Target Details
| UniProt AC | P06730 |
|---|---|
| Gene Symbol | EIF4E |
| Protein Name | Eukaryotic translation initiation factor 4E |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01652 (IF4E) |
Summary
- Multi-target molecules 46
- Clinical molecules 0
- Avg pChEMBL 7.21
KEGG Pathways (6)
Associated Diseases (1)
Active Molecules (46)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QFJCIRLUMZQUOT
|
9.3 | Kd | 9 | — | |
NQKUBPWGXDRNCR
|
8.5 | IC50 | 3 | — | |
YFVARPBUZODTDL
|
8.4 | IC50 | 2 | — | |
HKTBYUWLRDZAJK
|
8.3 | IC50 | 5 | — | |
BTVOPBCDBRHMPF
|
8.1 | IC50 | 3 | — | |
CYFVVHXJLAKHJY
|
8.1 | IC50 | 3 | — | |
REWHONSUJOGBSP
|
8.0 | IC50 | 2 | — | |
LVSWSCZOVNFBCZ
|
7.8 | IC50 | 3 | — | |
GQPLXSNGJYAHSH
|
7.7 | IC50 | 3 | — | |
HIIXSKLGSBCTAH
|
7.7 | IC50 | 3 | — | |
WSLNKDCNHNOGHL
|
7.7 | IC50 | 3 | — | |
ZUBOOCCOALVOHE
|
7.7 | Kd | 2 | — | |
DPFZKILBVWKIDP
|
7.6 | IC50 | 3 | — | |
KXZLWAAQYGMLJX
|
7.6 | IC50 | 3 | — | |
CXNIDEGZWPEOCF
|
7.5 | IC50 | 3 | — | |
FOQNSWUDBARUFL
|
7.5 | IC50 | 3 | — | |
XZUIPTFXIKGMGA
|
7.5 | IC50 | 3 | — | |
CLIORPUQKOJRDE
|
7.4 | IC50 | 3 | — | |
QUVIEDJGNUFDDH
|
7.4 | IC50 | 3 | — | |
BCANLOWELFOMRO
|
7.3 | Kd | 2 | — | |
KVGHGVHKZQAQLD
|
7.3 | IC50 | 3 | — | |
POSZZZFFLNLQCL
|
7.3 | IC50 | 3 | — | |
NFYSHFWLDDXPKM
|
7.2 | IC50 | 3 | — | |
FPQBGLUWBCLXFG
|
7.1 | IC50 | 3 | — | |
GXOJOLCVOSVXPG
|
7.0 | IC50 | 3 | — | |
HDKZJMGFRSXWSJ
|
7.0 | IC50 | 3 | — | |
AJGPWESAFONVCG
|
7.0 | IC50 | 3 | — | |
ZRIDICSQDPQVEH
|
6.9 | IC50 | 3 | — | |
MWXOTOIFWCYXRK
|
6.9 | IC50 | 3 | — | |
JMOODDNVNBVCOJ
|
6.9 | IC50 | 3 | — | |
GXUYZVYTXZYDQM
|
6.8 | IC50 | 3 | — | |
FXMBSEOFWALADX
|
6.7 | IC50 | 3 | — | |
UUQZSFPVUKCRKO
|
6.7 | IC50 | 3 | — | |
JIBSLIWLWMKJGN
|
6.7 | IC50 | 3 | — | |
VVQCEELTIIOFHE
|
6.7 | IC50 | 2 | — | |
BFUCQUQBTJOBTA
|
6.6 | IC50 | 3 | — | |
GLKYGVDXWJUOFW
|
6.6 | IC50 | 3 | — | |
CGMQSJXTBXHOTH
|
6.5 | IC50 | 9 | — | |
VQBHHVIUAXNAOC
|
6.5 | IC50 | 3 | — | |
LXNUFRAUJVQQOV
|
6.4 | IC50 | 3 | — | |
MWKSRKSEWLRPBL
|
6.4 | Kd | 1075 | — | |
PYHRNXAACBOPCP
|
6.4 | IC50 | 3 | — | |
MIVZVCNGBMCBAA
|
6.4 | IC50 | 3 | — | |
FWRFPHJSGLYXTD
|
6.3 | IC50 | 3 | — | |
WCADNSJQHAGKBX
|
6.2 | IC50 | 3 | — | |
WCADNSJQHAGKBX
|
6.1 | IC50 | 3 | — |