZAYODX
|
8.2 | IC50 | 2 | — | |
GYTCJTUMBCVRAA
|
8.2 | IC50 | 2 | — | |
LLJAASOTTFNJHX
|
8.2 | IC50 | 2 | — | |
ORYVBGZLSVZQOS
|
8.2 | IC50 | 3 | — | |
UBKWNMZGLKKYKI
|
8.2 | IC50 | 2 | — | |
XLYGKRZQPDXMEM
|
8.2 | IC50 | 3 | — | |
YQIZMAFWDNCDLY
|
8.2 | IC50 | 3 | — | |
GPNNVIVBATZBGX
|
8.2 | IC50 | 2 | — | |
KCRVIBMJQPGDDH
|
8.2 | IC50 | 3 | — | |
SRCAHUCFNDYNBV
|
8.2 | IC50 | 2 | — | |
IUYOOUVOXKZZKL
|
8.2 | IC50 | 2 | — |