Target Details
| UniProt AC | P06756 |
|---|---|
| Gene Symbol | ITGAV |
| Protein Name | Integrin alpha-V |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01839 (FG-GAP) PF08441 (Integrin_A_Ig_1) PF20805 (Integrin_A_Ig_2) PF20806 (Integrin_A_Ig_3) PF00357 (Integrin_alpha) |
Summary
- Multi-target molecules 1,632
- Clinical molecules 0
- Avg pChEMBL 7.69
KEGG Pathways (20)
- Arrhythmogenic right ventricular cardiomyopathy
- Cell adhesion molecule (CAM) interaction
- Cytoskeleton in muscle cells
- Dilated cardiomyopathy
- ECM-receptor interaction
- Efferocytosis
- Fluid shear stress and atherosclerosis
- Focal adhesion
- Hormone signaling
- Human cytomegalovirus infection
- Human papillomavirus infection
- Hypertrophic cardiomyopathy
- Integrin signaling
- PI3K-Akt signaling pathway
- Pathways in cancer
- Phagosome
- Proteoglycans in cancer
- Regulation of actin cytoskeleton
- Small cell lung cancer
- Thyroid hormone signaling pathway
Associated Diseases (1)
Active Molecules (1,632)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CUGPAWBXPURXLJ
|
10.7 | IC50 | 2 | — | |
OQLMEWQXUAYOHO
|
10.5 | IC50 | 2 | — | |
LEEJTINVSSJMDG
|
10.4 | IC50 | 2 | — | |
LEEJTINVSSJMDG
|
10.4 | IC50 | 3 | — | |
UJAJKKVATBUTAU
|
10.4 | IC50 | 2 | — | |
KBFHSTNZWSMOOM
|
10.3 | IC50 | 2 | — | |
JGRADSKQVRSSDT
|
10.2 | IC50 | 2 | — | |
HAMNCHGAVJSNBY
|
10.2 | IC50 | 3 | — | |
DMDDFJFCCZFCKL
|
10.2 | IC50 | 2 | — | |
VGNHZMRKYBWPOO
|
10.2 | IC50 | 3 | — | |
NCUDSCWWOMSIFO
|
10.1 | IC50 | 2 | — | |
NJDBZBVQIMZWPP
|
10.1 | IC50 | 2 | — | |
CFHPIPZTEAYFIR
|
10.1 | IC50 | 2 | — | |
BGDLLUWAZFBMGD
|
10.0 | IC50 | 2 | — | |
DRZSFOQHHTVBQV
|
10.0 | Ki | 2 | — | |
FWYCIUUIVROTKO
|
10.0 | Ki | 2 | — | |
LRJXQAWFNQBGLZ
|
10.0 | IC50 | 5 | — | |
QFKUDHXQVSUGKR
|
10.0 | IC50 | 2 | — | |
UFJUFUWNIIBKKK
|
10.0 | IC50 | 2 | — | |
WURWJPCCHUZQHY
|
10.0 | IC50 | 2 | — | |
HTJMDVDUBVVYKB
|
10.0 | IC50 | 2 | — | |
KKEMGRLKOQAUBU
|
10.0 | IC50 | 2 | — | |
KSQUEZUEYFZRQY
|
10.0 | IC50 | 2 | — | |
UHBUZZJODALKHF
|
10.0 | IC50 | 3 | — | |
YXLLXCYQWYHDOI
|
10.0 | IC50 | 2 | — | |
AJZHUKFTTKIGAR
|
9.9 | IC50 | 3 | — | |
ILIAIJBQDWEDLF
|
9.9 | IC50 | 2 | — | |
DOCHXGULTZHKAZ
|
9.8 | IC50 | 4 | — | |
FXUNUOYKSJCHND
|
9.8 | IC50 | 3 | — | |
CFXVNDHCOWFOSR
|
9.8 | IC50 | 3 | — | |
DOULIFPELQSYIR
|
9.8 | IC50 | 2 | — | |
OVLTXZRGJNTGSK
|
9.8 | IC50 | 2 | — | |
YJTFZPUDXPSWOJ
|
9.8 | IC50 | 2 | — | |
YNVYQJGEOYPMMJ
|
9.8 | IC50 | 2 | — | |
OXNNEMDLTGEMOR
|
9.8 | Ki | 2 | — | |
YYKYFRLZWKUEIZ
|
9.7 | IC50 | 3 | — | |
AXZHUMWCDZWWOZ
|
9.7 | IC50 | 2 | — | |
BERNMEVEBUTYSS
|
9.7 | IC50 | 2 | — | |
BERNMEVEBUTYSS
|
9.7 | IC50 | 2 | — | |
BZQOJXDBIMQBSY
|
9.7 | IC50 | 2 | — | |
JDAGFAQRQYOYIN
|
9.7 | IC50 | 2 | — | |
KNSPFVAZTITFFW
|
9.7 | IC50 | 3 | — | |
KQJRVLULCJERGE
|
9.7 | IC50 | 2 | — | |
NOWXQWGDOHATCX
|
9.7 | IC50 | 2 | — | |
SHRSEUHJTZQLRO
|
9.7 | IC50 | 8 | — | |
URFXLBUFCLGJGX
|
9.7 | IC50 | 2 | — | |
ZATLFCSNKBMFBH
|
9.7 | IC50 | 2 | — | |
VVIGVXDFMPIPRO
|
9.7 | IC50 | 4 | — | |
XBHBFRSVZRSVIA
|
9.7 | IC50 | 2 | — | |
AEZOMALWKBTDJK
|
9.7 | IC50 | 3 | — |